Internalization of constitutively active N111G mutant of AT1 receptor induced by angiotensin II-receptor antagonists candesartan, losartan, and telmisartan: Comparison with valsartan

Journal of Pharmacological Sciences

Volumn 112, Issue 4, 2010, Pages 459-462

  Bhuiyan, Mohiuddin Ahmed ^a   Hossain, Murad ^a   Nakamura, Takashi ^a   Ozaki, Masanobu ^a   Nagatomo, Takafumi ^a  

^a NIIGATA UNIVERSITY OF PHARMACY AND APPLIED LIFE SCIENCES   (Japan)

Author keywords

Angiotensin II type 1 (AT1) receptor; Constitutively active mutant; Internalization

Indexed keywords

ANGIOTENSIN 1 RECEPTOR; ANGIOTENSIN 2 RECEPTOR ANTAGONIST; CANDESARTAN; LOSARTAN; TELMISARTAN; VALSARTAN;

ANIMAL CELL; ARTICLE; CELL PROLIFERATION; CELL STRAIN COS7; CELL VIABILITY; CELLULAR DISTRIBUTION; CONTROLLED STUDY; DRUG BINDING; DRUG MECHANISM; ENDOCYTOSIS; INTERNALIZATION; LIGAND BINDING; NONHUMAN; RAT; SIGNAL TRANSDUCTION; SITE DIRECTED MUTAGENESIS;

EID: 77951211465     PISSN: 13478613     EISSN: 13478648     Source Type: Journal    
DOI: 10.1254/jphs.09343SC     Document Type: Article

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