Effect of water soluble polymers on dissolution profile of glipizide cyclodextrins complex

Indian Drugs

Volumn 45, Issue 1, 2008, Pages 31-36

  Patel, V P ^a   Patel, N M ^a   Chaudhari, B G ^a  

^a NONE

Author keywords

Complexation; Cyclodextrins; Glipizide; Stability; Water soluble polymers

Indexed keywords

BETA CYCLODEXTRIN; GLIPIZIDE; HYDROXYPROPYLMETHYLCELLULOSE; MACROGOL 4000; MACROGOL 6000; POLYMER; POVIDONE;

ARTICLE; COMPLEX FORMATION; CONTROLLED STUDY; DRUG DELIVERY SYSTEM; DRUG DOSAGE FORM COMPARISON; DRUG FORMULATION; DRUG SOLUBILITY; DRUG STABILITY; DRUG STORAGE;

EID: 77953392902     PISSN: 0019462X     EISSN: None     Source Type: Journal    
DOI: None     Document Type: Article

References (20)

1. Rx List web site, Description of glipizide, www.rxlist.com/cgi/generic/ glipxl.htm (Copyright 1998, Mosby Inc., Mosby's GenRx).
2. Frick, A., Moller, H. and Wirbitzki, E., Biopharmaceutical characterization of oral immediate release drug products. In vitro/in vivo comparison of Phenoxymethylpenicillin potassium, glipizide and levofloxacin. Eur. J. Pharm. Biopharm., 1998, 46, 305-311. (Pubitemid 29057678)
3. Massimo, M. B., Glipizide in type 2 diabetes mellitus: a review of the worldwide therapeutic experience. Clin. Ther., 2003, 25, 799-816. (Pubitemid 36459693)
4. Pitha J. and Fanco M., Hydroxypropyl-β-cyclodextrin: Preparation and Characterization; Effects on Solubility of Drugs, Int. J. Pharm., 1996, 29, 73-82.
5. Duchene, D., Cyclodextrins and Their Industrial Uses, Editions de Santé Paris, 1987.
6. Aungst, B.J., Novel formulation strategies for improving oral bioavailability of drugs with poor membrane permeation or presystemic metabolism. J. Pharm. Sci., 1993, 82, 979-987.
7. Martin. A., Bustamante, P. and Chun, A. H. C., Physical Pharmacy: Physical Chemical Principles in Pharmaceutical Sciences, 4th Edn. Lippincott Williams & Wilkins, 1993, pp. 260-261.
8. Higuchi, T. and Connors, K. A., Phase solubility technique. Adv. Anal.Chem. Instrum. 1965, 4, 117-212.
9. Uekama, K., Matsuo, N., Hirayama, F., Ichibagase, H., Arimori, K., Tsubaki, K. and Satake, K., Enhanced bioavailability of acetohexamide by betacyclodextrin complexation. Int. J. Pharm., 1980, 100, 903-909.
10. Ozkana, Y., Ataya, T., Dikmena, N., Isimera, A. and Aboul-Enein, H. Y., Improvement of water solubility and in vitro dissolution rate of gliclazide by complexation with β-cyclodextrin. Pharm. Acta Helv., 2000, 74, 365-370.
11. Sridevi, S., Chary, M. G., Krishna, D. R. and Diwan, P. V., Pharmacodynamics evaluation of transdermal drug delivery system of glibenclamide in rats. lnd. J. Pharmacol., 2000, 32, 309-312.
12. Veiga, F., Fernandes, C. and Teixeira, F., Oral bioavailability and hypoglycemic activity of tolbutamide/cyclodextrin inclusion complexes. Int. J. Pharm., 2000,202, 165-171.
13. Aggarwal, S., Singh, P. N. and Mishra, B., Studies on solubility and hypoglycemic activity of gliclazide beta-Cyclodextrin hydroxypropylmethylcellulose complexes. Pharmazie, 2002, 57, 191-193. (Pubitemid 34213912)
14. Del Valle, E. M. M., Cyclodextrins and their uses: a review. Process Biochem. 2004, 39, 1033-1046.
15. Loftsson, T., Magnusdottir, A., Masson, M. and Sigurjonsdottir, J. F., Self association and cyclodextrin solubilization of drugs. J. Pharm. Sci., 2002, 91, 2307-2316.
16. Corrigan, O. I. and Stanley, T., Mechanism of drug dissolution enhancement from β-cyclodextrin-drug systems. J. Pharm. Pharmacol., 1982, 34, 621-626.
17. Loftsson, T., Olafsd'ottir, B. J., Fridriksd'ottir, H. and Jonsdottir, S., Cyclodextrin complexation of NSAIDS: physicochemical characteristics. Eur. J. Pharm. Sci., 1993, 1, 95-101.
18. Loftsson, T., Sigurdardottir, A., The effect of polyvinylpyrrolidone and Hydroxypropyl methylcellulose on HP-β-CD complexation of hydrocortisone and its permeability through hairless mouse skin. Eur. J. Pharm. Sci., 1994, 2, 297-301. (Pubitemid 24360863)
19. Mura, P., Faucci, M. T. and Bettinetti, G. P., The influence of polyvinylpyrrolidone on naproxen complexation with hydroxypropyl-cyclodextrin. Eur. J. Pharm. Sci., 2001,13, 187-194. (Pubitemid 32288788)
20. Mura, P., Faucci, M. T. and Bettinetti, G. P., The influence of polyvinylpyrrolidone on naproxen complexation with hydroxypropyl-Cyclodextrin. Eur. J. Pharm. Sci., 2001, 13, 187-194. (Pubitemid 32288788)