Crystallo-co-agglomeration: A novel particle engineering technique

Asian Journal of Pharmaceutics

Volumn 4, Issue 1, 2010, Pages 4-10

  Paradkar, Anant ^a   Pawar, Atmaram ^b   Jadhav, Namdeo ^c  

^a UNIVERSITY OF BRADFORD   (United Kingdom)

^b BHARATI VIDYAPEETH DEEMED UNIVERSITY   (India)

^c BHARATI VIDYAPEETH COLLEGE OF PHARMACY   (India)

Author keywords

Crystallo co agglomeration; spansules; spherical agglomerates; tablet intermediates

Indexed keywords

BROMHEXINE; DILUENT; IBUPROFEN; NAPROXEN; PARACETAMOL; POLYMER; SOLVENT; STARCH; TALC;

CRYSTALLIZATION; CRYSTALLOCOAGGLOMERATION; DISPERSION; DRUG DELIVERY SYSTEM; DRUG RELEASE; PHARMACEUTICAL ENGINEERING; PROCESS DESIGN; REVIEW; SOLUBILIZATION; SUPERNATANT; TABLET COMPRESSION;

EID: 77953834396     PISSN: 09738398     EISSN: 1998409X     Source Type: Journal    
DOI: 10.4103/0973-8398.63975     Document Type: Review

References (51)

1. Kawashima Y. Spherical crystallization as a novel particle design technique for oral drug delivery system. Chin Pharm J 1989;41:163-172
2. Lachman L, Liberman HA, Kanig JL. Theory and Practice of Industrial Pharmacy. 2nd ed. Philadelphia, USA: Lea & Febiger; 1976. p. 317-324
3. Woodruff CW, Nuessle NO. Effect of processing variables on particles obtained by extrusion-spheronisation processing. J Pharm Sci 1972;61:787-790
4. Lachman L, Liberman HA, Kanig JL. Theory and Practice of Industrial Pharmacy. 2nd ed. Philadelphia, USA: Lea & Febiger; 1976. p. 338-339
5. Piera D, Mara S, Etienne JG. The spray drying of acetazolamide as a method to modify crystal properties and to improve compression behaviour. Int J Pharm 2001;213:209-221
6. Asker AF, Beeker CH. Some spray-dried formulations of sulfaethylthiadiazole for prolonged-release medication. J Pharm Sci 1966;55:90-94
7. Aerger JS, Price R. Processing of spherical crystalline particles via a novel solution atomisation and xtallisation by sonication (SAXS) technique. Pharm Res 2004;21:372-381
8. Paradkar AR, Maheshwari M, Chauhan B. Preparation and evaluation of ibuprofen beads by melt solidification technique. Int J Pharm 2003;255:33-42. (Pubitemid 36369588)
9. Paradkar AR, Maheshwari M, Jahagirdar HA. Melt sonocrystallisation of ibuprofen: Effect on crystal properties. Eur J Pharm Sci 2005;25:41-48
10. Jayasankar A, Somwangthanaroj A. Cocrystal formation during cogrinding and storage is mediated by amorphous phase. Pharm Res 2006;23:2381-2392
11. Kawashima Y, Okumura M, Takenaka H. Spherical crystallization: Direct spherical agglomeration of salicylic acid during crystallization. Science 1982;216:1127-1128
12. Kadam SS, Mahadik KR, Paradkar AR. A process for making agglomerates for use as or in a drug delivery system. Indian Patent 183036;1997.
13. Kadam SS, Mahadik KR, Paradkar AR. A process for making agglomerates for use as or in a drug delivery system. Indian Patent 183481;1997.
14. Tapia C, Buckton G, Newton J. Factors influencing the mechanism of release from sustained release matrix pellets produced by extrusion- spheronization. Int J Pharm 1993;92:211-218
15. Neau SH, Chow MY, Durrani MJ. Fabrication and characterization of extruded and spheronized beads containing carbopol 974P NF resin. Int J Pharm 1996;131:47-55.
16. Goskonda SR, Hileman GA, Upadrashta SM. Controlled release pellets by extrusion-spheronization. Int J Pharm 1994;111:89-97.
17. Jorgensen K, Christensen FN, Jacobsen L. Dissolution stability of multiparticulate controlled release tablets. Int J Pharm 1997;153:1-11.
18. Umprayn K, Chitropas P, Amarekajom S. Development of terbutaline sulfate sustained-release coated pellets. Drug Dev Ind Pharm 1999;25:477-491
19. Kojima M, Nakagami H. Development of controlled release matrix pellets by annealing with micronized water-insoluble or enteric polymers. J Control Release 2002;82:335-343
20. Bechgaard H, Hegermann NG. Controlled-release multiple-units and single-unit doses: a literature review. Drug Dev Ind Pharm 1978;4:53-67.
21. Tang SK, Chan LW, Heng WS. Coating of multiparticulates for sustained release. Am J Drug Deliv 2005;3:17-18
22. Freely LC, Khosla R, Davis SS. Investigating the gastric emptying of different sizes of non- disintegrating tablets in humans using gamma scintigraphy. J Pharm Pharmacol 1987;39:31-37
23. Bechgaard H. Critical factors influencing gastrointestinal absorption: What is the role of pellets? Acta Pharm Technol 1982;28:149-157
24. Devereux JE, Newton JM, Short MB. The influence of density on the gastrointestinal transit of pellets. J Pharm Pharmacol 1990;42:500-501
25. Clarke GM, Newton MJ, Short MD. Gastrointestinal transit of pellets of differing size and density. Int J Pharm 1993;100:81-92.
26. Tuleu C, Andrieux C, Boy P, Chaumeil JC. Gastrointestinal transit of pellets in rats: Effect of size and density. Int J Pharm 1999;180:123-131
27. Paradkar AR, Mahadik KR, Pawar AP. Spherical crystallization a novel particle design technique. Indian Drugs 1998;31:283-299
28. Jadhav NR. Studies on applications of crystallo-co-agglomeration technique in pharmaceutical formulations [doctoral thesis], Bharati Vidyapeeth University, Pune 2009.
29. Jadhav NR. Studies on agglomerates of bromhexine hydrochloride loaded talc prepared by crystallo-co-agglomeration [masters thesis], University of Pune 1998.
30. Pawar AP, Paradkar AR, Kadam SS, Mahadik KR. Agglomeration of ibuprofen with talc by novel crystallo-co-agglomeration technique. AAPS PharmSciTech 2004;5:1-6.
31. Pawar AP, Paradkar AR, Kadam SS, Mahadik KR. Crystallo-co-agglomeration: A novel process to obtain ibuprofen-paracetamol agglomerates. AAPS PharmSciTech 2004;5:1-8.
32. Gadekar SE. Studies on preparation of bromhexine hydrochloride loaded talc agglomerates by wet agglomeration technique [Masters thesis], University of Pune; 1997.
33. Pawar AP. Studies on spherical crystallisation of various pharmaceuticals [Doctoral thesis], University of Pune; 1999.
34. Kawashima Y, Aoki S, Takenaka H, Miyake Y. Preparation of spherically agglomerated crystals of aminophylline. J Pharm Sci 1984;73:1407-1410
35. Limzerwala RB. Optimization of the wet agglomeration of talc [Masters thesis], University of Pune; 1996.
36. Ganjian F, Cutie AJ, Jochsaberger T. In vitro adsorption studies of cimetidine. J Pharm Sci 1980;69:352-353
37. Maghsoodi M, Omid T, Martin GP, Nokhodchi A. Particle design of naproxen-disintegrant agglomerates for direct compression by a crystallo-co-agglomeration technique. Int J Pharm 2008;351:45-54.
38. Rao RP. Studies on talc agglomeration process [Masters thesis], University of Pune; 1997.
39. Jagdale SC. Studies on evaluation of crystallo-co-agglomerates of bromhexine hydrochloride loaded talc [Masters thesis], University of Pune; 2000.
40. Kawashima Y, Handa T, Hirofumi T, Okumura M. Effects of polyethylene glycol on size of agglomerated crystals of phenytoin prepared by the spherical crystallization technique. Chem Pharm Bull (Tokyo) 1986;34:3403-3407
41. Kawashima Y, Handa T, Tekeuchi H, Okumara M, Katou H, Nagata O. Crystal modification of phenytoin with polyethylene glycol for improving mechanical strength, dissolution rate and bioavailability by spherical crystallization technique. Chem Pharm Bull (Tokyo) 1986;34:3376-3383
42. Jadhav NR, Pawar AP, Paradkar AR. Design and evaluation of deformable talc agglomerates prepared by crystallo-co-agglomeration technique for generating heterogeneous matrix. AAPS PharmSciTech 2007;8:1-7.
43. Pawar AP, Paradkar AR, Kadam SS, Mahadik KR. Effect of polymers on crystallo-co-agglomeration of ibuprofen-paracetamol: Factorial design. Indian J Pharm Sci 2007;69:654-658
44. Sanghavi NM, Sivanand R, Kotwaney HN. Dissolution pattern of miniscular sulfisoxazole. Ind J Pharm Sci 1979;41:116-117
45. Alsaidan SM, Abdulhakeem AA, Eshra AG. Improved dissolution rate of indomethacin by adsorbents. Drug Dev Ind Pharm 1998;24:389-394
46. Aulton ME, Dyer AM, Khan KA. The strength and compaction of millispheres: The design of a controlled-release drug delivery system for ibuprofen in the form of a tablet comprising compacted polymer-coated millispheres. Drug Dev Ind Pharm 1994;20:3069-3104
47. Lin K, Peck GE. Development of agglomerated talc, I: Evaluation of fluidized bed granulation parameters on the physical properties of agglomerated talc. Drug Dev Ind Pharm 1995;21:159-173
48. Lin K, Peck GE. Development of agglomerated talc, II: Optimization of the processing parameters for the preparation of granulated talc. Drug Dev Ind Pharm 1995;21:447-460
49. Ho T, Hersey JA. Granulation using the agglomerative phase of comminution. Powder Technol 1979;23:191-195
50. Patki SR. Extended release beads of felodipine prepared by crystallo-co-agglomeration technique [Masters thesis], Kolhapur: Shivaji University; 2009.
51. Shouche PV. Use of talc beads as coating substrates [Masters thesis], Kolhapur: Shivaji University; 2009.