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Durable efficacy and safety of etravirine (ETR; TMC125) in treatment-experienced, HIV-1-infected patients: Pooled week 96 results from the Phase III DUET-1 and DUET-2 trials
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TMC125 in combination with other medications: Summary of drug-drug interaction studies
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Kakuda, T.N.1
Schöller-Gyüre, M.2
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Effect of etravirine on cytochrome P450 isozymes assessed by the Cooperstown 5+1 cocktail
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48th Interscience Conference on Antimicrobial Agents and Chemotherapy and 46th Infectious Disease Society of America Meeting. 25-28 October 2008, Washington, DC, USA
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Kakuda, T.N.2
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Pharmacokinetics of 2',3'-dideoxyadenosine and 2',3'-dideoxyinosine in patients with severe human immunodeficiency virus infection
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Pharmacokinetics of etravirine (ETR; TMC125) are not affected by sex, age, race, use of enfuvirtide (ENF) or treatment duration in HIV-1-infected subjects
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Drug interactions with TMC125, a potent next generation nonnucleoside reverse transcriptase inhibitor
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Baede, P.1
Piscitelli, S.2
Graham, N.3
Van't Klooster, G.4
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Clinical pharmacology of TMC114 - A new HIV protease inhibitor
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Hoetelmans, R.4
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Pharmacokinetics of amprenavir and TMC125 in HIVinfected volunteers receiving TMC125 with fosamprenavir/ritonavir
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47
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77957369802
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56
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Pharmacokinetics, safety, and efficacy of tipranavir boosted with ritonavir alone or in combination with other boosted protease inhibitors as part of optimized combination antiretroviral therapy in highly treatment-experienced patients (BI study 1182.51)
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Pharmacokinetics (PK) and safety of adding TMC125 to stable regimens of saquinavir (SQV), lopinavir (LPV), ritonavir (RTV) and NRTIs in HIV+ adults
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An open, randomized, two period, crossover study in 2 cohorts to investigate the effect of steady state TMC125 and the combination of TMC125/darunavir/ritonavir on the steady state pharmacokinetics of oral maraviroc in healthy subjects
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