Diversity-oriented pyrazol-3-one synthesis based on hydrazinodipeptide-like units prepared via the Ugi reaction

Tetrahedron Letters

Volumn 51, Issue 31, 2010, Pages 4095-4099

  Lakontseva, Ekaterina ^a,b   Krasavin, Mikhail ^a,b  

^a YAROSLAVL STATE PEDAGOGICAL UNIVERSITY   (Russian Federation)

^b Chemical Diversity Research Institute   (Russian Federation)

Author keywords

Diversity oriented synthesis; Hydrazino Ugi reaction; Monoalkylated pyrazol 3 ones; Multi component reactions; Peptidomimetics; Post Ugi modifications

Indexed keywords

ACETIC ACID DERIVATIVE; HYDRAZINE DERIVATIVE; PEPTIDE DERIVATIVE; PYRAZOLONE; TRIFLUOROACETIC ACID;

ARTICLE; CHEMICAL REACTION; CYCLIZATION; DRUG STRUCTURE; DRUG SYNTHESIS; HYDROGEN BOND; TEMPERATURE; UGI REACTION;

EID: 77953961000     PISSN: 00404039     EISSN: None     Source Type: Journal    
DOI: 10.1016/j.tetlet.2010.05.133     Document Type: Article

References (8)

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8. 3: C, 52.30; H, 6.45; N, 14.35. Found: C, 52.38; H, 6.46; N, 14.41.