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Volumn 1, Issue 1, 2010, Pages 54-60

Design, synthesis, and structure-activity relationships of indole-3-carboxamides as novel water soluble cannabinoid CB1 receptor agonists

(21) Adam, Julia M a Cairns, Jim a Caulfield, Wilson a Cowley, Phillip a Cumming, Iain a Easson, Morag a Edwards, Darren a Ferguson, Morag a Goodwin, Richard a Jeremiah, Fiona a Kiyoi, Takao a Mistry, Ashvin a Moir, Elizabeth a Morphy, Richard a Tierney, Jason a York, Mark a Baker, James a Cottney, Jean E a Houghton, Andrea K a Westwood, Paul J a Walker, Glenn a more..

a Schering Plough Research Institute (United Kingdom)

Author keywords

[No Author keywords available]

Indexed keywords

CANNABINOID 1 RECEPTOR; CANNABINOID 1 RECEPTOR AGONIST; CANNABINOID 2 RECEPTOR; ORG 28312; ORG 28611; UNCLASSIFIED DRUG;

ANALGESIC ACTIVITY; ANIMAL CELL; ANIMAL EXPERIMENT; ARTICLE; DOSE RESPONSE; DRUG BLOOD LEVEL; DRUG BRAIN LEVEL; DRUG CLEARANCE; DRUG DESIGN; DRUG METABOLISM; DRUG RECEPTOR BINDING; DRUG SOLUBILITY; DRUG STABILITY; DRUG SYNTHESIS; HUMAN; HUMAN CELL; MOUSE; NONHUMAN; PAIN; PRIORITY JOURNAL; STRUCTURE ACTIVITY RELATION;

EID: 77955426051 PISSN: 20402503 EISSN: 20402511 Source Type: Journal
DOI: 10.1039/c0md00022a Document Type: Article

Times cited : (31)

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