Novel interpenetrating network microspheres of xanthan gumpoly(vinyl alcohol) for the delivery of diclofenac sodium to the intestinein vitro and in vivo evaluation

Drug Delivery

Volumn 17, Issue 7, 2010, Pages 508-519

  Ray, Somasree ^a   Banerjee, Subham ^a   Maiti, Sabyasachi ^a   Laha, Bibek ^a   Barik, Saikat ^a   Sa, Biswanath ^b   Bhattacharyya, Uttam Kumar ^a  

^a GUPTA COLLEGE OF TECHNOLOGICAL SCIENCES   (India)

^b JADAVPUR UNIVERSITY   (India)

Author keywords

Diclofenac sodium; Microspheres; Poly (vinyl alcohol); Prolonged release; Xanthan gum

Indexed keywords

DICLOFENAC; GLUTARALDEHYDE; INTERPENETRATING NETWORK MICROSPHERE; MICROSPHERE; POLYVINYL ALCOHOL; UNCLASSIFIED DRUG; XANTHAN;

ANIMAL EXPERIMENT; AREA UNDER THE CURVE; ARTICLE; CONTROLLED RELEASE FORMULATION; CROSS LINKING; DRUG BLOOD LEVEL; DRUG DELIVERY SYSTEM; DRUG ELIMINATION; DRUG HALF LIFE; DRUG RELEASE; DRUG STABILITY; EMULSION; EVALUATION; MAXIMUM PLASMA CONCENTRATION; MICROENCAPSULATION; NONHUMAN; PARTICLE SIZE; PRIORITY JOURNAL; TIME TO MAXIMUM PLASMA CONCENTRATION;

ANIMALS; CALORIMETRY, DIFFERENTIAL SCANNING; DELAYED-ACTION PREPARATIONS; DICLOFENAC; DRUG DELIVERY SYSTEMS; FEMALE; HYDROGEN-ION CONCENTRATION; INTESTINES; MALE; MICROSCOPY, ELECTRON, SCANNING; MICROSPHERES; POLYSACCHARIDES, BACTERIAL; POLYVINYL ALCOHOL; RABBITS; SPECTROSCOPY, FOURIER TRANSFORM INFRARED; X-RAY DIFFRACTION;

EID: 77956146525     PISSN: 10717544     EISSN: 15210464     Source Type: Journal    
DOI: 10.3109/10717544.2010.483256     Document Type: Article

References (32)

1. Agnihotri, S.A., Aminabhavi, T.M. (2004a). Controlled release of clozapine through chitosan microparticles prepared by a novel method. J Contr Rel. 96:245-259
2. Agnihotri, S.A., Aminabhavi, T.M. (2004b). Formulation and evaluation of novel tableted chitosan microparticles for the controlled release of clozapine. J. Microencapsul. 21:709-718
3. Agnihotri, S.A., Aminabhavi, T.M. (2005). Development of novel interpenetrating network gellan gum-poly(vinyl alcohol) hydrogel microspheres for the controlled release of carvedilol. Drug Dev Ind Pharm. 31:491-503.
4. Al-Saidan, S.M., Krishnaiah, Y.S.R., Patro, S.S., Satyanaryana, V. (2005). In vitro and in vivo evaluation of guar gum matrix tablets for oral controlled release of water-soluble diltiazem hydrochloride. AAPS Pharm SciTech. 6:Article 5, E14-21.
5. Burugapalli, K., Bhatia, D., Koul, V., Choudhary, V. (2001). Interpenetrating polymer networks based on poly(acrylic acid) and gelatin. I: swelling and thermal behavior. J Appl Polym Sci. 82:217-227
6. Chandy, T., Wilson, R.F., Rao, G.H., Das, G.S. (2002). Changes in cisplatin delivery due to surface-coated poly(lactic acid)-poly(epsilon- caprolactone) microspheres. J Biomater Applic. 16: 275-291
7. Corradini, E., Pineda, E.A.G., Hechenleitner, A.A.W. (1999). Lignin-poly (vinyl alcohol) blends studied by thermal analysis. Polym Degrad Stabil. 66:199-208.
8. Desai, K.G.H. (2005). Preparation and characteristics of high-amylose corn starch/pectin blend microparticles: a technical note. AAPS Pharm. SciTech. 6:Article 30, E202-208.
9. Giagoudakis, G., Markantonis, S.L. (1998). An alternative high-performance liquid-chromatographic method for the determination of diclofenac and furbiprofen in plasma. J Pharm Biomed Anal. 17:897-901.
10. Gibaldi, M., Perrier, D. (1990). Pharmacokinetics. New York: Marcel Dekker.
11. Hejazi, R., Amiji, M. (2003). Chitosan based gastrointestinal delivery systems. J Contr Rel. 89:151-165
12. Itokazu, M., Yamemoto, K., Yang, W.Y., Aoki, T., Kato, N., Watanabe, K. (1997). The sustained release of antibiotics from freezedried fbrin-antibiotic compound and efcacies in rat model of osteomyelitis. Infection. 25:359-363
13. Katzbauer, B. (1998). Properties and applications of xanthan gum. Polym Degrad Stabil. 59:81-84
14. Kawaguchi, H. (2000). Functional polymer microspheres. Prog Polym Sci. 25:1171-1210
15. Korsmeyer, R.C., Peppas, N.A. (1981). Efect of the morphology of hydrophilic polymeric matrices on the difusion and release of water-soluble drugs. J Memb Sci. 9:211-227
16. Kottke, M.K., Rhodes, C.T. (1991). Limitations of presently available in vitro release data for the prediction of in vivo performance. Drug Dev Ind Pharm. 17:1157-1176
17. Kurkuri, M.D., Aminabhavi, T.M. (2004). Poly(vinyl alcohol) and poly(acrylic acid) sequential interpenetrating network pH sensitive microspheres for the delivery of diclofenac sodium to the intenstine. J Contr Rel. 96:9-20.
18. Peppas, N.A., Wright, S.L. (1998). Drug difusion and binding in ion-izable interpenetrating networks from poly(vinyl alcohol) and poly(acrylic acid). Eur J Pharm Biopharm. 4:15-29.
19. Piyakulawat, P., Praphairaksit, N., Chantarasiri, N., Muangsin, N. (2007). Preparation and evaluation of chitosan/carrageenan beads for controlled release of sodium diclofenac. AAPS Pharm.SciTech. 8:Article 97, E1-11.
20. Ray, S., Maiti, S., Sa, B. (2008). Preliminary investigation on the development of diltiazem resin complex loaded carboxymethyl xan-than beads. AAPS Pharm Sci Tech. 9:295-300.
21. Ritger, P.L., Peppas, N.A. (1987). A simple equation for description of solute release. II. Fickian and anomalous release from swellable devices. J Contr Rel. 5:37-42.
22. Rokhade, A.P., Agnihotri, S.A., Patil, S.A., Mallikarjuna, N.N., Kulkarni, P.V., Aminabhavi, T.M. (2006). Semi-interpenetrating polymer network microspheres of gelatin and sodium car-boxymethyl cellulose for controlled release of ketorolac trometh-amine. Carbohyd Polym. 65:243-252
23. Rokhade, A.P., Shelke, N.B., Patil, S.A., Aminabhavi, T.M. (2007). Novel interpenetrating polymer network microspheres of chitosan and methylcellulose for controlled release of theophylline. Carbohyd Polym. 69:678-687
24. Rowland, M., Tozer, T.N. (1996). Clinical pharmacokinetics: Concepts and applications. New Delhi, India: BI Waverly Pvt Ltd, 469-472
25. Santos, H., Veiga, F., Pina, M.E., Sousa, J.J. (2005). Compaction, compression and drug release properties of diclofenac sodium and ibuprofen pellets comprising xanthan gum as a sustained release agent. Int J Pharm. 295:17-27.
26. Soppimath, K.S., Aminabhavi, T.M. (2002). Water transport and drug release study from crosslinked polyacrylamide-grafted-guar gum hydrogel microspheres for the controlled release application. Eur J Pharm Biopharm. 53:87-98.
27. Soppimath, K.S., Kulkarni, A.R., Aminabhavi, T.M. (2000). Controlled release of antihypertensive drug from the interpenetrating network poly(vinyl alcohol)-guar gum hydrogel microspheres. J Biomater Sci Polym Ed. 11:27-43.
28. Sujja-areevath, J., Munday, D.L., Cox, P.J., Khan, K.A. (1996). Release characteristics of diclofenac sodium from encapsulated natural gum mini-matrix formulations. Int J Pharm. 139: 53-62.
29. Talukdar, M.M., Kinget, R. (1995). Swelling and drug release behaviour of xanthan gum tablets. Int J Pharm. 120:63-72.
30. Tanoo, B.C., Sunny, M.C., Jayakrishnan, A. (1993). Oral sustained release drug delivery systems using polycarbonate micro-spheres capable of foating on gastric fuid. J Pharm Pharmacol. 45:21-24
31. Tudja, P., Khan, M.Z.I., Mstrovíc, E., Horvat, M., Golja, P. (2001). Termal behaviour of diclofenac sodium: decomposition and melting characteristics. Chem Pharm Bull. 49:1245-1250
32. nd ed. Washington: American Pharmaceutical Association/London: Pharmaceutical Press, 562-563