Synthesis and antituberculosis activity of some new pyridazine derivatives. Part II

European Journal of Medicinal Chemistry

Volumn 45, Issue 11, 2010, Pages 5164-5168

  Mantu, Dorina ^a   Cǎtǎlina Luca, Mihaela ^b   Moldoveanu, Costel ^a   Zbancioc, Gheorghita ^a   Mangalagiu, Ionel I ^a  

^a ALEXANDRU IOAN CUZA UNIVERSITY OF IASI   (Romania)

^b GRIGORE T POPA UNIVERSITY OF MEDICINE AND PHARMACY   (Romania)

Author keywords

Antituberculosis; Pyridazine; SAR; Ultrasound

Indexed keywords

2 (PROP 2 YNYL) 6 4 TOLYLPYRIDAZIN 3(2H) ONE; 2 [3 (4 BROMOPHENYL) 6 OXOPYRIDAZIN 1(6H) YL]ACETAMIDE; 2 [3 (4 CHLOROPHENYL) 6 OXOPYRIDAZIN 1(6H) YL]ACETAMIDE; 2 [3 (4 CHLOROPHENYL) 6 OXOPYRIDAZIN 1(6H) YL]ACETATE; 2 [6 OXO 3 4 TOLYLPYRIDAZIN 1(6H) YL]ACETAMIDE; 2 ALLYL 6 (4 BROMOPHENYL)PYRIDAZIN 3(2H) ONE; 2 ALLYL 6 (4 CHLOROPHENYL)PYRIDAZIN 3(2H) ONE; 2 ALLYL 6 4 TOLYLPYRIDAZIN 3(2H) ONE; 6 (4 BROMOPHENYL) 2 (PROP 2 YNYL)PYRIDAZIN 3(2H) ONE; 6 (4 CHLOROPHENYL) 2 (PROP 2 YNYL)PYRIDAZIN 3(2H) ONE; ETHYL 2 [3 (4 BROMOPHENYL) 6 OXOPYRIDAZIN 1(6H) YL]ACETATE; ETHYL 2 [3 (4 BROMOPHENYL) 6 OXOPYRIDAZIN 1(6H) YL]PROPANOATE; ETHYL 2 [3 (4 CHLOROPHENYL) 6 OXOPYRIDAZIN 1(6H) YL]PROPANOATE; ETHYL 2 [6 OXO 3 4 TOLYLPYRIDAZIN 1(6H) YL]ACETATE; ETHYL 2 [6 OXO 3 4 TOLYLPYRIDAZIN 1(6H) YL]PROPANOATE; METHYL 2 [3 (4 BROMOPHENYL) 6 OXOPYRIDAZIN 1(6H) YL]ACETATE; METHYL 2 [3 (4 CHLOROPHENYL) 6 OXOPYRIDAZIN 1(6H) YL]ACETATE; METHYL 2 [6 OXO 3 4 TOLYLPYRIDAZIN 1(6H) YL]ACETATE; PYRIDAZINE DERIVATIVE; PYRIDAZINONE DERIVATIVE; TUBERCULOSTATIC AGENT; UNCLASSIFIED DRUG;

ANTIBACTERIAL ACTIVITY; ARTICLE; CONTROLLED STUDY; DRUG MECHANISM; DRUG STRUCTURE; DRUG SYNTHESIS; IC 50; IN VITRO STUDY; IRRADIATION; MYCOBACTERIUM TUBERCULOSIS; NONHUMAN; STRUCTURE ACTIVITY RELATION;

ANTITUBERCULAR AGENTS; MAGNETIC RESONANCE SPECTROSCOPY; MICROBIAL SENSITIVITY TESTS; MYCOBACTERIUM TUBERCULOSIS; PYRIDAZINES; STRUCTURE-ACTIVITY RELATIONSHIP;

EID: 77957842253     PISSN: 02235234     EISSN: 17683254     Source Type: Journal    
DOI: 10.1016/j.ejmech.2010.08.029     Document Type: Article

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