Design and synthesis of novel deoxybenzoin derivatives as FabH inhibitors and anti-inflammatory agents

Bioorganic and Medicinal Chemistry Letters

Volumn 20, Issue 6, 2010, Pages 2025-2028

  Li, Huan Qiu ^a   Luo, Yin ^a   Lv, Peng Cheng ^a   Shi, Lei ^a   Liu, Chang Hong ^a   Zhu, Hai Liang ^a  

^a NANJING UNIVERSITY   (China)

Author keywords

Anti inflammatory; ECE induced IL 8; Escherichia coli FabH; Halide deoxybenzoins

Indexed keywords

ANTIINFLAMMATORY AGENT; BETA KETOACYL ACYL CARRIER PROTEIN SYNTHASE III; DEOXYBENZOIN DERIVATIVE; ENZYME INHIBITOR; HALIDE; INTERLEUKIN 8; UNCLASSIFIED DRUG;

ANTIBACTERIAL ACTIVITY; ARTICLE; BIOLOGICAL ACTIVITY; CLINICAL RESEARCH; CONTROLLED STUDY; CYTOKINE PRODUCTION; DRUG DESIGN; DRUG SYNTHESIS; HUMAN; HUMAN CELL; MOLECULAR DOCKING; MUCOSA CELL; NONHUMAN; STOMACH MUCOSA;

ANTI-INFLAMMATORY AGENTS; BACTERIAL PROTEINS; BENZOIN; DRUG DESIGN; ENZYME-LINKED IMMUNOSORBENT ASSAY; MODELS, MOLECULAR;

ESCHERICHIA COLI; NEGIBACTERIA;

EID: 77549088194     PISSN: 0960894X     EISSN: None     Source Type: Journal    
DOI: 10.1016/j.bmcl.2010.01.032     Document Type: Article

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