Synthesis and biological evaluation of some novel 2-mercaptobenzothiazoles carrying 1,3,4-oxadiazole, 1,3,4-thiadiazole and 1,2,4-triazole moieties

South African Journal of Chemistry

Volumn 63, Issue , 2010, Pages 114-122

  Azam, M Afzal ^a   Suresh, Bhojraj ^a   Kalsi, Sandip S ^a   Antony, A Shinesh ^a  

^a JSS COLLEGE OF PHARMACY   (India)

Author keywords

1,3,4 oxadiazoles; 1,3,4 Thiadiazoles; 2 Mercaptobenzothiazoles; Anti inflammatory activity; Antimicrobial activity

Indexed keywords

EID: 77956921560     PISSN: 03794350     EISSN: None     Source Type: Journal    
DOI: None     Document Type: Article

References (26)

1. G. Dannhardt and W. Kiefer, Eur. J. Med. Chem., 2001, 36, 109-126.
2. Y. Song, D.T. Connor, R. Doubleday, R.J. Sorenson, A.D. Sercel, P.C. Unangst, B.D. Roth, R.B. Gilbertsen, K. Chan, D.J. Schrier, A. Guglietta, D.A. Bornemeier and R.D. Dyer, J. Med. Chem., 1999, 42, 1151-1160.
3. A.S. Kalgutkar, A.B. Marnett, B.C. Crews, R.P. Remmel and L.J. Marnett, J. Med. Chem., 2000, 43, 2860-2870.
4. S.M. Sondhi, N. Singhal, M. Johar, B.S. Narayan Reddy and J.W. Lown, Curr. Med. Chem., 2002, 9, 1045-1074.
5. M.C. Allison, A.G. Howatson, C.J. Torrance, F.D. Lee and R.I. Russell, N. Engl. J. Med., 1992, 327, 749-754.
6. R.J. Flower, Nat. Rev. Drug. Discov., 2003, 2, 179-191.
7. D.H. Boshelli, D.T. Connor, D.A. Bornemeier,R.D. Dyer, J.A.Kennedy, P.J. Kupiers, G.C. Okonkow, D.J. Schrier and C.D. Wright, J. Med. Chem., 1993, 36, 1802-1810.
8. M.D. Mullican, M.W. Wilson, D.T. Connor, C.R. Kostlan, D.J. Schrier and R.D. Dyer, J. Med. Chem., 1993, 36, 1090-1099.
9. H. Kumar, S.A. Javed, S.A. Khan and M. Amir, Eur. J. Med. Chem., 2008, 43, 2688-2698.
10. P.G. Baraldi, M.G. Pavani, M.C. Nunez, P. Brigidi, B.Vitali,R. Gambari and R. Romagnoli, Bioorg. Med. Chem., 2002, 10, 449-456.
11. A.A. Kadi, N.R. El-Brollosy, O.A. Al-Deeb, E.E. Haeeb, T.M. Ibrahim and A.A. El-Emam, Eur. J. Med. Chem., 2007, 42, 235-242.
12. V. Padmavathi, A.V.N. Mohan, P. Thriveni and A. Shazia, Eur. J. Med. Chem., 2009, 44, 2313-2321.
13. A. Naya, K. Kobayashi, M. Ishikawa, K. Ohwaki, T. Saeki, K. Noguchi and N. Ohtake, Chem. Pharm. Bull., 2003, 51, 697-701.
14. M.I. Hussain and V. Kumar, Indian J. Chem., 1993, 32B, 905-907.
15. K.G. Desai and K.R. Desai, Indian J. Chem., 2005, 44B, 2093-2096.
16. N. Karali, N. Cesur, A. Gursoy, O. Ates, S. Ozen, G. Otuk and S. Birteksoz, Indian J. Chem., 2004, 43B, 212-216.
17. K.G. Desai, J.P. Raval and K.R. Desai, J. Iranian Chem. Soc., 2006, 3, 233-241.
18. B.R. Rani, U.T. Bhalerao and M.F. Rahman, Indian J. Chem., 1990, 29B, 995-998.
19. S.K. Srivastava, R. Yadav and S.D. Srivastava, Indian J. Chem., 2004, 43B, 399-405.
20. M.I. Hussain and V. Kumar, Indian J. Chem., 1992, 31B, 673-675.
21. B.S. Furniss, A.J. Hannford, P.W.G. Smith and A.R. Tatchell, Vogel's Text Book of Practical Organic Chemistry, Pearson Education, Singapore, 2005, pp. 1249.
22. M. Mahalinga, B.S. Holla and N.S.Kumari, Eur. J. Med. Chem., 2008, 43, 25-31.
23. J.M. Glassman, Agents with AnalgesicActivity and Dependences Liability, in Screening Methods in Pharmacology (R.A. Turner and P. Hebborn eds.), Academic Press, New York, USA, 1971, 2, pp. 231-232.
24. C.A.Winter, E.A. Risley and G.N. Nuss, Proc. Soc. Exp. Biol., 1962, 111, 544-547.
25. V. Cioli, S. Putzolu, V. Rossi, P.S. Barcellona and C. Corradino, Toxicol. Appl. Pharmacol., 1979, 50, 283-289.
26. A.L.J. Barry, The Antimicrobial Susceptibility Test, Principle and Practices, 4th edn., ELBS, London, UK, 1999, pp. 180.