-
1
-
-
0023152230
-
Search of the digitalis replacement
-
Erhardt, P. W. In search of the digitalis replacement. J. Med. Chem. 1987, 30, 231-237
-
(1987)
J. Med. Chem.
, vol.30
, pp. 231-237
-
-
Erhardt, P.W.1
-
2
-
-
0026064751
-
2-Phenyl-3H-imidazo[4,5-b]pyridine-3- acetamides as nonbenzodiazepine anticonvulsants and anxiolytics
-
Tomczuk, B. E.; Taylor Jr., C. R.; Moses, L. M.; Sutherland, D. B.; Lo, Y. S.; Johnson, D. N.; Kinnier, W. B.; Kilpatrick, B. F. 2-Phenyl-3H-imidazo[4, 5-b]pyridine-3- acetamides as nonbenzodiazepine anticonvulsants and anxiolytics. J. Med. Chem. 1991, 34, 2993-3006
-
(1991)
J. Med. Chem.
, vol.34
, pp. 2993-3006
-
-
Tomczuk, B.E.1
Taylor Jr., R.C.2
Moses, L.M.3
Sutherland, D.B.4
Lo, Y.S.5
Johnson, D.N.6
Kinnier, W.B.7
Kilpatrick, B.F.8
-
3
-
-
33751157540
-
DNA-directed alkylating agents 6: Synthesis and antitumor activity of DNA minor groove-targeted aniline mustard analogs of pibenzimol (Hoechst 33258)
-
Gravatt, G. L.; Baguley, B. C.; Wilson, W. R.; Denny, W. A. DNA-directed alkylating agents, 6: Synthesis and antitumor activity of DNA minor groove-targeted aniline mustard analogs of pibenzimol (Hoechst 33258). J. Med. Chem. 1994, 37, 4338-4345.
-
(1994)
J. Med. Chem.
, vol.37
, pp. 4338-4345
-
-
Gravatt, G.L.1
Baguley, B.C.2
Wilson, W.R.3
Denny, W.A.4
-
4
-
-
0001325629
-
Substituted 2,50-bi-1Hbenzimidazoles: Topoisomerase i inhibition and cytotoxicity
-
Kim, J. S.; Gatto, B.; Yu, C.; Liu, A.; Liu, L. F.; LaVoie, E. J. Substituted 2,50-bi-1Hbenzimidazoles: Topoisomerase I inhibition and cytotoxicity. J. Med. Chem. 1996, 39, 992-998.
-
(1996)
J. Med. Chem.
, vol.39
, pp. 992-998
-
-
Kim, J.S.1
Gatto, B.2
Yu, C.3
Liu, A.4
Liu, L.F.5
Lavoie, E.J.6
-
5
-
-
0031463691
-
Synthesis and biological activity of novel nonnucleoside inhibitors of HIV-1 reverse transcriptase: 2-Aryl-substituted benzimidazoles
-
Roth, T.; Morningstar, M. L.; Boyer, P. L.; Hughes, S. H.; Buckheit Jr., R. W.; Michejda, C. J. Synthesis and biological activity of novel nonnucleoside inhibitors of HIV-1 reverse transcriptase: 2-Aryl-substituted benzimidazoles. J. Med. Chem. 1997, 40, 4199-4207.
-
(1997)
J. Med. Chem.
, vol.40
, pp. 4199-4207
-
-
Roth, T.1
Morningstar, M.L.2
Boyer, P.L.3
Hughes, S.H.4
Buckheit Jr., R.W.5
Michejda, C.J.6
-
6
-
-
33947458464
-
The chemistry of the benzimidazoles
-
Wright, J. B. The chemistry of the benzimidazoles. Chem. Rev. 1951, 48, 397-541.
-
(1951)
Chem. Rev.
, vol.48
, pp. 397-541
-
-
Wright, J.B.1
-
7
-
-
0017872205
-
Diarylamidine derivatives with one or both of the aryl moieties consisting of an indole or indole-like ring: Inhibitors of arginine-specific esteroproteases
-
Tidwell, R. R.; Geratz, J. D.; Dann, O.; Volz, G.; Zeh, D.; Loewe, H. Diarylamidine derivatives with one or both of the aryl moieties consisting of an indole or indole-like ring: Inhibitors of arginine-specific esteroproteases. J. Med. Chem. 1978, 21, 613-623
-
(1978)
J. Med. Chem.
, vol.21
, pp. 613-623
-
-
Tidwell, R.R.1
Geratz, J.D.2
Dann, O.3
Volz, G.4
Zeh, D.5
Loewe, H.6
-
8
-
-
0027253921
-
Structure DNA minor groove binding, and base pair specificity of alkyl- and aryl-linked bis(amidinobenzimidazoles) and bis(amidinoindoles)
-
Fairley, T. A.; Tidwell, R. R.; Donkor, I.; Naiman, N. A.; Ohemeng, K. A.; Lombardy, R. J.; Bentley, J. A.; Cory, M. Structure, DNA minor groove binding, and base pair specificity of alkyl- and aryl-linked bis(amidinobenzimidazoles) and bis(amidinoindoles). J. Med. Chem. 1993, 36, 1746-1753.
-
(1993)
J. Med. Chem.
, vol.36
, pp. 1746-1753
-
-
Fairley, T.A.1
Tidwell, R.R.2
Donkor, I.3
Naiman, N.A.4
Ohemeng, K.A.5
Lombardy, R.J.6
Bentley, J.A.7
Cory, M.8
-
9
-
-
0032500083
-
Trois Nouvelles Voies de Synthesis des Derives 1, 3-Azoliques Sous Micro-ondes
-
Bourgrin, K.; Loupy, A.; Soufiaoui, M. Trois Nouvelles Voies de Synthesis des Derives 1, 3-Azoliques Sous Micro-ondes. Tetrahedron 1998, 54, 8055-8064.
-
(1998)
Tetrahedron
, vol.54
, pp. 8055-8064
-
-
Bourgrin, K.1
Loupy, A.2
Soufiaoui, M.3
-
10
-
-
0030300024
-
[125I=127I] IodoHoechst 33342: Synthesis, DNA binding, and biodistribution
-
Harapanhalli, R. S.; McLaughlin, L. W.; Howell, R. W.; Rao, D. V.; Adelstein, S. J.; Kassis, A. I. [125I=127I]IodoHoechst 33342: Synthesis, DNA binding, and biodistribution. J. Med. Chem. 1996, 39, 4804-4809.
-
(1996)
J. Med. Chem.
, vol.39
, pp. 4804-4809
-
-
Harapanhalli, R.S.1
McLaughlin, L.W.2
Howell, R.W.3
Rao, D.V.4
Adelstein, S.J.5
Kassis, A.I.6
-
11
-
-
77956216179
-
Development of serine protease inhibitors displaying a multicentered short (van den Eynde, J. J.; Delfosse, F.; Lor, P.; Van Haverbeke, Y.A mild catalyst for the formation of carbon-nitrogen bonds
-
Verner, E.; Katz, B. A.; Spencer, J. R.; Allen, D.; Hataye, J.; Hruzewicz, W.; Hui, H. C.; Kolesnikov, A.; Li, Y.; Luong, C.; Martelli, A.; Radika, K.; Rai, R.; She, M.; Shrader, W.; Sprengeler, P. A.; Trapp, S.; Wang, J.; Young, W. B.; Mackman, R. L. Development of serine protease inhibitors displaying a multicentered short (van den Eynde, J. J.; Delfosse, F.; Lor, P.; van Haverbeke, Y.A mild catalyst for the formation of carbon-nitrogen bonds.Tetrahedron1995,51,5813-5818
-
(1995)
Tetrahedron
, vol.51
, pp. 5813-5818
-
-
Verner, E.1
Katz, B.A.2
Spencer, J.R.3
Allen, D.4
Hataye, J.5
Hruzewicz, W.6
Hui, H.C.7
Kolesnikov, A.8
Li, Y.9
Luong, C.10
Martelli, A.11
Radika, K.12
Rai, R.13
She, M.14
Shrader, W.15
Sprengeler, P.A.16
Trapp, S.17
Wang, J.18
Young, W.B.19
MacKman, R.L.20
more..
-
12
-
-
0029061671
-
A mild catalyst for the formation of carbon-nitrogen bonds
-
van den Eynde, J. J.; Delfosse, F.; Lor, P.; van Haverbeke, Y. A mild catalyst for the formation of carbon-nitrogen bonds. Tetrahedron 1995, 51, 5813-5818.
-
(1995)
Tetrahedron
, vol.51
, pp. 5813-5818
-
-
Van Den Eynde, J.J.1
Delfosse, F.2
Lor, P.3
Van Haverbeke, Y.4
-
13
-
-
0026596081
-
Dehydrogenations using benzofuroxan as oxidant
-
Patzold, F.; Zeuner, F.; Heyer, T. H.; Niclas, H.-J. Dehydrogenations using benzofuroxan as oxidant. Synth. Commun. 1992, 22, 281-284.
-
(1992)
Synth. Commun.
, vol.22
, pp. 281-284
-
-
Patzold, F.1
Zeuner, F.2
Heyer, T.H.3
Niclas, H.-J.4
-
14
-
-
0000586488
-
Development of new and efficient polymer-supported hypervalent iodine reagents
-
Bhatnagar, I.; George, M. V. Development of new and efficient polymer-supported hypervalent iodine reagents. Tetrahedron 1968, 24, 1293-1296.
-
(1968)
Tetrahedron
, vol.24
, pp. 1293-1296
-
-
Bhatnagar, I.1
George, M.V.2
-
15
-
-
0003140019
-
One-step high-throughput synthesis of benzimidazoles
-
Stephens, F. F.; Bower, J. D. One-step high-throughput synthesis of benzimidazoles. J. Chem. Soc. 1949, 2971-2976.
-
(1949)
J. Chem. Soc.
, pp. 2971-2976
-
-
Stephens, F.F.1
Bower, J.D.2
-
16
-
-
0043240483
-
Practical oxone-mediated, high-throughput, solution-phase synthesis of benzimidazolesfrom 1,2-phenylenediamines and aldehydes and its application to preparative-scale synthesis
-
Beaulieu, P. L.; Hache, B.; von Moos, E. A. Practical oxone-mediated, high-throughput, solution-phase synthesis of benzimidazolesfrom 1,2-phenylenediamines and aldehydes and its application to preparative-scale synthesis. Synthesis 2003, 11, 1683-1692.
-
(2003)
Synthesis
, vol.11
, pp. 1683-1692
-
-
Beaulieu, P.L.1
Hache, B.2
Von Moos, E.A.3
-
17
-
-
0035191889
-
A short synthesis of the PARP inhibitor 2-(4-trifluoro methylphenyl)benzimidazole-4-carboxamide
-
Austen, S. C.; Kane, J. M. A short synthesis of the PARP inhibitor 2-(4-trifluoro methylphenyl)benzimidazole-4-carboxamide. J. Heterocycl. Chem. 2001, 38, 979-980.
-
(2001)
J. Heterocycl. Chem.
, vol.38
, pp. 979-980
-
-
Austen, S.C.1
Kane, J.M.2
-
18
-
-
0029983537
-
Synthesis and DNA interactions of benzimidazole dications which have activity against opportunistic infections
-
Lombardy, R. L.; Tanious, F. A.; Ramachandran, K.; Tidwell, R. R.; Wilson, W. D. Synthesis and DNA interactions of benzimidazole dications which have activity against opportunistic infections. J. Med. Chem. 1996, 39, 1452-1462.
-
(1996)
J. Med. Chem.
, vol.39
, pp. 1452-1462
-
-
Lombardy, R.L.1
Tanious, F.A.2
Ramachandran, K.3
Tidwell, R.R.4
Wilson, W.D.5
-
19
-
-
19544370229
-
A simple and efficient procedure for the synthesis of benzimidazoles using air as the oxidant
-
Lin, S.; Yang, L. H. A simple and efficient procedure for the synthesis of benzimidazoles using air as the oxidant. Tetrahedron Lett. 2005, 46, 4315-4319.
-
(2005)
Tetrahedron Lett.
, vol.46
, pp. 4315-4319
-
-
Lin, S.1
Yang, L.H.2
-
20
-
-
0037631073
-
Synthèse chimiosélective des benzimidazoles sur silice traitée par le chlorure du thionyle
-
Abdelkrim, B. A.; Bakkas, S.; Soufiaoui, M. Synthèse chimiosélective des benzimidazoles sur silice traitée par le chlorure du thionyle. Tetrahedron Lett. 2003, 44, 5935-5937.
-
(2003)
Tetrahedron Lett.
, vol.44
, pp. 5935-5937
-
-
Abdelkrim, B.A.1
Bakkas, S.2
Soufiaoui, M.3
-
21
-
-
0038368363
-
Cyclodehydrogenation of N-benzylidene-o-phenylenediamines to 220-diaryl-110-bibenzimidazoles with dioxygen catalyzed by copper(I) chloride in pyridine: A structural study of 2,20-bis-( 3,4,5-trimethoxyphenyl)-1,10- bibenzimidazole
-
Speier, G.; Parkanyi, L. Cyclodehydrogenation of N-benzylidene-o- phenylenediamines to 2,20-diaryl-1,10-bibenzimidazoles with dioxygen catalyzed by copper(I) chloride in pyridine: A structural study of 2,20-bis-(3,4,5- trimethoxyphenyl)-1,10-bibenzimidazole. J. Org. Chem. 1986, 51, 218-221.
-
(1986)
J. Org. Chem.
, vol.51
, pp. 218-221
-
-
Speier, G.1
Parkanyi, L.2
-
22
-
-
0032500083
-
Trois Nouvelles Voies de Synthesis des Derives 1, 3-Azoliques Sous Micro-ondes
-
Bougrin, K.; Loupy, A.; Soufiaoui, M. Trois Nouvelles Voies de Synthesis des Derives 1, 3-Azoliques Sous Micro-ondes. Tetrahedron 1998, 54, 8055-8057.
-
(1998)
Tetrahedron
, vol.54
, pp. 8055-8057
-
-
Bougrin, K.1
Loupy, A.2
Soufiaoui, M.3
-
23
-
-
0027769722
-
A novel palladium-catalyzed synthesis of 2-arylbenzimidazoles
-
Perry, R. J.; Wilson, B. D. A novel palladium-catalyzed synthesis of 2-arylbenzimidazoles. J. Org. Chem. 1993, 58, 7016-7021.
-
(1993)
J. Org. Chem.
, vol.58
, pp. 7016-7021
-
-
Perry, R.J.1
Wilson, B.D.2
-
24
-
-
0000691918
-
Heterocycles from N-ethoxycarbonyl thioamides and dinucleophilic reagents 2: Five-membered rings containing two heteroatoms at 1,3- positions
-
George, B.; Papadopoulos, E. P. Heterocycles from N-ethoxycarbonyl thioamides and dinucleophilic reagents, 2: Five-membered rings containing two heteroatoms at 1,3- positions. J. Org. Chem. 1977, 42, 441-443.
-
(1977)
J. Org. Chem.
, vol.42
, pp. 441-443
-
-
George, B.1
Papadopoulos, E.P.2
|