Selective determinants of inositol 1,4,5-trisphosphate and adenophostin A interactions with type 1 inositol 1,4,5-trisphosphate receptors

British Journal of Pharmacology

Volumn 161, Issue 5, 2010, Pages 1070-1085

  Rossi, Ana M ^a   Sureshan, Kana M ^b   Riley, Andrew M ^b   Potter, Barry V L ^b   Taylor, Colin W ^a  

^a UNIVERSITY OF CAMBRIDGE   (United Kingdom)

^b University of Bath   (United Kingdom)

Author keywords

Adenophostin; Ca 2+ signal; IP 3 receptor; Structure activity relationship

Indexed keywords

ADENOPHOSTIN A; CATION; INOSITOL 1,4,5 TRISPHOSPHATE; INOSITOL 1,4,5 TRISPHOSPHATE RECEPTOR; INOSITOL 1,4,5 TRISPHOSPHATE RECEPTOR 1; UNCLASSIFIED DRUG;

AMINO TERMINAL SEQUENCE; ANIMAL EXPERIMENT; ARTICLE; BINDING AFFINITY; CALCIUM TRANSPORT; CONTROLLED STUDY; DRUG BINDING; DRUG POTENCY; DRUG STRUCTURE; DRUG SYNTHESIS; MALE; MUTATIONAL ANALYSIS; NONHUMAN; NUCLEOTIDE SEQUENCE; PRIORITY JOURNAL; RAT;

ADENOSINE; ANIMALS; CALCIUM; CALCIUM CHANNEL AGONISTS; INOSITOL 1,4,5-TRISPHOSPHATE; INOSITOL 1,4,5-TRISPHOSPHATE RECEPTORS; MALE; MUTATION; PROTEIN BINDING; RATS; RATS, WISTAR;

EID: 77958558893     PISSN: 00071188     EISSN: 14765381     Source Type: Journal    
DOI: 10.1111/j.1476-5381.2010.00947.x     Document Type: Article

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