Synthesis and in vitro antiprotozoal evaluation of substituted phenalenone analogues

Bioorganic and Medicinal Chemistry

Volumn 18, Issue 12, 2010, Pages 4530-4534

  Rosquete, Laura I ^a   Cabrera Serra, M Gabriela ^a   Piñero, José E ^a   Martín Rodríguez, Patricia ^b,c   Fernández Pérez, Leandro ^b,c   Luis, Javier G ^a   McNaughton Smith, Grant ^a,c   Abad Grillo, Teresa ^a  

^a UNIVERSIDAD DE LA LAGUNA   (Spain)

^b UNIVERSITY OF LAS PALMAS DE GRAN CANARIA   (Spain)

^c CEAMED SA   (Spain)

Author keywords

Antiprotozoal activities; Substituted phenalenones; Synthesis

Indexed keywords

4 METHOXYPHENYL; 9 OXO 9H PHENALENE 1 CARBONITRILE; ANTIPARASITIC AGENT; ANTIPROTOZOAL AGENT; BENZNIDAZOLE; DOXORUBICIN; MOLECULAR SCAFFOLD; PENTAMIDINE; PHENALENE DERIVATIVE; PHENALENONE 1 ONE; UNCLASSIFIED DRUG; PHENALEN-1-ONE;

ANTIPROTOZOAL ACTIVITY; ARTICLE; CONTROLLED STUDY; DRUG SYNTHESIS; HUMAN; HUMAN CELL; IN VITRO STUDY; LEISHMANIASIS; NONHUMAN; TRYPANOSOMA CRUZI; TRYPANOSOMIASIS; CHEMISTRY; DRUG EFFECTS; SYNTHESIS; TOXICITY; TUMOR CELL LINE;

ANTIPROTOZOAL AGENTS; CELL LINE, TUMOR; HUMANS; LEISHMANIASIS; PENTAMIDINE; PHENALENES; TRYPANOSOMA CRUZI; TRYPANOSOMIASIS;

TRYPANOSOMA CRUZI;

EID: 77953139020     PISSN: 09680896     EISSN: None     Source Type: Journal    
DOI: 10.1016/j.bmc.2010.04.062     Document Type: Article

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