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Volumn 35, Issue 10, 2000, Pages 931-940

6-Substituted 1H-quinolin-2-ones and 2-methoxy-quinolines: Synthesis and evaluation as inhibitors of steroid 5α reductases types 1 and 2

(3) Baston, Eckhard a Palusczak, Anja a Hartmann, Rolf W a

a SAARLAND UNIVERSITY (Germany)

Author keywords

1H quinolin 2 ones; 5 reductase isozymes 1 and 2; Methoxyquinolines; Nonsteroidal inhibitors

Indexed keywords

6 [4 (N,N DIISOPROPYLCARBAMOYL)PHENYL] 1H QUINOLIN 2 ONE; FINASTERIDE; PYRIDONE DERIVATIVE; QUINOLINE DERIVATIVE; STEROID 5ALPHA REDUCTASE INHIBITOR; UNCLASSIFIED DRUG;

ARTICLE; CONTROLLED STUDY; DRUG ACTIVITY; DRUG SELECTIVITY; DRUG STRUCTURE; DRUG SYNTHESIS; ENZYME DEFICIENCY; HUMAN; HUMAN CELL; REACTION ANALYSIS;

EID: 0033738449 PISSN: 02235234 EISSN: None Source Type: Journal
DOI: 10.1016/S0223-5234(00)01167-3 Document Type: Article

Times cited : (54)

References (27)

1
- 0030338705
- (1996) Scand. J. Urol. Nephrol. , vol.30 , Issue.SUPPL. 180 , pp. 1-55
- Hansen, B.J.¹

2
- 0030913442
- (1997) J. Med. Chem. , vol.40 , pp. 1293-1315
- Kenny, B.¹ Ballard, S.² Blagg, J.³ Fox, D.⁴

3
- 0028072025
- (1994) J. Clin. Endocrinol. Metab. , vol.79 , pp. 991-996
- Rhodes, L.¹ Harper, J.² Uno, H.³ Gaito, G.⁴ Audette-Arruda, J.⁵ Kurata, S.⁶ Berman, C.⁷ Primka, R.⁸ Pikounis, B.⁹

4
- 0027531675
- (1993) J. Med. Chem. , vol.36 , pp. 421-423
- Jones, C.D.¹ Audia, J.E.² Lawhorn, D.E.³ McQuaid, L.A.⁴ Neubauer, B.L.⁵ Pike, A.J.⁶ Pennington, P.A.⁷ Stamm, N.B.⁸ Toomey, R.E.⁹ Hirsch, K.S.¹⁰

5
- 0343144447
- (1998) Nat. Prod. Reports , pp. 495-512
- Jarman, M.¹ Smith, H.J.² Nicholls, P.J.³ Simons, C.⁴

6
- 0029055505
- (1995) Steroids , vol.60 , pp. 430-441
- Li, X.¹ Chen, C.² Singh, S.M.³ Labrie, F.⁴

7
- 0016359646
- (1974) Science , vol.186 , pp. 1213-1215
- Imperato-McGinley, J.¹ Guerrero, L.² Gautier, T.³ Peterson, R.E.⁴

8
- 0028147948
- (1994) Clin. Endocrinol. , vol.41 , pp. 139-147
- Schroder, F.H.¹

9
- 0025303307
- (1990) Proc. Natl. Acad. Sci. USA , vol.87 , pp. 3640-3644
- Andersson, S.¹ Russell, D.W.²

10
- 0022971248
- (1986) J. Med. Chem. , vol.29 , pp. 2298-2315
- Rasmusson, G.H.¹ Reynolds, G.F.² Steinberg, N.G.³ Walton, E.⁴ Patel, G.F.⁵ Liang, T.⁶ Cascieri, M.A.⁷ Cheung, A.H.⁸ Brooks, J.R.⁹ Nerman, C.¹⁰

11
- 0025240643
- (1990) J. Med. Chem. , vol.33 , pp. 943-950
- Holt, D.A.¹ Levy, M.A.² Oh, H.J.³ Erb, J.M.⁴ Heaslip, J.I.⁵ Brandt, M.⁶ Lan-Hargest, H.Y.⁷ Metcalf, B.W.⁸

12
- 0028035187
- (1994) Eur. J. Med. Chem. , vol.29 , pp. 807-817
- Hartmann, R.W.¹ Reichert, M.² Gohring, S.³

13
- 0027430833
- (1993) Synthesis , pp. 1079-1080
- Tietze, L.F.¹ Schneider, C.² Pretor, M.³

14
- 4243489506
- (1993) Chem. Rev. , vol.93 , pp. 2117-2188
- Knochel, P.¹ Singer, R.D.²

15
- 0042270897
- (1996) Synlett , pp. 573-575
- Rottlander, M.¹ Palmer, N.² Knochel, P.³

16
- 0007162425
- (1983) Aust. J. Chem. , vol.26 , pp. 50-54
- Fong, C.W.¹ Grant, H.G.²

17
- 0002714801
- (1996) Curr. Pharm. Des. , vol.2 , pp. 59-84
- Frye, S.V.¹

18
- 0001631092
- (1991) J. Org. Chem. , vol.56 , pp. 5311-5318
- Lewis, F.D.¹ Reddy, G.D.² Ellbert, J.E.³ Tillberg, B.E.⁴ Meltzer, J.A.⁵ Kojima, M.⁶

19
- 0003760238
- Wiley, New York
- (1993) Enzyme Kinetics: Behaviour and Analysis of Rapid Equilibrium and Steady-State Enzyme Systems
- Segel, I.H.¹

20
- 0003492942
- Wiley, New York
- (1962) Theory and Application of Ultraviolet Spectroscopy
- Jaffe, H.H.¹ Richin, M.²

21
- 0003550135
- Thieme, Stuttgart, New York
- (1991) Reaktionen und Synthesen im Organisch-Chemischen Praktikum und Forschungslaboratorium
- Tietze, L.F.¹ Eicher, T.²

22
- 37049079948
- (1993) J. Chem. Soc., Perkin Trans. 1 , vol.2 , pp. 181-184
- Osborne, A.G.¹ Miller, L.A.D.²

23
- 0023764494
- (1988) J. Med. Chem. , vol.31 , pp. 2048-2056
- Alabaster, C.T.¹ Bell, A.S.² Campbell, S.F.³ Ellis, P.⁴ Henderson, C.G.⁵ Roberts, D.A.⁶ Ruddock, K.S.⁷ Samuels, G.M.R.⁸ Stefaniak, M.H.⁹

24
- 0015236546
- (1971) Biochem. Biophys. Acta , vol.242 , pp. 519-522
- Lee, H.J.¹ Wilson, I.B.²

25
- 0028301655
- (1994) J. Steroid Biochem. Mol. Biol. , vol.48 , pp. 347-352
- Delos, S.¹ Jehle, C.² Martin, P.M.³ Raynaud, J.P.⁴

26
- 3042981033
- (1996) J. Steroid Biochem. Mol. Biol. , vol.58 , pp. 195-205
- Kaefer, M.¹ Audia, J.E.² Bruchoversusky, N.³ Goode, R.L.⁴ Hsiao, K.C.⁵ Leibovitch, I.Y.⁶ Krushinski, J.H.⁷ Lee, C.⁸ Steidle, C.P.⁹ Sutkowski, D.M.¹⁰ Neubauer, B.L.¹¹

27
- 2642697958
- (1997) J. Med. Chem. , vol.40 , pp. 1112-1129
- Guarna, A.¹ Belle, C.² Machetti, F.³ Occhiato, E.G.⁴ Payne, A.H.⁵ Cassiani, C.⁶ Comerci, A.⁷ Danza, G.⁸ De Bellis, A.⁹ Dini, S.¹⁰ Marrucci, A.¹¹ Serio, M.¹²

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