Selection, preparation, and evaluation of small-molecule inhibitors of toll-like receptor 4

ACS Medicinal Chemistry Letters

Volumn 1, Issue 5, 2010, Pages 194-198

  Bevan, Douglas E ^a   Martinko, Alexander J ^a   Loram, Lisa C ^a   Stahl, Joshua A ^a   Taylor, Frederick R ^a   Joshee, Sampada ^a   Watkins, Linda R ^a   Yin, Hang ^a  

^a UNIVERSITY OF COLORADO   (United States)

Author keywords

[No Author keywords available]

Indexed keywords

MORPHINE; PROTEIN MD 2; PYRAZOLE; RECEPTOR BLOCKING AGENT; TOLL LIKE RECEPTOR 1; TOLL LIKE RECEPTOR 2; TOLL LIKE RECEPTOR 3; TOLL LIKE RECEPTOR 4; TOLL LIKE RECEPTOR 4 INHIBITOR; TOLL LIKE RECEPTOR 6; TOLL LIKE RECEPTOR 7; UNCLASSIFIED DRUG;

ANALGESIA; ANIMAL CELL; ARTICLE; CONTROLLED STUDY; DRUG POTENCY; DRUG RECEPTOR BINDING; DRUG SCREENING; DRUG SELECTIVITY; DRUG SYNTHESIS; ENANTIOSELECTIVITY; HUMAN; HUMAN CELL; IN VIVO STUDY; MANNICH REACTION; MOLECULAR DOCKING; NONHUMAN; PRIORITY JOURNAL; RECEPTOR UPREGULATION;

ANIMALIA;

EID: 77956141419     PISSN: None     EISSN: 19485875     Source Type: Journal    
DOI: 10.1021/ml100041f     Document Type: Article

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