Genomic action of permanently charged tamoxifen derivatives via estrogen receptor-α

Bioorganic and Medicinal Chemistry

Volumn 18, Issue 15, 2010, Pages 5593-5601

  Rivera Guevara, Claudia ^a   Pérez Alvarez, Víctor ^a   García Becerra, Rocío ^b   Ordaz Rosado, David ^b   Morales Ríos, Martha Sonia ^a   Hernández Gallegos, Elizabeth ^a   Cooney, Austin J ^c   Bravo Gómez, María Elena ^d   Larrea, Fernando ^b   Camacho, Javier ^a  

^a DEPARTAMENTO DE FÍSICA   (Mexico)

^b INSTITUTO NACIONAL DE CIENCIAS MÉDICAS Y NUTRICIÓN SALVADOR ZUBIRÁN   (Mexico)

^c BAYLOR COLLEGE OF MEDICINE   (United States)

^d UNIVERSIDAD NACIONAL AUTÓNOMA DE MÉXICO   (Mexico)

Author keywords

Breast cancer; Estrogen receptor; Genomic action; Tamoxifen; Tamoxifen derivatives

Indexed keywords

ANTINEOPLASTIC AGENT; ESTROGEN RECEPTOR ALPHA; PERMANENTLY CHARGED TAMOXIFEN DERIVATIVE; SELECTIVE ESTROGEN RECEPTOR MODULATOR; TAMOXIFEN; TAMOXIFEN BUTYL BROMIDE; TAMOXIFEN DERIVATIVE; TAMOXIFEN ETHYL BROMIDE; TAMOXIFEN ISOPROPYL BROMIDE; TAMOXIFEN METHYL BROMIDE; TAMOXIFEN METHYL IODIDE; TAMOXIFEN PROPYL BROMIDE; UNCLASSIFIED DRUG; ANTINEOPLASTIC HORMONE AGONISTS AND ANTAGONISTS; PROTEIN BINDING;

ANTINEOPLASTIC ACTIVITY; ARTICLE; CELL PROLIFERATION; CELL STRAIN MCF 7; DRUG MECHANISM; DRUG RECEPTOR BINDING; DRUG STRUCTURE; ELECTRON MICROSCOPY; FEMALE; GENETIC TRANSCRIPTION; HELA CELL; HIGH PERFORMANCE LIQUID CHROMATOGRAPHY; HUMAN; HUMAN CELL; HUMAN CELL CULTURE; LIQUID CHROMATOGRAPHY; MASS SPECTROMETRY; NUCLEAR MAGNETIC RESONANCE; PHARMACOGENETICS; STRUCTURE ACTIVITY RELATION; UTERINE CERVIX CANCER; X RAY DIFFRACTION; CHEMISTRY; CONFORMATION; DRUG EFFECTS; GENETICS; METABOLISM; TUMOR CELL LINE; X RAY CRYSTALLOGRAPHY;

ANTINEOPLASTIC AGENTS, HORMONAL; CELL LINE, TUMOR; CRYSTALLOGRAPHY, X-RAY; ESTROGEN RECEPTOR ALPHA; HUMANS; MOLECULAR CONFORMATION; PROTEIN BINDING; STRUCTURE-ACTIVITY RELATIONSHIP; TAMOXIFEN; TRANSCRIPTION, GENETIC;

EID: 77955413286     PISSN: 09680896     EISSN: None     Source Type: Journal    
DOI: 10.1016/j.bmc.2010.06.039     Document Type: Article

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