Gallium labeled NOTA-based conjugates for peptide receptor-mediated medical imaging

Bioorganic and Medicinal Chemistry Letters

Volumn 20, Issue 24, 2010, Pages 7345-7348

  De Sá, Arsénio ^a   Matias, Áurea A ^b   Prata, M Isabel M ^b   Geraldes, Carlos F G C ^c   Ferreira, P M T ^a   André, João P ^a  

^a UNIVERSITY OF MINHO   (Portugal)

^b UNIVERSITY OF COIMBRA   (Portugal)

^c UNIVERSITY OF COIMBRA   (Portugal)

Author keywords

Bifunctional chelators; Gallium; Integrin 3 receptor; Orthogonal protection; Radiopharmacy; Triaza

Indexed keywords

1,4,7 TRIAZACYCLONONANE 1,4,7 TRIACETIC ACID; 1,4,7 TRIAZACYCLONONANE N DECANAMIDE (GLYCINE ARGININE GLYCINEASPARTIC ACID GLYCINE) N',N'' DIACETIC ACID; 1,4,7 TRIAZACYCLONONANE N OCTANAMIDE (GLYCINE ARGININE GLYCINEASPARTIC ACID GLYCINE) N',N'' DIACETIC ACID; [1,4,7 TRIAZACYCLONONANE N HEXANAMIDE (GLYCINE ARGININE GLYCINEASPARTIC ACID GLYCINE) N',N'' DIACETIC ACID; [1,4,7 TRIAZACYCLONONANE N HEXANAMIDE (GLYCINE ARGININE GLYCINEASPARTIC ACID GLYCINE) N',N'' DIACETIC ACID GALLIUM 67; ACETIC ACID; AMINO ACID; GALLIUM; GALLIUM 67; GALLIUM 71; GLYCINE ARGININE GLYCINE ASPARTIC ACID GLYCINE; RADIOISOTOPE; UNCLASSIFIED DRUG; VITRONECTIN RECEPTOR;

AQUEOUS SOLUTION; ARTICLE; CANCER CELL; DIAGNOSTIC IMAGING; DRUG CONJUGATION; DRUG STRUCTURE; DRUG SYNTHESIS; HUMAN; HUMAN CELL; ISOTOPE LABELING; NUCLEAR MAGNETIC RESONANCE SPECTROSCOPY; RECEPTOR BINDING;

AMINO ACID SEQUENCE; CELL LINE, TUMOR; CONTRAST MEDIA; COORDINATION COMPLEXES; GALLIUM; HETEROCYCLIC COMPOUNDS; HUMANS; INTEGRIN ALPHAVBETA3; PEPTIDES;

EID: 78449295632     PISSN: 0960894X     EISSN: None     Source Type: Journal    
DOI: 10.1016/j.bmcl.2010.10.059     Document Type: Article

References (37)

1. M. Fani, J.P. André, and H.R. Maecke Contrast Media Mol. Imaging 3 2008 67
2. C.J. Anderson, and M.J. Welch Chem. Rev. 99 1999 2219
3. A.E. Martell, R.J. Motekaitis, and M.J. Welch J. Chem. Soc., Chem. Commun. 1990 1748
4. A. de Sa, M.I.M. Prata, C.F.G.C. Geraldes, and J.P. Andre J. Inorg. Biochem. 104 2010 1051
5. E.T. Clarke, and A.E. Martell Inorg. Chim. Acta 181 1991 273
6. C.J. Anderson, C.S. John, Y.J. Li, R.D. Hancock, T.J. McCarthy, A.E. Martell, and M.J. Welch Nucl. Med. Biol. 22 1995 165
7. J.P. André, and H.R. Mäcke J. Inorg. Biochem. 97 2003 315
8. Y.Z. Sun, C.J. Anderson, T.S. Pajeau, D.E. Reichert, R.D. Hancock, R.J. Motekaitis, A.E. Martell, and M.J. Welch J. Med. Chem. 39 1996 458
9. T.M. Jones-Wilson, R.J. Motekaitis, Y. Sun, C.J. Anderson, A.E. Martell, and M.J. Welch Nucl. Med. Biol. 22 1995 859
10. W.R. Harris, and A.E. Martell Inorg. Chem. 15 1976 713
11. M.A. Green, and M.J. Welch Int. J. Rad. Appl. Instrum. B 16 1989 435
12. E. Cole, D. Parker, G. Ferguson, J.F. Gallagher, and B. Kaitner J. Chem. Soc., Chem. Commun. 1991 1473
13. J.P. André, H.R. Maecke, M. Zehnder, L. Macko, and K.G. Akyel Chem. Commun. 1998 1301
14. M.I.M. Prata, A.C. Santos, C.F.G.C. Geraldes, and J.J.P. de Lima Nucl. Med. Biol. 26 1999 707
15. R.J. Motekaitis, Y. Sun, and A.E. Martell Inorg. Chim. Acta 198 1992 421
16. R. Ma, M.J. Welch, J. Reibenspies, and A.E. Martell Inorg. Chim. Acta 236 1995 75
17. E.T. Clarke, and A.E. Martell Inorg. Chim. Acta 186 1991 103
18. P.J. Riss, C. Kroll, V. Nagel, and F. Rosch Bioorg. Med. Chem. Lett. 18 2008 5364
19. S. Liu Chem. Soc. Rev. 33 2004 445
20. R.E. Weiner, and M.L. Thakur BioDrugs 19 2005 145
21. C.J. Smith, W.A. Volkert, and T.J. Hoffman Nucl. Med. Biol. 32 2005 733
22. M. Béhé, and T.M. Behr Biopolymers 66 2002 399
23. A. Heppeler, J.P. Andre, I. Buschmann, X.J. Wang, J.C. Reubi, M. Hennig, T.A. Kaden, and H.R. Maecke Chem. Eur. J. 14 2008 3026
24. H.R. Maecke, and J.P. André PET Chemistry The Driving Force in Molecular Imaging 2007 Springer Berlin
25. R. Hwang, and J. Varner Hematol. Oncol. Clin. North Am. 18 2004 991
26. J. Folkman Semin. Oncol. 29 2002 15
27. S. Zitzmann, V. Ehemann, and M. Schwab Cancer Res. 62 2002 5139
28. J. Folkman Nat. Med. 1 1995 27
29. I. Dijkgraaf, J.A. Kruijtzer, S. Liu, A.C. Soede, W.J. Oyen, F.H. Corstens, R.M. Liskamp, and O.C. Boerman Eur. J. Nucl. Med. Mol. Imaging 34 2007 267
30. S. Liu Mol. Pharm. 3 2006 472
31. J.B. Miller J. Org. Chem. 24 1959 560
32. -1).
33. A.S. Craig, D. Parker, H. Adams, and N.A. Bailey J. Chem. Soc., Chem. Commun. 1989 1793
34. X.Y. Chen, R. Park, A.H. Shahinian, J.R. Bading, and P.S. Conti Nucl. Med. Biol. 31 2004 11
35. D. Yahalom, A. Wittelsberger, D.F. Mierke, M. Rosenblatt, J.M. Alexander, and M. Chorev Biochemistry 41 2002 8321
36. Fontes, A.; Prata, M. I. M.; Geraldes, C. F. G. C.; Andre, J. P. Nucl. Med. Biol. in press.
37. Results not published.