메뉴 건너뛰기




Volumn 5, Issue 3, 2004, Pages

Crystallo-co-agglomeration: A novel technique to obtain ibuprofen paracetamol agglomerates

Author keywords

Crystallo co agglomeration; Drug combination; Ibuprofen; Paracetamol; Tableting properties

Indexed keywords

DICHLOROMETHANE; ETHYL CELLULOSE; GLUCOSE; IBUPROFEN; MACROGOL 6000; PARACETAMOL; POVIDONE; WATER;

EID: 23144461820     PISSN: 15309932     EISSN: 15309932     Source Type: Journal    
DOI: 10.1208/pt050344     Document Type: Article
Times cited : (68)

References (30)
  • 1
    • 0031808764 scopus 로고    scopus 로고
    • Physicochemical characterization of the orthorhombic polymorph of paracetamol crystallized from solution
    • Nicholas G, Frampton CS. Physicochemical characterization of the orthorhombic polymorph of paracetamol crystallized from solution. J Pharm Sci. 1998;87:684-693.
    • (1998) J. Pharm. Sci. , vol.87 , pp. 684-693
    • Nicholas, G.1    Frampton, C.S.2
  • 3
    • 0028908594 scopus 로고
    • Compaction behavior of paracetamol powders of different crystal shapes
    • Wang H, Zhang R. Compaction behavior of paracetamol powders of different crystal shapes. Drug Dev Ind Pharm. 1995;21:863-868.
    • (1995) Drug Dev. Ind. Pharm. , vol.21 , pp. 863-868
    • Wang, H.1    Zhang, R.2
  • 4
    • 0021311811 scopus 로고
    • The effect of temperature on the spherical crystallization of salicylic acid
    • Kawashima Y, Okumara M, Takenaka H. The effect of temperature on the spherical crystallization of salicylic acid. Powder Technol. 1984;39:41-47.
    • (1984) Powder Technol. , vol.39 , pp. 41-47
    • Kawashima, Y.1    Okumara, M.2    Takenaka, H.3
  • 6
    • 0021149943 scopus 로고
    • Preparation of spherically agglomerated crystals of aminophylline
    • Kawashima Y, Aoki S, Takenama H, Miyake Y. Preparation of spherically agglomerated crystals of aminophylline. J Pharm Sci. 1984;73:1407-1409.
    • (1984) J. Pharm. Sci. , vol.73 , pp. 1407-1409
    • Kawashima, Y.1    Aoki, S.2    Takenama, H.3    Miyake, Y.4
  • 7
    • 0031844920 scopus 로고    scopus 로고
    • Evaluation of tableting properties of agglomerates obtained by spherical crystallisation of trimethoprim
    • Pawar PH, Pawar AP, Mahadik KR, Paradkar AR. Evaluation of tableting properties of agglomerates obtained by spherical crystallisation of trimethoprim. Indian J Pharm Sci. 1998; 60:24-28.
    • (1998) Indian J. Pharm. Sci. , vol.60 , pp. 24-28
    • Pawar, P.H.1    Pawar, A.P.2    Mahadik, K.R.3    Paradkar, A.R.4
  • 8
    • 0028371395 scopus 로고
    • Improvement in flowability and compressibility of pharmaceutical crystals for direct tableting by spherical crystallization with a two solvent system
    • Kawashima Y, Cui F, Takeuchi H, Niwa T, Hino T, Kiuchi K. Improvement in flowability and compressibility of pharmaceutical crystals for direct tableting by spherical crystallization with a two solvent system. Powder Technol. 1994;78:151-156.
    • (1994) Powder Technol. , vol.78 , pp. 151-156
    • Kawashima, Y.1    Cui, F.2    Takeuchi, H.3    Niwa, T.4    Hino, T.5    Kiuchi, K.6
  • 9
    • 0027443919 scopus 로고
    • Preparation of microcapsules masking the bitter taste of enoxacin by using one continuous process of agglomeration and microencapsulation
    • Ueda M, Nakamura Y, Makita H, Kawashima Y. Preparation of microcapsules masking the bitter taste of enoxacin by using one continuous process of agglomeration and microencapsulation. J Microencapsul. 1993;10:461-473.
    • (1993) J. Microencapsul. , vol.10 , pp. 461-473
    • Ueda, M.1    Nakamura, Y.2    Makita, H.3    Kawashima, Y.4
  • 10
    • 0019977953 scopus 로고
    • Direct agglomeration of sodium theophylline crystals produced by salting out in liquid
    • Kawashima Y, Lin SY, Naito M, Takenama H. Direct agglomeration of sodium theophylline crystals produced by salting out in liquid. Chem Pharm Bull (Tokyo). 1982;30:1837-1843.
    • (1982) Chem. Pharm. Bull. (Tokyo) , vol.30 , pp. 1837-1843
    • Kawashima, Y.1    Lin, S.Y.2    Naito, M.3    Takenama, H.4
  • 11
    • 0022354197 scopus 로고
    • Prolonged release microcapsules of indomethacin through spherical crystallization technique
    • Kawashima Y, Lin Y, Ogawa M, Handa T, Takenaka H. Prolonged release microcapsules of indomethacin through spherical crystallization technique. J Pharm Sci. 1985;74:1152-1156.
    • (1985) J. Pharm. Sci. , vol.74 , pp. 1152-1156
    • Kawashima, Y.1    Lin, Y.2    Ogawa, M.3    Handa, T.4    Takenaka, H.5
  • 12
    • 33544459039 scopus 로고    scopus 로고
    • A process for making agglomerates for use as or in a drug delivery system
    • inventors. February
    • Kadam SS, Mahadik KR, Paradkar AR, inventors. A process for making agglomerates for use as or in a drug delivery system. Indian patent 183036. February 14, 1997.
    • Indian Patent 183036 , vol.14 , pp. 1997
    • Kadam, S.S.1    Mahadik, K.R.2    Paradkar, A.R.3
  • 13
    • 33544459039 scopus 로고    scopus 로고
    • A process for making agglomerates for use as or in a drug delivery system
    • inventors. February
    • Kadam SS, Mahadik KR, Paradkar AR, inventors. A process for making agglomerates for use as or in a drug delivery system. Indian patent 183481. February 14, 1997.
    • Indian Patent 183481 , vol.14 , pp. 1997
    • Kadam, S.S.1    Mahadik, K.R.2    Paradkar, A.R.3
  • 14
    • 0027622964 scopus 로고
    • Micromeritic characteristics and agglomeration mechanisms in the spherical crystallization of bucillamine by the spherical agglomeration and the emulsion solvent diffusion methods
    • Morishima K, Kawashima Y, Takeuchi H, Niwa T, Hino T. Micromeritic characteristics and agglomeration mechanisms in the spherical crystallization of bucillamine by the spherical agglomeration and the emulsion solvent diffusion methods. Powder Technol. 1993;76:57-64.
    • (1993) Powder Technol. , vol.76 , pp. 57-64
    • Morishima, K.1    Kawashima, Y.2    Takeuchi, H.3    Niwa, T.4    Hino, T.5
  • 17
    • 0020611968 scopus 로고
    • Comparison of granule strength and tablet strength
    • Jarosz PJ, Parrot EJ. Comparison of granule strength and tablet strength. J Pharm Sci. 1983;72:530-535.
    • (1983) J. Pharm. Sci. , vol.72 , pp. 530-535
    • Jarosz, P.J.1    Parrot, E.J.2
  • 18
    • 0000292691 scopus 로고
    • Density - Pressure relationships in powder compaction
    • Heckel RW. Density - pressure relationships in powder compaction. Trans Mettall Soc AIME. 1961;221:671-675.
    • (1961) Trans. Mettall. Soc. AIME , vol.221 , pp. 671-675
    • Heckel, R.W.1
  • 19
    • 0000693333 scopus 로고
    • An analysis of powder compaction phenomena
    • Heckel RW. An analysis of powder compaction phenomena. Trans Mettall Soc AIME. 1961;221:1001-1008.
    • (1961) Trans. Mettall. Soc. AIME , vol.221 , pp. 1001-1008
    • Heckel, R.W.1
  • 20
    • 0018152610 scopus 로고
    • A universal friability test for tablet granules
    • Rubinstein MH, Musikabhumma P. A universal friability test for tablet granules. Pharm Acta Helv. 1978;53:125-129.
    • (1978) Pharm. Acta Helv. , vol.53 , pp. 125-129
    • Rubinstein, M.H.1    Musikabhumma, P.2
  • 21
    • 0025159227 scopus 로고
    • Thermodynamics of paracetamol solubility in sugar-water cosolvent systems
    • Etman MA, Naggar VF. Thermodynamics of paracetamol solubility in sugar-water cosolvent systems. Int J Pharm. 1990;58:177-184.
    • (1990) Int. J. Pharm. , vol.58 , pp. 177-184
    • Etman, M.A.1    Naggar, V.F.2
  • 22
    • 0024445139 scopus 로고
    • Preparation and characterization of microspheres containing the anti-inflammatory agents, indomethacin, ibuprofen and ketoprofen
    • Bodmeier R, Chen H. Preparation and characterization of microspheres containing the anti-inflammatory agents, indomethacin, ibuprofen and ketoprofen. J Control Release. 1989;10:167-175.
    • (1989) J. Control Release , vol.10 , pp. 167-175
    • Bodmeier, R.1    Chen, H.2
  • 23
    • 33544473441 scopus 로고    scopus 로고
    • Preparation and evaluation of ibuprofen beads by melt solidification technique
    • Paradkar AR, Maheshwari M, Ketkar AR, Chauhan B. Preparation and evaluation of ibuprofen beads by melt solidification technique. Int J Pharm. 2003;7427:1-10.
    • (2003) Int. J. Pharm. , vol.7427 , pp. 1-10
    • Paradkar, A.R.1    Maheshwari, M.2    Ketkar, A.R.3    Chauhan, B.4
  • 24
    • 0023018035 scopus 로고
    • Effect of polyethylene glycol on size of agglomerated crystals of phenytoin prepared by the spherical crystallization technique
    • Kawashima Y, Handa T, Takeuchi H, Okumura M. Effect of polyethylene glycol on size of agglomerated crystals of phenytoin prepared by the spherical crystallization technique. Chem Pharm Bull (Tokyo). 1986;34:3403-3407.
    • (1986) Chem. Pharm. Bull. (Tokyo) , vol.34 , pp. 3403-3407
    • Kawashima, Y.1    Handa, T.2    Takeuchi, H.3    Okumura, M.4
  • 25
    • 0022993268 scopus 로고
    • Crystal modification of phenytoin with polyethylene glycol for improving mechanical strength, dissolution rate and bioavailability by a spherical crystallization technique
    • Kawashima Y, Handa T, Takeuchi H, Okumura M, Katou H, Nagata O. Crystal modification of phenytoin with polyethylene glycol for improving mechanical strength, dissolution rate and bioavailability by a spherical crystallization technique. Chem Pharm Bull (Tokyo). 1986;34:3376-3383.
    • (1986) Chem. Pharm. Bull. (Tokyo) , vol.34 , pp. 3376-3383
    • Kawashima, Y.1    Handa, T.2    Takeuchi, H.3    Okumura, M.4    Katou, H.5    Nagata, O.6
  • 26
    • 0029969203 scopus 로고    scopus 로고
    • A study of the mechanism of wet spherical agglomeration of pharmaceutical powders
    • Chow AHL, Leung MWM. A study of the mechanism of wet spherical agglomeration of pharmaceutical powders. Drug Dev Ind Pharm. 1996;22:357-362.
    • (1996) Drug Dev. Ind. Pharm. , vol.22 , pp. 357-362
    • Chow, A.H.L.1    Leung, M.W.M.2
  • 27
    • 0030881924 scopus 로고    scopus 로고
    • An investigation into the melting behavior of binary mixer and solid dispersion of paracetamol and PEG 4000
    • Lloyd GR, Craig DQ, Smith A. An investigation into the melting behavior of binary mixer and solid dispersion of paracetamol and PEG 4000. J Pharm Sci. 1997;86:991-196.
    • (1997) J. Pharm. Sci. , vol.86 , pp. 196-991
    • Lloyd, G.R.1    Craig, D.Q.2    Smith, A.3
  • 28
    • 23144448142 scopus 로고    scopus 로고
    • Influence of ibuprofen as a solid-state plasticizer in Eudragit RS 30 D on the physicochemical properties of coated beads
    • Wu C, McGinity JW. Influence of ibuprofen as a solid-state plasticizer in Eudragit RS 30 D on the physicochemical properties of coated beads. AAPS PharmSciTech. 2001;2:E24.
    • (2001) AAPS PharmSciTech. , vol.2
    • Wu, C.1    McGinity, J.W.2
  • 29
    • 0025836698 scopus 로고
    • Ibuprofen-loaded ethylcellulose microspheres: Analysis of the matrix structure by thermal analysis
    • Dubernet C, Rouland JC, Benoit JP. Ibuprofen-loaded ethylcellulose microspheres: analysis of the matrix structure by thermal analysis. J Pharm Sci. 1991;80:1029-1133.
    • (1991) J. Pharm. Sci. , vol.80 , pp. 1029-1133
    • Dubernet, C.1    Rouland, J.C.2    Benoit, J.P.3
  • 30
    • 0023908724 scopus 로고
    • The effects of interacting variables on the tensile strength, disintegration and dissolution of paracetamol tablets
    • Zubir S, Esezobo S, Pilpel N. The effects of interacting variables on the tensile strength, disintegration and dissolution of paracetamol tablets. J Pharm Pharmacol. 1988;40:278-281.
    • (1988) J. Pharm. Pharmacol. , vol.40 , pp. 278-281
    • Zubir, S.1    Esezobo, S.2    Pilpel, N.3


* 이 정보는 Elsevier사의 SCOPUS DB에서 KISTI가 분석하여 추출한 것입니다.