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Bioorganic and Medicinal Chemistry Letters

Volumn 20, Issue 22, 2010, Pages 6854-6857

Development of the next generation of HIV-1 integrase inhibitors: Pyrazolone as a novel inhibitor scaffold

(6) Hadi, Victor a Koh, Yung Hyo a Sanchez, Tino Wilson a Barrios, Danielle a Neamati, Nouri a Jung, Kyung Woon a

a UNIVERSITY OF SOUTHERN CALIFORNIA (United States)

Author keywords

HIV; Integrase inhibition; Pyrazolone scaffold

Indexed keywords

3 BROMOPHENYL; 3 CHLOROPHENYL; 3 FLUOROPHENYL; 3 IODOPHENYL; 3 NITROPHENYL; 3 PHENYLPHENYL; 3 TOLYL; 3 TRIFLUOROMETHYLPHENYL; 3,5 DICHLOROPHENYL; 4 BROMOPHENYL; 4 CARBOXYLPHENYL; 4 IODOPHENYL; 4 SULFONYAMIDOPHENYL; BENZOTHIAZOLYL; CARBOXYLIC ACID; CARBOXYLIC ACID ETHYL ESTER; ELVITEGRAVIR; ETHYL 6 DEOXY 3,5 DI O METHYL 6 (3 METHYL 3 NITROSOUREIDO) ALPHA GLUCOFURANOSIDE; HOMOACETATE; HYDRAZINE; INTEGRASE INHIBITOR; METHYL HOMOACETATE; METHYLENE BLUE; PHENYL GROUP; PYRAZOLONE; TRIFLUOROACETAMIDE DERIVATIVE; TRIFLUOROMETHYL; UNCLASSIFIED DRUG;

ARTICLE; BINDING AFFINITY; CYCLIZATION; DRUG ACTIVITY; DRUG DESIGN; DRUG SYNTHESIS; HUMAN IMMUNODEFICIENCY VIRUS 1; IC 50; IN VITRO STUDY; PHARMACOPHORE; STRUCTURE ACTIVITY RELATION;

CATALYSIS; HIV INTEGRASE INHIBITORS; HIV-1; MODELS, MOLECULAR; MUTATION; PYRAZOLONES; STRUCTURE-ACTIVITY RELATIONSHIP;

HUMAN IMMUNODEFICIENCY VIRUS 1;

EID: 77958035040 PISSN: 0960894X EISSN: None Source Type: Journal
DOI: 10.1016/j.bmcl.2010.08.057 Document Type: Article

Times cited : (99)

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