One-pot production of 18F-biotin by conjugation with 18F-FDG for pre-targeted imaging: Synthesis and radio-labelling of a PEGylated precursor

Applied Radiation and Isotopes

Volumn 69, Issue 2, 2011, Pages 418-422

  Simpson, Michael ^a   Trembleau, Laurent ^a   Cheyne, Richard W ^a   Smith, Tim A D ^a  

^a UNIVERSITY OF ABERDEEN   (United Kingdom)

Author keywords

18F FDG; Avidin; Biotin; Pre target

Indexed keywords

18F-FDG; AVIDIN; BIOTIN; BIOTIN-AVIDIN; ONE POT; PRE-TARGET; TARGETED IMAGING;

SYNTHESIS (CHEMICAL);

COENZYMES;

AVIDIN; BIOTIN; FLOURINE 5 (2 OXO HEXAHYDRO THIENO[3,4 D]IMIDAZOL 4 YL) PENTANOIC ACID [2[2[2[2[2[2[2[2(2AMINOOXY ACETYLAMINO) ETHOXY]ETHOXY]ETHOXY]ETHOXY]ETHOXY]ETHOXY]ETHOXY]ETHYL]AMIDE DIHYDROCHLORIDE F 18; RADIOPHARMACEUTICAL AGENT; UNCLASSIFIED DRUG; DIAGNOSTIC AGENT; DRUG DERIVATIVE; FLUORINE; FLUORODEOXYGLUCOSE F 18; MACROGOL DERIVATIVE; OXIME;

ARTICLE; BINDING AFFINITY; CONTROLLED STUDY; DIAGNOSTIC IMAGING; DRUG STRUCTURE; DRUG SYNTHESIS; HIGH PERFORMANCE LIQUID CHROMATOGRAPHY; ISOTOPE LABELING; MOLECULAR STABILITY; MOLECULAR WEIGHT; POSITRON EMISSION TOMOGRAPHY; PRIORITY JOURNAL; CHEMISTRY; SYNTHESIS;

AVIDIN; BIOTIN; FLUORINE RADIOISOTOPES; FLUORODEOXYGLUCOSE F18; OXIMES; POLYETHYLENE GLYCOLS;

EID: 78650304565     PISSN: 09698043     EISSN: None     Source Type: Journal    
DOI: 10.1016/j.apradiso.2010.10.012     Document Type: Article

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