Assessment of milling-induced disorder of two pharmaceutical compounds

Journal of Pharmaceutical Sciences

Volumn 100, Issue 5, 2011, Pages 1793-1804

  Otte, Andrew ^a   Carvajal, M Teresa ^a,b  

^a PURDUE UNIVERSITY   (United States)

^b PURDUE UNIVERSITY   (United States)

Author keywords

Crystal defects; Milling; Solid state; Surface chemistry; Thermal analysis

Indexed keywords

GRISEOFULVIN; KETOCONAZOLE;

ARTICLE; COOLING; CRYOMILLING; CRYSTAL STRUCTURE; CRYSTALLIZATION; DIFFERENTIAL SCANNING CALORIMETRY; ENERGY; GRINDING; HEATING; INVERSE GAS CHROMATOGRAPHY; PARTICLE SIZE; PHASE TRANSITION; SURFACE PROPERTY; TEMPERATURE; X RAY POWDER DIFFRACTION;

EID: 79952218722     PISSN: 00223549     EISSN: 15206017     Source Type: Journal    
DOI: 10.1002/jps.22415     Document Type: Article

References (27)

1. Bisrat M, Nystrom C. 1988. Physicochemical aspects of drug release. viii. The relation between particle size and surface specific dissolution rate in agitated suspensions. Int J Pharm 47:223-231.
2. Feng T, Pinal R, Carvajal MT. 2008. Process induced disorder in crystalline materials: Differentiating defective crystals from the amorphous form of griseofulvin. J Pharm Sci 97:3207-3221.
3. Chamarthy SP, Pinal R. 2008. The nature of crystal disorder in milled pharmaceutical materials. Colloid and Surface A 331:68-75.
4. Grimsey IM, Sunkersett M, Osborn JC, York P, Rowe RC. 1999. Interpretation of the differences in the surface energetics of two optical forms of mannitol by inverse gas chromatography and molecular modeling. Int J Pharm 191:43-50.
5. Price R, Young PM. 2005. On the physical transformations of processed pharmaceutical solids. Micron 36:519-524.
6. Mackin L, Sartnurak S, Thomas I, Moore S. 2002. The impact of low levels of amorphous material <5% on the blending characteristics of a direct compression formulation. Int J Pharm 231:213-226.
7. Adolfsson A, Caramella C, Nystrom C. 1998. The effect of milling and addition of dry binder on the interparticulate bonding mechanisms in sodium chloride tablets. Int J Pharm 160:187-195.
8. Rasenack N, Muller BW. 2002. Dissolution rate enhancement by in situ micronization of poorly water-soluble drugs. Pharm Res 19:1894-1900.
9. Ticehurst M, Rowe R, York P. 1994. Determination of the surface properties of two batches of salbutamol sulphate by inverse gas chromatography. Int J Pharm 111:241-249.
10. Feeley JC, York P, Sumby BS, Dicks H. 1998. Determination of surface properties and flow characteristics of salbutamol sulphate, before and after micronisation. Int J Pharm 172:89-96.
11. Surana R, Randall L, Pyne A, Vemuri NM, Suryanarayanan R. 2003. Determination of glass transition temperature and in situ study of the plasticizing effect of water by inverse gas chromatography. Pharm Res 20:1647-1654.
12. Planinsek O, Zadnik J, Kunaver M, Srcic S, Godec A. 2010. Structural evolution of indomethacin particles upon milling: Time-resolved quantification and localization of disordered structure studied by igc and dsc. J Pharm Sci 99:1968-1981.
13. York P, Ticehurst MD, Osborn JC, Roberts RJ, Rowe RC. 1998. Characterisation of the surface energetics of milled dl-propranolol hydrochloride using inverse gas chromatography and molecular modeling. Int J Pharm 174:179-186.
14. Ohta M, Buckton G. 2004. Determination of the changes in surface energetics of cefditoren pivoxil as a consequence of processing induced disorder and equilibration to different relative humidities. Int J Pharm 269:81-88.
15. Newell H, Buckton G. 2004. Inverse gas chromatography: Investigating whether the technique preferentially probes high energy sites for mixtures of crystalline and amorphous lactose. Pharm Res 21:1440-1444.
16. Heng JYY, Thielmann F, Williams DR. 2006. The effects of milling on the surface properties of form I paracetamol crystals. Pharm Res 23:1918-1927.
17. Ho R, Hinder SJ, Watts JF, Dilworth SE, Williams DR, Heng JYY. 2010. Determination of surface heterogeneity of D-mannitol by sessile drop contact angle and finite concentration inverse gas chromatography. Int J Pharm 387:79-86.
18. Burnett D, Thielmann F, Booth J. 2004. Determining the critical relative humidity for moisture-induced phase transitions. Int J Pharm 287:123-133.
19. Puig CC, Meijer HEH, Michels MAJ, Segeren LH, Vancso GJ. 2004. Characterization of glass transition temperature and surface energy of bituminous binders by inverse gas chromatography. Energy Fuels 18:63-67.
20. Hamieh T J, Schultz J. 2002. New approach to characterise physicochemical properties of solid substrates by inverse gas chromatography at infinite dilution. ii. Study of the transition temperatures of poly(methyl methacrylate) at various tacticities and of poly(methyl methacrylate) adsorbed on alumina and silica. J Chromatogr A. 969:27-36.
21. Schultz J, Lavielle L, Martin C. 1987. The role of the interface in carbon fibre-epoxy composites. J Adhesion 23:45-60.
22. th ed., Weinheim, Germany: VCH.
23. Morup S, Jiang JZ, Bodker F, Horsewell A. 2001. Crystal growth and the steady-state grain size during high-energy ball-milling. Europhys Lett 56:441-446.
24. Hellstern E, Fecht HJ, Fu Z, Johnson WL. 1989. Structural and thermodynamic properties of heavily mechanically deformed Ru and AlRu. J Appl Phys 65:305-310.
25. OweBerg TG, Avis LE. 1970. Exploratory experiments on kinetics of comminution. Powder Tech 4:27-31.
26. Vanden Mooter G, Wuyts M, Blaton N, Busson R, Grobet P, Augustijns P, Kinget R. 2001. Physical stabilisation of amorphous ketoconazole in solid dispersions with polyvinylpyrrolidone k25. Euro J Pharm Sci 12:261-269.
27. Elamin AA, Ahlneck C, Alderborn G, Nystrom C. 1994. Increased metastable solubility of milled griseofulvin, depending on the formation of a disordered surface structure. Int J Pharm 111:159-170.