New 6-amino-[1,2,4]triazolo[3,4-b][1,3,4]thiadiazines and [1,2,4]triazolo[3,4-b] [1,3,4]thiadiazin-6-ones: Synthesis, characterization and antibacterial activity evaluation

European Journal of Medicinal Chemistry

Volumn 45, Issue 7, 2010, Pages 3191-3195

  Almajan, Gabriela Laura ^a   Barbuceanu, Stefania Felicia ^a   Saramet, Ioana ^a   Draghici, Constantin ^b  

^a CAROL DAVILA UNIVERSITY OF MEDICINE AND PHARMACY   (Romania)

^b INSTITUTE OF ORGANIC CHEMISTRY   (Romania)

Author keywords

Amino triazolothiadiazines; Antibacterial activity; Cyclodehydration; Triazolothiadiazinones

Indexed keywords

1,2,4 TRIAZOLE DERIVATIVE; 2 CHLORO N PHENYLACETAMIDE; 3 [ 4 ( 4 BROMOPHENYLSULFONYL)PHENYL] 5H [ 1,2,4 ]TRIAZOLO[ 3,4 B][ 1,3,4 ]THIADIAZINE 6,7 DIONE; 3 [ 4 ( 4 HYDROPHENYLSULFONYL)PHENYL] 5H [ 1,2,4 ]TRIAZOLO] 3,4 B][ 1,3,4 ]THIADIAZIN 6 (7H) ONE; 4 AMINO 5 [ 4 ( 4 BROMOPHENYLSULFONYL)PHENYL] 4H 1,2,4 TRIAZOLE 3 THIOL; 4 AMINO 5 [ 4 ( 4 CHLOROPHENYLSULFONYL)PHENYL] 4H 1,2,4 TRIAZOLE 3 THIOL; 4 AMINO 5 [ 4 ( 4 HYDROPHENYLSULFONYL)PHENYL] 4H 1,2,4 TRIAZOLE 3 THIOL; ACETAMIDE DERIVATIVE; AMPICILLIN; BROMINE; BROMODIETHYLMALONATE; CHLORIDE; CHLORINE; CHLOROACETIC ACID; HYDROGEN; MALONIC ACID DERIVATIVE; OXALYLCHLORIDE; TETRACYCLINE; THIADIAZINE DERIVATIVE; TRIAZOLE DERIVATIVE; UNCLASSIFIED DRUG;

ANTIBACTERIAL ACTIVITY; ARTICLE; BACTERIAL STRAIN; CONTROLLED STUDY; DRUG STRUCTURE; DRUG SYNTHESIS; ESCHERICHIA COLI; INFRARED SPECTROSCOPY; INTERMOLECULAR CONDENSATION REACTION; MINIMUM INHIBITORY CONCENTRATION; NONHUMAN; NUCLEAR MAGNETIC RESONANCE SPECTROSCOPY; POLYMERIZATION; PSEUDOMONAS AERUGINOSA; STAPHYLOCOCCUS AUREUS; STAPHYLOCOCCUS EPIDERMIDIS;

EID: 77954349618     PISSN: 02235234     EISSN: 17683254     Source Type: Journal    
DOI: 10.1016/j.ejmech.2010.02.057     Document Type: Article

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