Quantitative structure-activity relationship analysis of 4(3H)-quinazolone derivatives as tyrosine kinase inhibitors by multiple linear regression

Cancer Biotherapy and Radiopharmaceuticals

Volumn 25, Issue 5, 2010, Pages 559-562

  Srivastava, Vikas ^a,b   Sinha, Deepa ^a   Tiwari, Anjani K ^a   Sharma, Himanshu ^c   Bala Sharma, Raj ^b   Singh, Vinay K ^a   Mishra, Anil K ^a  

^a INSTITUTE OF NUCLEAR MEDICINE AND ALLIED SCIENCES   (India)

^b Meerul College   (India)

^c Translam Institute of Technology and Management   (India)

Author keywords

4(3H) quinozolone; computational chemistry; MLR; QSAR

Indexed keywords

4(3H) QUINAZOLINONE DERIVATIVE; PROTEIN TYROSINE KINASE INHIBITOR;

ARTICLE; DRUG ABSORPTION; DRUG DISTRIBUTION; DRUG EXCRETION; DRUG METABOLISM; DRUG SCREENING; MATHEMATICAL MODEL; MINIMUM INHIBITORY CONCENTRATION; MULTIPLE LINEAR REGRESSION ANALYSIS; PRIORITY JOURNAL; QUANTITATIVE STRUCTURE ACTIVITY RELATION;

ALGORITHMS; ENZYME INHIBITORS; MODELS, CHEMICAL; MOLECULAR STRUCTURE; PROTEIN-TYROSINE KINASES; QUANTITATIVE STRUCTURE-ACTIVITY RELATIONSHIP; QUINAZOLINES; REGRESSION ANALYSIS; SOFTWARE;

EID: 77958164935     PISSN: 10849785     EISSN: None     Source Type: Journal    
DOI: 10.1089/cbr.2010.0791     Document Type: Article

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