SCOPUS 정보 검색 플랫폼

Volumn 18, Issue 19, 2010, Pages 7092-7100

Structure-based virtual screening of novel tubulin inhibitors and their characterization as anti-mitotic agents

(9) Kim, Nam Doo a,c Park, Eun Sook b Kim, Young Hoon c Moon, Seung Kee d Lee, Sung Sook d Ahn, Soon Kil e Yu, Dae Yeul f No, Kyoung Tai a Kim, Kyun Hwan b

a Yonsei University (South Korea)

b Konkuk University (South Korea)

c Equispharm Co Ltd (South Korea)

d Chong Kun Dang Research Institute (South Korea)

e SolarLight Ltd (South Korea)

f Korea Research Institute of Bioscience and Biotechnology (KRIBB) (South Korea)

Author keywords

Colchicine; Microtubule; Molecular docking; Pharmacophore; Virtual screening

Indexed keywords

ANTIMITOTIC AGENT; ANTINEOPLASTIC AGENT; COLCHICINE; PODOPHYLLOTOXIN; TUBULIN; TUBULIN INHIBITOR; UNCLASSIFIED DRUG;

APOPTOSIS; ARTICLE; CELL CYCLE ARREST; CELL CYCLE G2 PHASE; CELL CYCLE M PHASE; CELL CYCLE PROGRESSION; CELL DIVISION; CELL MOTION; CELL STRAIN HL 60; CRYSTAL STRUCTURE; CYTOSKELETON; DRUG ACTIVITY; DRUG PROTEIN BINDING; DRUG SCREENING; DRUG STRUCTURE; HUMAN; HUMAN CELL; IN VITRO STUDY; MICROTUBULE; MICROTUBULE ASSEMBLY; MOLECULAR DOCKING; MOLECULAR MODEL;

APOPTOSIS; CELL CYCLE; CELL DIVISION; CELL PROLIFERATION; CRYSTALLOGRAPHY, X-RAY; DRUG DISCOVERY; DRUG SCREENING ASSAYS, ANTITUMOR; G2 PHASE; HUMANS; MITOSIS; MODELS, MOLECULAR; MOLECULAR STRUCTURE; SMALL MOLECULE LIBRARIES; STEREOISOMERISM; STRUCTURE-ACTIVITY RELATIONSHIP; TUBULIN; TUBULIN MODULATORS; TUMOR CELLS, CULTURED;

EID: 77956649106 PISSN: 09680896 EISSN: None Source Type: Journal
DOI: 10.1016/j.bmc.2010.07.072 Document Type: Article

Times cited : (49)

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