A convenient route to functionalized 3-amino-6-bromofuro[3,2-b]pyridine-2-carboxamides

Tetrahedron

Volumn 66, Issue 25, 2010, Pages 4490-4494

  Bretéché, Anne ^a   Marchand, Pascal ^a   Nourrisson, Marie Renée ^a   De Nanteuil, Guillaume ^b   Duflos, Muriel ^a  

^a UNIVERSITÉ DE NANTES   (France)

^b INSTITUT DE RECHERCHES SERVIER   (France)

Author keywords

3 Amino 6 bromofuro 3,2 b pyridine 2 carbonitrile; 3 Amino 6 bromofuro 3,2 b pyridine 2 carboxamides; Heteroannulation

Indexed keywords

3 AMINO 6 BROMOFURO[3,2 B]PYRIDINE 2 CARBONITRILE; 3 AMINO 6 BROMOFURO[3,2 B]PYRIDINE 2 CARBOXAMIDE DERIVATIVE; AMIDE; CYANIDE; UNCLASSIFIED DRUG;

ARTICLE; CHEMICAL STRUCTURE; PRIORITY JOURNAL; SYNTHESIS;

EID: 77953230907     PISSN: 00404020     EISSN: None     Source Type: Journal    
DOI: 10.1016/j.tet.2010.04.071     Document Type: Article

References (22)

1. Kawaguchi, T.; Akatsuka, H.; Iijima, T.; Watanabe, T.; Murakami, J; Mitsui, T. Preparation of fused furan compounds as inhibitors of activated blood coagulation factor X PCT Int. Appl. WO 2004/063202, 2004.
2. Shiohara, H.; Nakamura, T.; Mukaiyama, H.; Kobayashi, S.; Jo, K. Preparation of furopyridine derivatives as adenosine A2A receptor antagonists PCT Int. Appl. WO 2006/137350, 2006.
3. Leger, S.; Hutchinson, J.H. Preparation of furo[3,2-b]pyridines and thieno[3,2-b]pyridines as inhibitors of leukotriene biosynthesis PCT Int. Appl. WO 9422869, 1994.
4. Mathes B.M., Hudziak K.J., Schaus J.M., Xu Y.-C., Nelson D.L., Wainscott D.B., Nutter S.E., Gough W.H., Branchek T.A., Zgombick J.M., and Filla S.A. Bioorg. Med. Chem. Lett. 14 (2004) 167-170
5. Chartoire A., Comoy C., and Fort Y. Tetrahedron 64 (2008) 10867-10873
6. Arcadi A., Cacchi S., Di Giuseppe S., Fabrizi G., and Marinelli F. Synlett (2002) 453-457
7. Cailly T., Lemaître S., Fabis F., and Rault S. Synthesis 20 (2007) 3247-3251
8. Brenner E., Baldwin R.M., and Tamagnan G. Tetrahedron Lett. 45 (2004) 3607-3610
9. Morgentin R., Jung F., Lamorlette M., Maudet M., Ménard M., Plé P., Pasquet G., and Renaud F. Tetrahedron 65 (2009) 757-764
10. Lin W., Chen L., and Knochel P. Tetrahedron 63 (2007) 2787-2797
11. Koch V., and Schnatterer S. Synthesis (1990) 497-498
12. Harris, N.; Higgs, C.; Wren S.; Dyke, H.J.; Price, S.; Cramp, S. Pyrimidine compounds as histamine modulators PCT Int. Appl. WO 2006/050965, 2006.
13. Zhang H.-Z., Kasibhatla S., Kuemmerle J., Kemnitzer W., Ollis-Mason K., Qiu L., Crogan-Grundy C., Tseng B., Drewe J., and Cai S.X. J. Med. Chem. 48 (2005) 5215-5223
14. Vicini P., Geronikaki A., Incerti M., Busonera B., Poni G., Cabras C.A., and La Colla P. Bioorg. Med. Chem. 11 (2003) 4785-4789
15. Nawrocka W., Sztuba B., Kowalska M.W., Liszkiewicz H., Wietrzyk J., Nasulewicz A., Pełczyńska M., and Opolski A. II Farmaco 59 (2004) 83-91
16. Abarghaz M., Kerbal A., and Bourguignon J.-J. Tetrahedron Lett. 36 (1995) 6463-6466
17. Mederski W.W.K.R., Osswald M., Dorsch D., Christadler M., Schmitges C.-J., and Wilm C. Bioorg. Med. Chem. Lett. 9 (1999) 619-622
18. Basel Y., and Hassner A. J. Org. Chem. 65 (2000) 6368-6380
19. Boger D.L., McKie J.A., Nishi T., and Ogiku T. J. Am. Chem. Soc. 118 (1996) 2301-2302
20. Hernández J.N., Crisóstomo F.R.P., Martín T., and Martín V.S. Eur. J. Org. Chem. (2007) 5050-5058
21. Varma R.S., and Naicker K.P. Org. Lett. 1 (1999) 189-191
22. Ji J., Schrimpf M.R., Sippy K.B., Bunnelle W.H., Li T., Anderson D.J., Faltynek C., Surowy C.S., Dyhring T., Ahring P.K., and Meyer M.D. J. Med. Chem. 50 (2007) 5493-5508