Structure-activity relationship of indoline-2-carboxylic acid N-(substituted)phenylamide derivatives

Bioorganic and Medicinal Chemistry Letters

Volumn 20, Issue 15, 2010, Pages 4620-4623

  Kwak, Jae Hwan ^a   Kim, Yoseob ^a   Park, Hyunjeong ^a   Jang, Jae Yong ^a   Lee, Keun Kuk ^a   Yi, Wonhui ^a   Kwak, Jeong Ah ^a   Park, Song Gyu ^b   Kim, Hwanmook ^b   Lee, Kiho ^b   Kang, Jong Soon ^b   Han, Sang Bae ^a   Hwang, Bang Yeon ^a   Hong, Jin Tae ^a   Jung, Jae Kyung ^a   Kim, Youngsoo ^a   Cho, Jungsook ^c   Lee, Heesoon ^a  

^a Chungbuk National University   (South Korea)

^b Korea Research Institute of Bioscience and Biotechnology (KRIBB)   (South Korea)

^c Dongguk University   (South Korea)

Author keywords

Cytotoxic activity; Indoline 2 carboxamide; NF B inhibitors

Indexed keywords

ANILIDE; ANTINEOPLASTIC AGENT; CYTOTOXIC AGENT; IMMUNOGLOBULIN ENHANCER BINDING PROTEIN;

AMIDATION; ARTICLE; CANCER CELL CULTURE; CYTOTOXICITY; DRUG POTENCY; DRUG SYNTHESIS; GENETIC TRANSCRIPTION; HUMAN; HUMAN CELL; STRUCTURE ACTIVITY RELATION;

ANTINEOPLASTIC AGENTS; BENZYLAMINES; CELL LINE, TUMOR; CHROMANS; DRUG SCREENING ASSAYS, ANTITUMOR; HUMANS; INDOLES; NF-KAPPA B; STRUCTURE-ACTIVITY RELATIONSHIP;

EID: 77955418470     PISSN: 0960894X     EISSN: None     Source Type: Journal    
DOI: 10.1016/j.bmcl.2010.06.004     Document Type: Article

References (14)

1. T.D. Gilmore Oncogene 18 1999 6842
2. M.S. Hayden, and S. Ghosh Gene Dev. 18 2004 2195
3. T.D. Gilmore Oncogene 25 2006 6680
4. A. Israel, O. Le Bail, D. Hatat, J. Piette, M. Kieran, F. Logeat, D. Wallach, M. Fellous, and P. Kourilsky EMBO J. 8 1989 3793
5. L. Osborn, S. Kunkel, and G.J. Nabel Proc. Natl. Acad. Sci. U.S.A. 86 1989 2336
6. C. Michiels, E. Minet, D. Mottet, and M. Raes Free Radical Biol. Med. 33 2002 1231
7. N.D. Perkins, and T.D. Gilmore Cell Death Differ. 13 2006 759
8. B.H. Kim, A.M. Reddy, K.H. Lee, E.Y. Chung, S.M. Cho, H. Lee, K.R. Min, and Y. Kim Biochem. Biophys. Res. Commun. 325 2004 223
9. J.H. Kwak, B.H. Kim, J.K. Jung, Y. Kim, J. Cho, and H. Lee Arch. Pharm. Res. 30 2007 1210
10. J.H. Kwak, S.W. Won, T.J. Kim, E. Roh, H.Y. Kang, H.W. Lee, J.K. Jung, B.Y. Hwang, Y. Kim, J. Cho, and H. Lee Arch. Pharm. Res. 31 2008 133
11. J.H. Kwak, S.W. Won, T.J. Kim, W. Yi, E.H. Choi, S.C. Kim, H. Park, E. Roh, J.K. Jung, B.Y. Hwang, J.T. Hong, Y. Kim, J. Cho, and H. Lee Arch. Pharm. Res. 32 2009 167
12. Z. Gan, P.T. Reddy, S. Quevillon, S. Couve-Bonnaire, and P. Arya Angew. Chem., Int. Ed. 44 2005 1366
13. R.R. Poondra, N.N. Kumar, K. Bijian, M. Prakesch, V. Campagna-Slater, A. Reayi, P.T. Reddy, A. Choudhry, M.L. Barnes, D.M. Leek, M. Daroszewska, C. Lougheed, B. Xu, M. Schapira, M.A. Alaoui-Jamili, and P. Arya J. Comb. Chem. 11 2009 303
14. F.H. Sarkar, Y. Li, Z. Wang, and D. Kong Int. Rev. Immunol. 27 2008 293