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Volumn 8, Issue 10, 2010, Pages 2457-2464

Synthesis of sulfonamide-based kinase inhibitors from sulfonates by exploiting the abrogated SN2 reactivity of 2,2,2- trifluoroethoxysulfonates

(6) Wong, Christopher a Griffin, Roger J a Hardcastle, Ian R a Northen, Julian S c Wang, Lan Zhen b Golding, Bernard T a

a NEWCASTLE UNIVERSITY (United Kingdom)

b NEWCASTLE UNIVERSITY (United Kingdom)

c Onyx Scientific Limited (United Kingdom)

Author keywords

[No Author keywords available]

Indexed keywords

ARYL RINGS; ATP-BINDING; CATALYTIC HYDROGENATION; DIMETHYLAMINOPYRIDINE; HUMAN CYCLIN-DEPENDENT KINASE 2; INHIBITORY ACTIVITY; KINASE INHIBITORS; METHYLENE GROUPS; N-ALKYLATION; NITRO GROUP; POTENTIAL INHIBITORS; STERIC EFFECT; STRUCTURE-ACTIVITY STUDIES; TETRA-HYDROFURAN; THREONINE KINASE; TRIFLUOROETHANOL;

AMINO ACIDS; CHLORINE COMPOUNDS; DEUTERIUM; ESTERS; ETHANOL; HEATING; HYDROCARBONS; HYDROGENATION; ORGANIC POLYMERS; PHOSPHATASES; SYNTHESIS (CHEMICAL);

SULFUR COMPOUNDS;

CYCLIN DEPENDENT KINASE 2; PROTEIN KINASE INHIBITOR; PURINE DERIVATIVE; SULFONAMIDE; SULFONIC ACID DERIVATIVE;

ARTICLE; CHEMISTRY; DRUG ANTAGONISM; HUMAN; SYNTHESIS;

CYCLIN-DEPENDENT KINASE 2; HUMANS; PROTEIN KINASE INHIBITORS; PURINES; SULFONAMIDES; SULFONIC ACIDS;

EID: 77952363221 PISSN: 14770520 EISSN: None Source Type: Journal
DOI: 10.1039/b922717b Document Type: Article

Times cited : (19)

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