Lecithinised microemulsions for topical delivery of tretinoin

International Journal of Drug Development and Research

Volumn 2, Issue 4, 2010, Pages 711-719

  Khanna, Surabhi ^a   Katare, O P ^b   Drabu, Sushma ^a  

^a GURU GOBIND SINGH INDRAPRASTHA UNIVERSITY   (India)

^b PANJAB UNIVERSITY   (India)

Author keywords

Acne; Lecithin; Microemulsions; Topical delivery; Tretinoin

Indexed keywords

ALCOHOL; MYRISTIC ACID ISOPROPYL ESTER; PHOSPHATE; PHOSPHATIDYLCHOLINE; POLYSORBATE 80; RETINOIC ACID;

ANIMAL TISSUE; ARTICLE; DRUG DELIVERY SYSTEM; DRUG FORMULATION; DRUG SOLUBILITY; GEL; IN VITRO STUDY; MICROEMULSION; MOUSE; NONHUMAN; PH; SKIN PERMEABILITY; TOPICAL DRUG ADMINISTRATION;

EID: 79952434400     PISSN: None     EISSN: 09759344     Source Type: Journal    
DOI: None     Document Type: Article

References (34)

1. Kantaria, S., Rees, G.D., Lawrence M.J., Formulation of electrically conducting microemulsion based organogels, Int. J. Pharm., 2003, 250, 65-83 (Pubitemid 35447938)
2. Tenjarla, S., Microemulsions : an overview and pharmaceutical applications, Crit. Rev. Ther. Carr. Sys., 1999, 16, 461-521
3. Constantinides, P.P., Lipid microemulsions for improving drug dissolution and oral absorption: physical and biopharmaceutical aspects, Pharm. Res., 1995, 12, 1561-1572 (Pubitemid 26005509)
4. Gasco M.R., Microemulsions in the pharmaceutical field: perspectives and applications in; Industrial Applications of Microemulsions, Marcel Dekker Inc., New York, 1997, 97-122
5. Gasco M., Gallarate M., Trotta M., Gremmo E., Chiappero O., Microemulsions as topical delivery vehicles : ocular administeration of timolol, J. Pharm. Biomed. Anal., 1989, 7(4), 433-439 (Pubitemid 19156054)
6. Delgado-Charro M.B., Iglesias Vilas G, Blanco-Mendez J., Lopez Quintela M.A., Marty J.P., Guy R.H., Delivery of a hydrophilic solute through the skin from novel microemulsion systems, Eur. J. Pharm. Biopharm. 43(1997), 37-42. (Pubitemid 28298808)
7. Beer, W.E., Smith, N.P., Hyperkeratotic porokeratosis with psoriasis-response to an aromatic retinoid, Clin. Exp. Dermatol., 1984, 9, 509-513. (Pubitemid 14037172)
8. Orfanos, C.E., Ehlert, R., Gollnick, H., The Retinoids, A review of their clinical pharmacology and therapeutic use, Drugs, 1987, 34, 459-503. (Pubitemid 17143097)
9. Ong, E.S., Dyek, J.A., Nuclear receptor that identifies a novel retinoic acid pathway, Nature, 1990, 345, 224-229.
10. Elder, J.T., Astrom, A., Differential regulation of retinoic acid receptors and binding proteins in human skin, J. Invest. Dermatol., 1992, 98, 673-679.
11. Brime B., Moreno M., Frutos G., Ballesteros P., Frutos P., Amphotericin B in oil- water lecithin based microemulsions : Formulation and toxicity evaluation, J. Pharm. Scs., 2002, 91(4), 1178-1185 (Pubitemid 34640942)
12. Baroli B., Quintela M.A., Chaero M. B., Fadda A. M., Mandez J. B., Microemulsions for topical delivery of 8-Methoxsalen, Int. J. Pharm., 2000, 69, 209-218
13. Benita S. and Levy M. Y., Drug release from submicronised o/w emulsion : A new in vitro kinetic evaluation method, Int. J. Pharm., 1990, 66, 29-37
14. Benita S., Levy M. Y., Submicron emulsions as colloidal drug carriers for intravenous administration : comprehensive physicochemical characterization, J. Pharm. Scs., 1993, 82(11), 1069-1079 (Pubitemid 24004434)
15. Bentley B., Vitoria M., Kedor E., Vianna F., Collett J., The effect of urea and lecithin on the in vitro permeation of hydrocortisone acetate through skin from hairless mouse, Int. J. Pharm., 1997, 146, 255-262 (Pubitemid 27110796)
16. Bhargava, H.N., Narurkar, A., Leils, L.M., Using microemulsions for drug delivery, Pharm. Technol., 1987, 11, 46-54
17. Bolzinger, M.A., Carduner, T.C., Poelman, M.C., Bicontinuous sucrose ester microemulsion : a new vehicle for topical delivery of niflumic acid, Int. J. Pharm., 1998, 176, 39-45 (Pubitemid 28544970)
18. Brime B., Moreno M., Frutos G., Ballesteros P., Frutos P., Amphotericin B in oil- water lecithin based microemulsions : Formulation and toxicity evaluation, J. Pharm. Scs., 2002, 91(4), 1178-1185 (Pubitemid 34640942)
19. Brisaert M., Gabriels M., Mathijs V., Liposomes with tretinoin: a physical and chemical evaluation, Int. J. Pharm., 2001, 26, 909-917 (Pubitemid 32971703)
20. Chen, S.H., Lin, T.l., In: Surfactants in solutions, 1986, Plenum Press, Vol 6, New York, 1315-1330
21. Cirkel, P.A., Ploeg, J.P.M., Koper, G.J.M., Branching and percolation in lecithin wormlike micelles studied by dielectric spectroscopy, Phys. Rev. 1998, E57, 6875-6883 (Pubitemid 128625094)
22. Constantinides P. P., Scalarat J., Formulation and physical characterization of water in oil microemulsions containing long versus medium - chain triglycerides, Int. J. Pharm.,1997, 158, 57-68 (Pubitemid 27504474)
23. Constantinides P.P., Lipid microemulsions for improving drug dissolution and oral absorption: Physical and biopharmaceutical aspects, Pharm. Res., 1995, 12(11), 1561
24. Constantinides, P.P., Scalart, J.P., Formulation and Physical characterization of w/o microemulsions containing long versus medium chain length glycerides, Int. J. Pharm., 1997, 158, 57-68 (Pubitemid 27504474)
25. Constantinides, P.P., Yiv, S.H., Particle size determination of phase inverted w/o microemulsions under different dilution and storage conditions, Int. J. Pharm., 1995, 115, 225-234
26. Friberg, S.E., Venable, R.L., Microemulsions In: Encyclopedia of emulsion technology, (Bechner P ed.), Marcel Dekker Inc., New York, 1983, Vol 1, 287-336
27. Gallarate, M., Gasco, M.R., Trotta, M., Chetoni, P., Saettone, M.F., Preparation and evaluation in vitro of solutions and o/w microemulsions containing levobunolol as ion pair, Int. J. Pharm., 1993, 100, 219-225 (Pubitemid 23316335)
28. Gilis J. C. and Goa K. L., Tretinoin: A review of its pharmacodynamic and pharmacokinetic properties and management of acute promyelocytic leukemia, Drugs, 1995, 50, 897-923
29. Kreilgaard, M., Pederson, E.J., Jaroszewski, J. W., NMR characterization and transdermal drug delivery potential of microemulsion systems, J. Cont. Rel., 2000, 69, 421-433
30. Krielgaard M., Influence of microemulsions on cutaneous drug delivery, Adv. Drug Del. Rev., 2002, 54 Suppl 1, S77-S98
31. Krielgaard, M., Dermal Pharmacokinetics of microemulsion formulation determined by in vivo microdialysis, Pharm. Res., 2001, 18 (3), 367
32. Ktistis, G., Effect of polysorbate 80 and sorbitol concentration on the in vitro release of indomethacin from microemulsions, J. Disp. Sci. Technol., 1997, 18, 49-61 (Pubitemid 127718008)
33. Kuneida, H., Solans, C., In: Industrial applications of microemulsions, Marcel Dekker, New York, 1997, 21
34. Vohra S, Lecithinsed microemulsions for topical delivery of tretinoin and methyl salicylate, Panjab University, Chandigarh (2004)