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Bioorganic and Medicinal Chemistry Letters

Volumn 20, Issue 17, 2010, Pages 5143-5146

Fluorescent retinoid X receptor ligands for fluorescence polarization assay

(9) Yamada, Shoya a Ohsawa, Fuminori a,b Fujii, Shuji a Shinozaki, Ryosuke a Makishima, Makoto c Naitou, Hirotaka d Enomoto, Shuichi a,b Tai, Akihiro e Kakuta, Hiroki a

a OKAYAMA UNIVERSITY (Japan)

b RIKEN (Japan)

c NIHON UNIVERSITY (Japan)

d UNIVERSITY OF SHIZUOKA (Japan)

e PREFECTURAL UNIVERSITY OF HIROSHIMA (Japan)

Author keywords

Carbostyril; Fluorescence polarization; Molecular design; Retinoid X receptor

Indexed keywords

6 [ETHYL (1 ISOBUTYL 2 OXO 4 TRIFLUOROMETHYL 1,2 DIHYDROQUINOLIN 7 YL) AMINO] NICOTINIC ACID; BEXAROTENE; CARBOSTYRIL DERIVATIVE; NICOTINIC ACID DERIVATIVE; RETINOID X RECEPTOR; UNCLASSIFIED DRUG;

ARTICLE; DRUG DESIGN; DRUG STRUCTURE; DRUG SYNTHESIS; FLUORESCENCE POLARIZATION; HIGH THROUGHPUT SCREENING; LIPOPHILICITY;

DIMERIZATION; FLUORESCENCE POLARIZATION; LIGANDS; RETINOID X RECEPTORS;

EID: 77955661848 PISSN: 0960894X EISSN: None Source Type: Journal
DOI: 10.1016/j.bmcl.2010.07.011 Document Type: Article

Times cited : (11)

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