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78651240360
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note
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i values were the average of at least two independent determinations. The assay-to-assay variation was generally ±2-fold.
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30
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78651238960
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note
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3H N-α- methylhistamine and 10 μM thioperamide for non-specific binding or assay buffer for total binding. Incubations were performed in quadruplet and stopped by rapid filtration on a Brandel Harvester using Unifilter-96, GF/B plates presoaked in 0.3% PEI for 30 min. The remining radioactivity was measured on a Packard TopCount-NTX. Specific binding was calculated by subtracting the non-specific binding from the total.
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