Heteroarylimino-4-thiazolidinones as inhibitors of cartilage degradation

Bioorganic Chemistry

Volumn 39, Issue 1, 2011, Pages 48-52

  Panico, Anna Maria ^a   Vicini, Paola ^b   Geronikaki, Athina ^c   Incerti, Matteo ^b   Cardile, Venera ^a   Crasc, Lucia ^a   Messina, Rossella ^a   Ronsisvalle, Simone ^a  

^a UNIVERSITY OF CATANIA   (Italy)

^b UNIVERSITY OF PARMA   (Italy)

^c ARISTOTLE UNIVERSITY OF THESSALONIKI   (Greece)

Author keywords

Glycosaminoglycans; Heteroarylimino 4 thiazolidinones; Metalloproteinases; Nitric oxide; Osteoarthritis

Indexed keywords

2 (BENZO[D]ISOTHIAZOL 3 YLIMINO)THIAZOLIDIN 4 ONE; 2 (BENZO[D]THIAZOL 2 YLIMINO)THIAZOLIDIN 4 ONE; 5 (4 METHOXY BENZYLIDENE) 2 (BENZO[D]ISOTHIAZOL 3 YLIMINO)THIAZOLIDIN 4 ONE; COLLAGENASE 3; GLYCOSAMINOGLYCAN; INTERLEUKIN 1BETA; NITRIC OXIDE; STROMELYSIN; THIAZOLE DERIVATIVE; UNCLASSIFIED DRUG;

ARTICLE; CARTILAGE CELL; CARTILAGE DEGENERATION; CELL CULTURE; CELL VIABILITY; CONTROLLED STUDY; ENZYME INHIBITION; HUMAN; HUMAN CELL; OSTEOARTHRITIS; PRIORITY JOURNAL;

CARTILAGE; CELLS, CULTURED; CHONDROCYTES; GLYCOSAMINOGLYCANS; HUMANS; INTERLEUKIN-1BETA; METALLOPROTEASES; NITROGEN OXIDES; OSTEOARTHRITIS; THIAZOLIDINES;

EID: 78751646205     PISSN: 00452068     EISSN: 10902120     Source Type: Journal    
DOI: 10.1016/j.bioorg.2010.11.002     Document Type: Article

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