Three austin family compounds from Penicillium brasilianum exhibit selective blocking action on cockroach nicotinic acetylcholine receptors

NeuroToxicology

Volumn 32, Issue 1, 2011, Pages 123-129

  Kataoka, Saori ^a   Furutani, Shogo ^a   Hirata, Koichi ^a   Hayashi, Hideo ^b   Matsuda, Kazuhiko ^a  

^a KINKI UNIVERSITY   (Japan)

^b Osaka Prefecture University   (Japan)

Author keywords

Acetoxydehydroaustin; Austin; Dehydroaustin; Nicotinic acetylcholine receptor; Periplaneta americana; Whole cell patch clamp electrophysiology

Indexed keywords

4 AMINOBUTYRIC ACID RECEPTOR; ACETOXYDEHYDROAUSTIN; AUSTIN DERIVATIVE; CHOLINERGIC RECEPTOR; DEHYDROAUSTIN; EPIBATIDINE; GLUTAMATE RECEPTOR; NATURAL PRODUCT; NICOTINIC RECEPTOR; UNCLASSIFIED DRUG;

AMPLITUDE MODULATION; ARTICLE; CHOLINERGIC RECEPTOR BLOCKING; COCKROACH; CONCENTRATION RESPONSE; CONTROLLED STUDY; ELECTROSTIMULATION; IC 50; NERVOUS SYSTEM ELECTROPHYSIOLOGY; NONHUMAN; PATCH CLAMP; PENICILLIUM; PENICILLIUM BRASILIANUM; PRIORITY JOURNAL; PROTEIN EXPRESSION; TOXICITY TESTING;

ANIMALS; COCKROACHES; DOSE-RESPONSE RELATIONSHIP, DRUG; MALE; NICOTINIC ANTAGONISTS; PENICILLIUM; PERIPLANETA; RECEPTORS, NICOTINIC; TERPENES;

BLATTARIA; HEXAPODA; PENICILLIUM BRASILIANUM; PERIPLANETA AMERICANA;

EID: 78951469514     PISSN: 0161813X     EISSN: None     Source Type: Journal    
DOI: 10.1016/j.neuro.2010.10.003     Document Type: Article

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