Characterization of Polymorphic Systems Using Thermal Analysis

Polymorphism: in the Pharmaceutical Industry

Volumn , Issue , 2006, Pages 43-79

  Craig, Duncan Q M ^a  

^a UNIVERSITY OF EAST ANGLIA   (United Kingdom)

Author keywords

Additional thermal methods; Characterization of polymorphic systems; Combined approaches; Differential scanning calorimetry; Microthermal analysis; Pharmaceutical industry; Polymorphism; Thermal analysis; Thermal microscopy; Thermogravimetric analysis

Indexed keywords

EID: 77952030349     PISSN: None     EISSN: None     Source Type: Book    
DOI: 10.1002/3527607889.ch3     Document Type: Chapter

References (73)

1. H.G. Brittain, Physical Characterization of Pharmaceutical Solids, Marcel Dekker, New York, 1995.
2. H.G. Brittain, Polymorphism in Pharmaceutical Solids, Marcel Dekker, New York, 1999.
3. J. L. Ford, P. Timmins, Pharmaceutical Thermal Analysis, Ellis Horwood, Chichester, 1989.
4. D. Giron, Thermochim. Acta 1995, 248, 1-59.
5. W. C. Schinzer, M.S. Bergren, D. S. Aldrich, R. S. Chao, M.J. Dunn, A. Jeganathan, L.M. Madden, J. Pharm. Sci., 1997, 86, 1426-1431.
6. S. P. Velaga, R. Berger, J. Carlfors, Pharm. Res., 2002, 19, 1564-1571.
7. A. Burger, Sci. Pharm. 1977, 45, 269.
8. A. Burger, Acta Pharm. Technol. 1982, 28, 1-20.
9. Z. Dong, B. E. Padden, J. S. Salsbury, E. J. Munson, S. A. Schroeder, I. Prakash, D.J.W. Grant, Pharm. Res. 2002, 19, 330-336.
10. I.M. Vitez, J. Therm. Anal. Calorim. 2004, 78, 33-45.
11. P.M. Gosselin, R. Thibert, M. Preda, J. N. McMullen, Int. J. Pharm. 2003, 252, 225-233.
12. S. P. Velaga, R. Berger, J. Carlfors, Pharm. Res. 2002, 19, 1564-1571.
13. T. Oguchi, N. Sasaki, T. Hara, Y. Tozuka, K. Yamamoto, Int. J. Pharm., 2003, 253, 81-88.
14. E. Yonemochi, Y. Inoue, G. Buckton, A. Moffat, T. Oguchi, K. Yamamoto, Pharm. Res., 1999, 16, 835-840.
15. K. R. Morris, U.J. Griesser, C. J. Eckhardt, J. G. Stowell, Adv. Drug Deliv. Rev., 2001, 48, 91-114.
16. R. Panchagnula, P. Sundaramurthy, O. Pillai, S. Agrawal, Y. Raj, J. Pharm. Sci., 2004, 93, 1019-1029.
17. C. Telang, R. Suryanarayanan, L. Yu, Pharm. Res., 2003, 20, 1939-1945.
18. S. Chongprasert, S. A. Knopp, S. L. Nail, J. Pharm. Sci., 2001, 90. 1720-1728.
19. N. Zajc, A. Obreza, M. Bele, S. Srcic, Int. J. Pharm., 2005, 291, 51-58.
20. A. Burger, J.O. Henck, S. Hetz, J.M. Rollinger, A.A. Weissnicht, H. Stottner, J. Pharm. Sci., 2000, 89, 457-468.
21. C. P. Buckley, A. J. Kovacs, Coll. Polym. Sci., 1976, 254, 695-715.
22. K. Sato, Chem. Eng. Sci. 2001, 56, 2255-2265.
23. J. Hamdani, A. J. Moes, K. Amighi, Int. J. Pharm., 2003, 260, 47-57.
24. N. Khan, D.Q.M. Craig, J. Pharm. Sci., 2004, 93, 2962-2971.
25. J. B. Brubach, M. Ollivon, V. Jannin, B. Mahler, Bull. Tech. Gattefosse, 2004, 97, 41-50.
26. M.L.P. Leitao, J. Canotilho, M.S. C. Cruz, J. C. Pereira, A.T. Sousa, J. S. Redinha, J. Therm. Anal. Calorim., 2002, 68, 397-412.
27. Y. Yoshihashi, H. Kitano, E. Yonemochi, K. Terada, Int. J. Pharm., 2004, 204, 1-6.
28. D.Q.M. Craig, J.M. Newton, Int. J. Pharm., 1991, 74, 43-48.
29. M. Naoki, T. Yoshizawa, N. Fukushima, M. Ogiso, M. Yoshino, J. Phys. Chem. B, 1999, 103, 6309-6313.
30. L. Yu, J. Pharm. Sci. 1995, 84, 966.
31. M.R. Caira, S. A. Bourne, C. L. Oliver J. Therm. Anal. Calorim., 2004, 77, 597-605.
32. D. Giron, J. Therm. Anal. Calorim., 2001, 64, 37-60.
33. M. Grcman, F. Vrecer, A. Meden, J. Therm. Anal. Calorim., 2002, 68, 373-387.
34. F. Giordano, A. Rossi, J. R. Moyano, A. Gazzaniga, V. Massarotti, M. Bini, D. Capsoni, T. Peveri, E. Redenti, L. Carima, M.D. Alberi, M. Zanol, J. Pharm. Sci., 2001, 90, 1154-1163.
35. A. C. Schmidt, V. Niederwanger, U. J. Griesser, J. Therm. Anal. Calorim., 2004, 77, 639-652.
36. G. G.Z. Zhang, C. Gu, M.T. Zell, R.T. Burkhardt, E. J. Munson, D. J.W. Grant, J. Pharm. Sci., 2002, 91, 1089-1100.
37. J. Wouters, S. Vandevoorde, C. Culot, F. Docquir, D.M. Lambert, Chem. Phys. Lipids, 2002, 119, 13-21.
38. M. Ramakrishnan, V. Sheeba, S. S. Koormath, M.J. Swamy, Biochim. Biophys. Acta 1997, 1329, 302-310.
39. S. Pfeffer-Hennig, P. Piechon, M. Bellus, C. Goldbronn, E. Tedesco, J. Therm. Anal. Calorim., 2004, 77, 663-679.
40. F. G. Vogt, D.E. Cohen, J. D. Bowman, G. P. Spoors, G. E. Zuber, G.A. Trescher, P. C. Dell'Orco, L.M. Katrincic, C.W. Debrosse, R. C. Haltiwanger, J. Pharm. Sci., 2005, 94, 651-665.
41. M.R. Caira, K. A. Alkhamis, R.M. Obaidat, J. Pharm. Sci., 2004, 93, 601-611.
42. C. Nunes, R. Suryanarayanan, C. E. Botez, P.W. Stephens, J. Pharm. Sci., 2004, 93, 2800-2809.
43. A. D. Edwards, B.Y. Shekunov, R.T. Forbes, J. G. Grossman, P. York, J. Pharm. Sci., 2001, 90, 1106-1114.
44. P. Espeau, R. Ceolin, J.-L. Tamarit, M.-A. Perrin, J.-P. Gauchi, F. Leveiller, J. Pharm. Sci., 2005, 94, 524-539.
45. D. Giron, J. Therm. Anal. Calorim., 2002, 68, 335-357.
46. D. Giron, J. Therm. Anal. Calorim., 2001, 64, 37-60.
47. J. C. Sprunt, U.A. Jayasooriya, R.H. Wilson, Phys. Chem. Chem. Phys., 2000, 2, 4299-4305.
48. J. C. Sprunt, U.A. Jayasooriya, Appl. Spectrosc., 1997, 51, 1410.
49. C. Allais, G. Keller, P. Lesieur, M. Ollivon, F. Artzner, J. Therm. Anal. Calorim., 2003, 74, 723-728.
50. J. B. Brubach, M. Ollivon, V. Jannin, B. Mahler, C. Bourgaux, P. Lesieur, P. Roy, J. Phys. Chem. B, 2004, 108, 17721-17729.
51. M. Kuhnert-Brandstatter, Thermomicroscopy in the Analysis of Pharmaceuticals, International Series of Monographs on Analytical Chemistry, Vol. 45, Permagon Press, Oxford, 1971.
52. M. Kuhnert-Brandstatter, Thermomicroscopy of Organic Compounds, in Comprehensive Analytical Chemistry, Vol. 16, G. Svehla (ed.), Elsevier, Amsterdam, 1982.
53. I.M. Vitez, A.W. Newman, M. Davidovich, C. Kiesnowski, Thermochim. Acta, 1998, 324, 187.
54. S. L. Childs, L. J. Chyall, J.T. Dunlap, D.A. Coates, B. C. Stahly, G.P. Stahly, Cryst. Growth Design, 2004, 4, 441-449.
55. N.E. Variankaval, K. I. Jacob, S.M. Dinh, J. Cryst. Growth, 2000, 217, 320-331.
56. M. Szelagiewicz, C. Marcolli, S. Cianferani, A. P. Hard, A. Vit, A. Burkhard, M. von Raumer, U.C. Hofmeier, A. Zilian, E. Francotte, R. Schenker, J. Therm. Anal. Calorim., 1999, 57, 23-43.
57. P. O. Souillac, P. Dave, J. H. Rytting, Int. J. Pharm., 2002, 231, 185-196.
58. C.-H. Gu, D. J. W. Grant, J. Pharm. Sci., 2001, 90, 1277-1287.
59. M. Reading, Thermochim. Acta, 1994, 238, 295-307.
60. M. Reading, D. Elliot, V. L. Hill, J. Therm. Anal., 1993, 40, 949-955.
61. N. Coleman, D. Q.M. Craig, Int. J. Pharm., 1996, 135, 13-29.
62. B. Keymolen, J. L. Ford, M.W. Powell, A. R. Rajabi-Siahboomi, Thermochim. Acta, 2003, 397, 103-117.
63. K. Six, C. Leuner, J. Dressman, G. Verreck, J. Peeters, N. Blaton, P. Augustjins, R. Kinget, G. Van Den Mooter, J. Therm. Anal. Calorim., 2002, 68, 591-601.
64. K. Kawakami, Y. Ida, Thermochim. Acta, 2005, 427, 93-99.
65. R. Manduva, D.Q.M. Craig, V. L. Kett, D.A. Adkin, Am. Assoc. Pharmaceutical Sci., 2003, 5, T2267.
66. C. McGregor, M.H. Saunders, G. Buckton, R.D. Saklatvala, Thermochim. Acta, 2004, 417, 231-237.
67. A. Hammiche, D.M. Price, E. Dupas, G. Mills, A. Kulik, M. Reading, J.M.R. Weaver, H.M. Pollack, J. Microscopy- Oxford, 2000, 199, 180-190.
68. D.Q.M. Craig, V. L. Kett, C. S. Andrews, P. G. Royall, J. Pharm. Sci., 2002, 91, 1205-1213.
69. G.H.W. Sanders, C. J. Roberts, A. Danesh, A. J. Murray, D.M. Price, M.C. Davies, S. J. B. Tendler, M.J. Wilkins, J. Microsc.-Oxford, 2000, 198, 77-81.
70. J. R. Murphy, C.S. Andrews, D.Q.M. Craig, Pharm. Res., 2003, 20, 500-507.
71. R. Manduva, V. L. Kett, D.A. Adkin, D.Q.M. Craig, J. Pharm. Pharmacol., 2004, 56, 65S.
72. R. A. Shmeis, S. L. Krill, Thermochim. Acta, 2005, 427, 61-68.
73. N. Boutonnet-Fagegaltier, J. Menegotto, A. Lamure, H. Duplaa, A. Caron, C. Lacabanne, M. Bauer, J. Pharm. Sci., 2002, 91, 1548-1560.