Highly efficient production of [18F]fallypride using small amounts of base concentration

Applied Radiation and Isotopes

Volumn 68, Issue 12, 2010, Pages 2279-2284

  Seok Moon, Byung ^a,b   Hyung Park, Jun ^a   Jin Lee, Hong ^a   Sun Kim, Ji ^a   Sup Kil, Hee ^c   Se Lee, Byoung ^c   Yoon Chi, Dae ^c   Chul Lee, Byung ^a,b   Kyeong Kim, Yu ^a   Eun Kim, Sang ^a,b  

^a Seoul National University Bundang Hospital   (South Korea)

^b Seoul National University College of Medicine   (South Korea)

^c Sogang University   (South Korea)

Author keywords

18F Fallypride; Automated radiosynthesis; Dopamine D2 D3 receptor; PET

Indexed keywords

[18F]FALLYPRIDE; AUTOMATED SYNTHESIS; DOPAMINE D2/D3 RECEPTOR; EFFICIENT PRODUCTION; OPTIMAL LABELING; PET; PHASE-TRANSFER CATALYSTS; RADIOCHEMICAL YIELD; RADIOSYNTHESIS; SOLID-PHASE; TETRABUTYLAMMONIUM; TOTAL SYNTHESIS;

ACETONITRILE; BRAIN; CATALYSTS; DEIONIZED WATER; ION EXCHANGE; ORGANIC SOLVENTS; PURIFICATION;

AUTOMATION;

ACETONITRILE; CRYPTAND 2.2.2; FLUORINE 18; N [(1 ALLYL 2 PYRROLIDINYL)METHYL] 5 (3 FLUOROPROPYL) 2,3 DIMETHOXYBENZAMIDE F 18; OXYGEN 18; RADIOPHARMACEUTICAL AGENT; TETRABUTYLAMMONIUM; UNCLASSIFIED DRUG;

ARTICLE; AUTOMATION; CONCENTRATION PROCESS; DRUG ISOLATION; DRUG PURIFICATION; DRUG STRUCTURE; DRUG SYNTHESIS; HIGH PERFORMANCE LIQUID CHROMATOGRAPHY; PRIORITY JOURNAL; PROCESS OPTIMIZATION; RADIOCHEMISTRY; REACTION TIME; SOLVENT EFFECT; TEMPERATURE SENSITIVITY;

CATALYSIS; FLUORIDES;

EID: 77956411632     PISSN: 09698043     EISSN: None     Source Type: Journal    
DOI: 10.1016/j.apradiso.2010.06.016     Document Type: Article

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