-
1
-
-
3142676436
-
-
Shah, N. P.; Tran, C.; Lee, F. Y.; Chen, P.; Norris, D.; Sawyers, C. L. Science 2004, 305, 399.
-
(2004)
Science
, vol.305
, pp. 399
-
-
Shah, N.P.1
Tran, C.2
Lee, F.Y.3
Chen, P.4
Norris, D.5
Sawyers, C.L.6
-
2
-
-
19944428353
-
-
Lombardo, L. J.; Lee, F. Y.; Chen, P.; Norris, D.; Barrish, J. C.; Behnia, K.; Castaneda, S.; Cornelius L. A. M.; Das, J.; Doweyko, A. M.; Fairchild, C.; Hunt, J. T.; Inigo, I.; Johnston, K.; Kamath, A.; Kan, D.; Klei, H.; Marathe, P.; Pang, S.; Peterson, R.L.; Pitt, S.; Schieven, G. L.; Schmidt, R. J.; Tokarski, J.; Wen, M.-L.; Wityak, J.; Borzilleri, R. J. Med. Chem. 2004, 47, 6658.
-
(2004)
J. Med. Chem.
, vol.47
, pp. 6658
-
-
Lombardo, L.J.1
Lee, F.Y.2
Chen, P.3
Norris, D.4
Barrish, J.C.5
Behnia, K.6
Castaneda, S.7
Cornelius, L.A.M.8
Das, J.9
Doweyko, A.M.10
Fairchild, C.11
Hunt, J.T.12
Inigo, I.13
Johnston, K.14
Kamath, A.15
Kan, D.16
Klei, H.17
Marathe, P.18
Pang, S.19
Peterson, R.20
Pitt, S.21
Schieven, G.L.22
Schmidt, R.J.23
Tokarski, J.24
Wen, M.-L.25
Wityak, J.26
Borzilleri, R.27
more..
-
3
-
-
33744486584
-
-
Copland, M.; Hamilton, A.; Elrick, L. J.; Baird, J. W.; Allan, E. K.; Jordanides, N.; Barow, M.; Mountford, J. C.; Holyoake, T. L. Blood 2006, 107, 4532.
-
(2006)
Blood
, vol.107
, pp. 4532
-
-
Copland, M.1
Hamilton, A.2
Elrick, L.J.3
Baird, J.W.4
Allan, E.K.5
Jordanides, N.6
Barow, M.7
Mountford, J.C.8
Holyoake, T.L.9
-
4
-
-
33745191477
-
-
McIntyre, J. A.; Castaner, J.; Bayes, M. Drugs of the Future 2006, 31, 291
-
(2006)
Drugs of the Future
, vol.31
, pp. 291
-
-
McIntyre, J.A.1
Castaner, J.2
Bayes, M.3
-
5
-
-
33745283618
-
-
Tokarski, J. S.; Newitt, J. A.; Chang, C. Y. J.; Cheng, J. D.; Wittekind, M.; Kiefer, S. E.; Kish, K.; Lee, F. Y. F.; Borzillerri, R.; Lombardo, L. J.; Xie, D.; Zhang, Y.; Klei, H. E. Cancer Res. 2006, 66, 5790.
-
(2006)
Cancer Res.
, vol.66
, pp. 5790
-
-
Tokarski, J.S.1
Newitt, J.A.2
Chang, C.Y.J.3
Cheng, J.D.4
Wittekind, M.5
Kiefer, S.E.6
Kish, K.7
Lee, F.Y.F.8
Borzillerri, R.9
Lombardo, L.J.10
Xie, D.11
Zhang, Y.12
Klei, H.E.13
-
6
-
-
21144451094
-
-
O'Hare, T.; Walters, D. K.; Stoffregen, E. P.; Jia, T.; Manley, P. W.; Mestan, J.; Cowan-Jacob, S. W.; Lee, F. Y.; Heinrich, M. C.; Deininger, M. W.; Druker, B. J. Cancer Res. 2005; 65, 4500.
-
(2005)
Cancer Res.
, vol.65
, pp. 4500
-
-
O'Hare, T.1
Walters, D.K.2
Stoffregen, E.P.3
Jia, T.4
Manley, P.W.5
Mestan, J.6
Cowan-Jacob, S.W.7
Lee, F.Y.8
Heinrich, M.C.9
Deininger, M.W.10
Druker, B.J.11
-
7
-
-
33750989362
-
-
Das, J.; Chen, P.; Norris, D.; Padmanabha, R.; Lin, J.; Moquin, R. V.; Shen, Z.; Cook, L. S.; Doweyko, A. M.; Pitt, S.; Pang, S.; Shen, D. R.; Fang, Q.; de Fex, H. F.; McIntyre, K. W.; Shuster, D. J.; Gillooly, K. M.; Behnia, K.; Schieven, G. L.; Wityak, J.; Barrish, J. C. J. Med. Chem. 2006, 49, 6819.
-
(2006)
J. Med. Chem.
, vol.49
, pp. 6819
-
-
Das, J.1
Chen, P.2
Norris, D.3
Padmanabha, R.4
Lin, J.5
Moquin, R.V.6
Shen, Z.7
Cook, L.S.8
Doweyko, A.M.9
Pitt, S.10
Pang, S.11
Shen, D.R.12
Fang, Q.13
De Fex, H.F.14
McIntyre, K.W.15
Shuster, D.J.16
Gillooly, K.M.17
Behnia, K.18
Schieven, G.L.19
Wityak, J.20
Barrish, J.C.21
more..
-
8
-
-
0035843401
-
-
Zhao, R.; Gove, S., Sundeen, J. E.; Chen, B.-C. Tetrahedron Lett. 2001, 42, 2101
-
(2001)
Tetrahedron. Lett.
, vol.42
, pp. 2101
-
-
Zhao, R.1
Gove, S.2
Sundeen, J.E.3
Chen, B.-C.4
-
9
-
-
0001065532
-
-
For previous reports on N-bromination of amides with NBS, see
-
For previous reports on N-bromination of amides with NBS, see: Armstrong, R. W.; Tellew, J. E.; Moran, E. J. J. Org. Chem. 1992, 57, 2208.
-
(1992)
J. Org. Chem.
, vol.57
, pp. 2208
-
-
Armstrong, R.W.1
Tellew, J.E.2
Moran, E.J.3
-
11
-
-
77953367466
-
-
Shin, C.-G.; Nanjo, K.; Nishino, T.; Sato, Y.; Yoshimura, J. Bull. Chem. Soc. Jpn. 1975, 48, 2492.
-
(1975)
Bull. Chem. Soc. Jpn.
, vol.48
, pp. 2492
-
-
Shin, C.-G.1
Nanjo, K.2
Nishino, T.3
Sato, Y.4
Yoshimura, J.5
-
12
-
-
77953396115
-
-
Sato, Y.; Yonezawa, Y.; Shin, C. Heterocycles 1982, 19, 1463.
-
(1982)
Heterocycles
, vol.19
, pp. 1463
-
-
Sato, Y.1
Yonezawa, Y.2
Shin, C.3
-
13
-
-
3042634493
-
-
For previous reports on phenyl ring brominations of anilinides with NBS, see
-
For previous reports on phenyl ring brominations of anilinides with NBS, see: Occhiato, E. G.; Ferrali, A.; Menchi, G.; Guarna, A.; Danza, G.; Comerci, A.; Mancina, R.; Serio, M.; Garotta, G.; Cavalli, A.; Vivo, M. D.; Recanatini, M. J. Med. Chem. 2004, 47, 3546.
-
(2004)
J. Med. Chem.
, vol.47
, pp. 3546
-
-
Occhiato, E.G.1
Ferrali, A.2
Menchi, G.3
Guarna, A.4
Danza, G.5
Comerci, A.6
Mancina, R.7
Serio, M.8
Garotta, G.9
Cavalli, A.10
Vivo, M.D.11
Recanatini, M.12
-
15
-
-
0034079340
-
-
Andersh, B.; Murphy, D. L.; Olson, R. J. Synth. Commun. 2000, 12, 2091.
-
(2000)
Synth. Commun.
, vol.12
, pp. 2091
-
-
Andersh, B.1
Murphy, D.L.2
Olson, R.J.3
-
16
-
-
33746338291
-
-
Elmorsy, S. S.; Badawy, D. S.; Khatab, T. K. Phosphorus, Sulfur Silicon Relat. Elem. 2006, 181, 2005.
-
(2006)
Phosphorus, Sulfur Silicon Relat. Elem
, vol.181
, pp. 2005
-
-
Elmorsy, S.S.1
Badawy, D.S.2
Khatab, T.K.3
-
18
-
-
0031025752
-
-
Hoshino, Y.; Miyazawa, S.; Nakata, H.; Etoh, H.; Furitsu, M.; Abe, S. J. Labelled Compd. Radiopharm. 1997, 39, 109.
-
(1997)
J. Labelled Compd. Radiopharm
, vol.39
, pp. 109
-
-
Hoshino, Y.1
Miyazawa, S.2
Nakata, H.3
Etoh, H.4
Furitsu, M.5
Abe, S.6
-
19
-
-
0023022233
-
-
For previous reports on preparation of β-alkoxy acrylamides from β-alkoxy acryloyl chlorides, see
-
For previous reports on preparation of β-alkoxy acrylamides from β-alkoxy acryloyl chlorides, see: Leclerc, G.; Marciniak, G.; Decker, N.; Schwartz, J. J. Med. Chem. 1986, 29, 2427.
-
(1986)
J. Med. Chem.
, vol.29
, pp. 2427
-
-
Leclerc, G.1
Marciniak, G.2
Decker, N.3
Schwartz, J.4
-
20
-
-
0024344270
-
-
Bell, A. S.; Campbell, S. F.; Morris, D. S.; Roberts, D. A.; Stefaniak, M. H. J. Med. Chem. 1989, 32, 1552.
-
(1989)
J. Med. Chem.
, vol.32
, pp. 1552
-
-
Bell, A.S.1
Campbell, S.F.2
Morris, D.S.3
Roberts, D.A.4
Stefaniak, M.H.5
-
21
-
-
0019179780
-
-
Yoshizaki, S.; Osaki, M.; Nakagawa, K.; Tamura, Y. Chem. Pharm. Bull. 1980, 28, 3441.
-
(1980)
Chem. Pharm. Bull.
, vol.28
, pp. 3441
-
-
Yoshizaki, S.1
Osaki, M.2
Nakagawa, K.3
Tamura, Y.4
-
22
-
-
0022571466
-
-
Tominaga, M.; Yo, E.; Ogawa, H.; Yamashita, S.; Yabuuchi, Y.; Nakagawa, K. Chem. Pharm. Bull. 1986, 34, 682.
-
(1986)
Chem. Pharm. Bull.
, vol.34
, pp. 682
-
-
Tominaga, M.1
Yo, E.2
Ogawa, H.3
Yamashita, S.4
Yabuuchi, Y.5
Nakagawa, K.6
-
23
-
-
0020623851
-
-
Baron, M.; Giorgi-Renault, S.; Renault, J.; Paoletti, C.; Cros, S. Eur. J. Med. Chem. Chim. Ther. 1983, 18, 134.
-
(1983)
Eur. J. Med. Chem. Chim. Ther.
, vol.18
, pp. 134
-
-
Baron, M.1
Giorgi-Renault, S.2
Renault, J.3
Paoletti, C.4
Cros, S.5
-
24
-
-
0033738449
-
-
Baston, E.; Palusczak, A.; Hartmann, R. W. Eur. J. Med. Chem. Chim. Ther. 2002, 35, 931.
-
(2002)
Eur. J. Med. Chem. Chim. Ther.
, vol.35
, pp. 931
-
-
Baston, E.1
Palusczak, A.2
Hartmann, R.W.3
-
25
-
-
0035904860
-
-
Ashwell, M. A.; Solvibile, W. R.; Han, S.; Largis, E.; Mulvey, R.; Tillet, J. Bioorg. Med. Chem. Lett. 2001, 24, 3123.
-
(2001)
Bioorg. Med. Chem. Lett.
, vol.24
, pp. 3123
-
-
Ashwell, M.A.1
Solvibile, W.R.2
Han, S.3
Largis, E.4
Mulvey, R.5
Tillet, J.6
-
26
-
-
8844271817
-
-
Chen, P.; Norris, D.; Das, J.; Spergel, S. H.; Wityak, J.; Leith, L.; Zhao, R.; Chen, B.-C.; Pitt, S.; Pang, S.; Shen, D. R.; Zhang, R.; De Fex, H. F.; Doweyko, A. M.; McIntyre, K. W.; Shuster, D. J.; Behnia, K.; Schieven, G. L.; Barrish, J. C. Bioorg. Med. Chem. Lett. 2004, 14, 6061.
-
(2004)
Bioorg. Med. Chem. Lett.
, vol.14
, pp. 6061
-
-
Chen, P.1
Norris, D.2
Das, J.3
Spergel, S.H.4
Wityak, J.5
Leith, L.6
Zhao, R.7
Chen, B.-C.8
Pitt, S.9
Pang, S.10
Shen, D.R.11
Zhang, R.12
De Fex, H.F.13
Doweyko, A.M.14
McIntyre, K.W.15
Shuster, D.J.16
Behnia, K.17
Schieven, G.L.18
Barrish, J.C.19
-
27
-
-
0142031003
-
-
McCluskey, A.; Keller, P. A.; Morgan, J.; Garner, J. Org. Biomol. Chem. 2003, 1, 3353.
-
(2003)
Org. Biomol. Chem.
, vol.1
, pp. 3353
-
-
McCluskey, A.1
Keller, P.A.2
Morgan, J.3
Garner, J.4
-
28
-
-
0035847696
-
-
Tian, X.; Hsin, L.-W.; Webster, E. L.; Contoreggi, C.; Chrousos, G. P.; Gold, P. W.; Habib, K.; Ayala, A.; Eckelman, W. C.; Jacobson, A. E.; Rice, K. C. Bioorg. Med. Chem. Lett. 2001, 11, 331.
-
(2001)
Bioorg. Med. Chem. Lett.
, vol.11
, pp. 331
-
-
Tian, X.1
Hsin, L.-W.2
Webster, E.L.3
Contoreggi, C.4
Chrousos, G.P.5
Gold, P.W.6
Habib, K.7
Ayala, A.8
Eckelman, W.C.9
Jacobson, A.E.10
Rice, K.C.11
-
30
-
-
32444446491
-
-
Weber, C.; Demeter, A.; Greiner, I. Tetrahedron 2006, 62, 2304.
-
(2006)
Tetrahedron.
, vol.62
, pp. 2304
-
-
Weber, C.1
Demeter, A.2
Greiner, I.3
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