Recrystallization of erlotinib hydrochloride and fulvestrant using supercritical antisolvent process

Journal of Supercritical Fluids

Volumn 55, Issue 1, 2010, Pages 292-299

  Tien, Yao Chun ^a   Su, Chie Shaan ^b   Lien, Ling Hsiao ^b   Chen, Yan Ping ^a  

^a NATIONAL TAIWAN UNIVERSITY   (Taiwan)

^b ScinoPharm Taiwan Ltd   (Taiwan)

Author keywords

Antisolvent; Erlotinib hydrochloride; Fulvstrant; Micronization; Polymorphism; Supercritical carbon dioxide

Indexed keywords

ANTI-SOLVENTS; ERLOTINIB; FULVSTRANT; MICRONIZATIONS; SUPERCRITICAL CARBON DIOXIDES;

CARBON DIOXIDE; CARBON DIOXIDE PROCESS; DISSOLUTION; PARTICLE SIZE; PARTICLE SIZE ANALYSIS; POLYMORPHISM; PRESSURE EFFECTS; RECRYSTALLIZATION (METALLURGY); TEMPERATURE;

SUPERCRITICAL FLUID EXTRACTION;

EID: 78049312661     PISSN: 08968446     EISSN: None     Source Type: Journal    
DOI: 10.1016/j.supflu.2010.06.009     Document Type: Article

References (35)

1. 2 in green chemical synthesis and processing Journal of Supercritical Fluids 28 2004 121 191
2. A.S. Teja, and C.A. Eckert Commentary on supercritical fluids: research and applications Industrial & Engineering Chemistry Research 39 2000 4442 4444
3. E. Reverchon, and G. Della Porta Particle design using supercritical fluids Chemical Engineering & Technology 26 2003 840 845
4. A. Martin, and M.J. Cocero Micronization processes with supercritical fluids: fundamentals and mechanism Advanced Drug Delivery Reviews 60 2008 339 350 (Pubitemid 351215568)
5. J. Jung, and M. Perrut Particle design using supercritical fluids: literature and patent survey Journal of Supercritical Fluids 20 2001 179 219
6. B.Y. Shekunov, and P. York Crystallization processes in pharmaceutical technology and drug delivery design Journal of Crystal Growth 211 2000 122 136
7. S.L. Morissette, Ö. Almarsson, M.L. Peterson, J.F. Remenar, M.J. Read, A.V. Lemmo, S. Ellis, M.J. Cima, and C.R. Gardner High-throughput crystallization: polymorphs, salts, co-crystals and solvates of pharmaceutical solids Advanced Drug Delivery Reviews 56 2004 275 300
8. A. Llins, and J.M. Goodman Polymorph control: past, present and future Drug Discovery Today 13 2008 198 210
9. S. Gracin, M. Uusi-Penttilä, and.C. Rasmuson Influence of ultrasound on the nucleation of polymorphs of p-aminobenzoic acid Crystal Growth Design 5 2005 1787 1794
10. Y. Wang, Y. Wang, J. Yang, R. Pfeffer, R. Dave, and B. Michniak The application of a supercritical antisolvent process for sustained drug delivery Powder Technology 164 2006 94 102
11. S.J. Park, S.Y. Jeon, and S.D. Yeo Recrystallization of a pharmaceutical compound using liquid and supercritical antisolvents Industrial & Engineering Chemistry Research 45 2006 2287 2293
12. C.S. Su, and Y.P. Chen Recrystallization of salicylamide using a batch supercritical anisolvent process Chemical Engineering & Technology 28 2005 1177 1181
13. Y.P. Chang, M. Tang, and Y.P. Chen Micronization of sulfamethoxazole using the supercritical anti-solvent process Journal of Materials Science 43 2008 2328 2335
14. C.S. Yoon, H.D. Park, S.Y. Kim, and S.H. Kim High molecular weight poly(l-lactide) and its microsphere synthesized in the supercritical dimethyl ether Macromolecular Symposia 249-250 2007 515 520
15. K.H. Song, C.H. Lee, J.S. Lim, and Y.W. Lee Preparation of L-PLA submicron particles by a continuous supercritical antisolvent precipitation process Korean Journal of Chemical Engineering 19 2002 139 145
16. E. Reverchon, R. Adami, G. Caputo, and I.D. Marco Spherical microparticles production by supercritical antisolvent precipitation: interpretation results Journal of Supercritical Fluids 47 2008 70 84
17. R. Sordella, D.W. Bell, D.A. Haber, and J. Settleman Gefitinib- sensitizing EGFR mutations in lung cancer activate anti-apoptotic pathways Science 305 2004 1163 1167
18. T. Norris, J.W. Raggon, R.D. Connell, J.D. Moyer, M.J. Morin, S.M. Kajiji, B.A. Foster, K.J. Ferrante, S.L. Silberman, Stable polymorph on N-(3-ethynylphenyl)-6,7-bis(2methoxyethoxy)-4-quinazolinamine hydrochloride, methods of production, and pharmaceutical uses thereof, US patent 6,900,221 B1, 2005.
19. A.G. Bubendorf, M. Hennig, P. Hidber, G. Rimmler, F. Rohrer, Polymorph of {6,7-bis(2-methoxy-ethoxy)-quinazolin-4-yl}-(3E), WO patent 2004/072049 A1, 2004.
20. S. Kansra, S. Yamagata, L. Sneade, L. Foster, and N. Ben-Jonathan Differential effects of estrogen receptor antagonists on pituitary lactotroph proliferation and prolactin release Molecular and Cellular Endocrinology 239 2005 27 36
21. L. Hong, J.Z. Guo, Y. Gao, and W.K. Yuan Precipitation of microparticulate organic pigment powders by a supercritical antisolvent process Industrial & Engineering Chemistry Research 39 2000 4882 4887
22. The United States Pharmacopeia 31th ed. 2008 The United States Pharmacopeial Convention Rockville, MD, USA
23. R. Adami, E. Reverchon, E. Järvenpää, and R. Huopalahti Supercritical antisolvent micronization of nalmefene HCl on laboratory and pilot scale Powder Technology 182 2008 105 112
24. E. Reverchon, and I. De Marco Supercritical antisolvent precipitation of cephalosporins Powder Technology 164 2006 139 146
25. S.D. Yeo, S.J. Park, J.W. Kim, and J.C. Kim Critical properties of carbon dioxide + methanol, +ethanol, +1-propanol, and +1-butanol Journal of Chemical and Engineering Data 45 2000 932 935
26. 2 Pharmaceutical Research 18 2001 682 688
27. H.H.Y. Tong, B.Y. Shekunov, P. York, and A.H.L. Chow Influence of operating temperature and pressure on the polymorphic transition of salmeterol xinafoate in supercritical fluids Journal of Pharmaceutical Sciences 97 2008 1025 1029
28. S.P. Velaga, R. Berger, and J. Carlfors Supercritical fluids crystallization of budesonide and flunisolide Pharmaceutical Research 19 2002 1564 1571
29. C.S. Su, M. Tang, and Y.P. Chen Micronization of nabumetone using the rapid expansion of supercritical solution (RESS) process Journal of Supercritical Fluids 50 2009 69 76
30. T. Holderbaum, and J. Gmehling PSRK: a group contribution equation of state based on UNIFAC Fluid Phase Equilibria 70 1991 251 265
31. J. Gmehling, J. Li, and K. Fischer Further development of the PSRK model for the prediction of gas solubilities and vapor-liquid equilibria at low and high pressure II Fluid Phase Equilibria 141 1997 113 127
32. K. Fischer, and J. Gmehling Further development, status and results of the PSRK method for the prediction of vapor-liquid equilibria and gas solubilities Fluid Phase Equilibria 121 1996 185 206
33. S. Horstmann, K. Fischer, and J. Gmehling PSRK group contribution of state: revision and extension III Fluid Phase Equilibria 167 2000 173 186
34. G.R. Borges, A. Junges, E. Franceschi, F.C. Corazza, M.L. Corazza, J.V. Oliveira, and C. Dariva High-pressure vapor-liquid equilibrium data for systems involving carbon dioxide + organic solvent + β-carotene Journal of Chemical and Engineering Data 52 2007 1437 1441
35. M.S. Kim, S. Lee, J.S. Park, J.S. Woo, and S.J. Hwang Micronization of cilostazol using supercritical antisolvent (SAS) process: effect of process parameters Powder Technology 177 2007 64 70 (Pubitemid 47224964)