Synthesis and in vitro antimicrobial activity of some new 1-thiazolyl-2-pyrazoline derivatives

International Journal of Pharmaceutical Sciences Review and Research

Volumn 1, Issue 2, 2010, Pages 44-48

  Dawane, Bhaskar S ^a   Konda, Shankaraiah G ^a   Shaikh, Baseer M ^a   Chobe, Santosh S ^a   Khandare, Namdev T ^a   Kamble, Vinod T ^b   Bhosale, Raghunath B ^c  

^a Organic Research Laboratory   (India)

^b SWAMI RAMANAND TEERTH MARATHWADA UNIVERSITY   (India)

^c SOLAPUR UNIVERSITY   (India)

Author keywords

1 thizolyl 2 pyrazoline; Antimicrobial activity; Polyethylene glycol 400

Indexed keywords

1 THIAZOLYL 2 PYRAZOLINE DERIVATIVE; 4 (2' HYDROXY 5' CHLOROPHENYL) 2 HYDRAZINO THIAZOLE; CHALCONE DERIVATIVE; MACROGOL 400; NYSTATIN; PYRAZOLINE DERIVATIVE; TETRACYCLINE; THIAZOLE; UNCLASSIFIED DRUG;

ANTIBACTERIAL ACTIVITY; ANTIFUNGAL ACTIVITY; ARTICLE; BACTERIAL STRAIN; BACTERIUM; CATALYSIS; CONTROLLED STUDY; DRUG SCREENING; DRUG STRUCTURE; DRUG SYNTHESIS; FUNGUS; IN VITRO STUDY; MELTING POINT; NONHUMAN;

EID: 79952035328     PISSN: None     EISSN: 0976044X     Source Type: Journal    
DOI: None     Document Type: Article

References (38)

1. Cohen, M. L. Science 1992, 257, 1050
2. Allen, N. E. In Progress in Medicinal Chemistry; Ellis, G. P.; Luscombe, D. K.; Eds.; Elsevier Science: New York, 1995, Vol. 32, Chapter 4, pp 157-238
3. Hayes, J. D.; Wolf, C. R. Biochem. J. 1990, 272, 281
4. Spratt, B. G. Science 1994, 264, 388
5. Nikaido, H. Science 1994, 264, 382.
6. Russel, A. D. In Progress in Medicinal Chemistry; Ellis, G. P.; Luscombe, D. K.; Eds.; Oxford, A. W., Eds.; Elsevier Science: New York, 1998; Vol. 35, Chapter 4
7. Fuchs, T. M. Naturwissenschaften 1998, 85, 99
8. Cunha, B. A. Drugs of Today 1998, 34, 691.
9. Harris, C. R.; Thorarensen, A. Curr. Med. Chem. 2004, 11, 2213.
10. Rubinstein, E. Science 1994, 264, 360.
11. Brumfitt, W.; Hamilton-Miller, J. M. T. Drug Exp. Clin. Res.1994, 20(6), 215.
12. Neu, H. C. Science 1992, 257, 1064.
13. Jungheim, L. N.; Sigmund, S. K.; Fisher, J. W. Tetrahedron Lett. 1987, 28, 285.
14. Jungheim, L. N.; Sigmund, S. K.; Jones, N. D.; Swartz-Endruber, J. K. Tetrahedron Lett. 1987, 28, 289.
15. Boyd, D. B.; In Theoretical and Physiological Studies on β-Lactum Antibiotics, Chemistry and Biology; Morin, R. B.; Gorman, M. Eds.; Academic Press: New York, 1982, Vol. 1, pp 437-545.
16. th Interscience conference on Antimicrobial Agents and Chemotherapy, New Orleans, LA, Sept. 28 - Oct. 1; 1998, Paper 601.
17. th Interscience conference on Antimicrobial Agents and chemotherapy, Los Angels, CA, Oct 23 - 26, 1998, Paper 240.
18. Nasr, M. N. A.; Said, S. A. Arch. Pharm. Pharm. Med. Chem. 2003, 336, 551.
19. Turan-Zitouni, G.; Chevallet, P.; Killic, F. S.; Erol, K. Eur. J. Med. Chem. 2000, 35, 635.
20. Sangwan, N. K.; Dhindsa, K. S.; Malik, O. P.; Malik, M. S.; Chim. Acta Turc. 1983, 11, 65
21. Safak, C.; Tayhan, A.; Sarack, S. J. Indian Chem. Soc. 1990, 67, 571
22. Nauduri, D. Reddy, G. S. Chem. Pharm. Bull. 1998, 46, 1254
23. Grant, N.; Mishriky, N.; Asaad, F. M.; Fawzy, N. G. Pharmazie 1998, 53, 543
24. Turan-Zitouni, G.; Ozdemir, A.; Guven, K. Arch. Pharm. Pharm. Med. Chem. 2005, 338, 96
25. Turan-Zitouni, G.; Ozdemir, A.; Kaplancikli, Z. A.; Chevallet, P.; Tunali, Y. Phosphorous Sulfur Silicon Relat. Elem. 2005, 180, 2717.
26. Gupta, R. R.; Kumar, M.; Gupta, V. In Heterocyclic Chemistry of Five membered Heterocycles; Springer- Verlag: Berlin, Heidelber, New York, 1999, pp. 416.
27. Ashtekar, D. R.; Fernandes, F.; Khadse, B. G.; Shirodkar, M. V. A. Chemotherapy, 1987, 33, 22.
28. Maass, G.; Immendoerfer, U.; Koenig, B.; Leser, U.; Mueller, B.; Goody, R.; Pfatt, B.; Antimicrob. Agents Chemother. 1993, 37, 2612.
29. Fhamy, H. T. Pharmazie 1997, 52, 750
30. Pandeya, S. N.; Sriram, D.; Nath, G. Eur. J. Pharm. Sci. 1999, 9, 25
31. Ates, O.; Altintas, H.; Otuk, G. Arzheimittelforschung 2000, 50, 569
32. Lakhan, R.; Sharma, B. P.; Shukla, B. N. Farmaco 2000, 55, 331
33. Kaplancikli, Z. A.; Turan-Zitouni, G.; Revial, G.; Guven, K. Arch. Pharm. Res. 2004, 27, 1081
34. Turan-Zitouni, G.; Demirayak, S.; Ozdemir, A.; Kaplancikli, Z. A. Yildiz, M. T. Eur. J. Med. Chem. 2004, 39, 267.
35. R. L. Lankey and P. T. Anastas, Life-cycle approaches for assessing green chemistry technologies, Ind. Eng. Chem. Res. 41 (2002) 4498- 4502; DOI: 10.1021/ie0108191.
36. Dawane, B. S.; Konda, S. G.; Mandawad, G. G.; Shaikh, B. M. Poly (ethylene glycol) (PEG-400) as an alternative reaction solvent for the synthesis of some new 1-(4-(4'-chlorophenyl)-2-thiazolyl)-3-aryl-5-(2- butyl-4-chloro-1H-imidazol-5yl)-2-pyrazolines and their in vitro antimicrobial evaluation. Eur. J. Med.Chem. 2010, 45, 387.
37. Davane, B. S.; Bhosale, R. B.; Pekamwar, S. S. J Pharm. Res. 2007, 6(2), 119.
38. D. Shrinivasan; N. Sangeetha; T. Suresh; P. Lakshmanaperumalsamy, J. Ethnophrmacol 2001, 74, 217.