Characterization of anticancer properties of 2,6-diisopropylphenol-docosahexaenoate and analogues in breast cancer cells

Bioorganic and Medicinal Chemistry

Volumn 18, Issue 5, 2010, Pages 1866-1874

  Harvey, Kevin A ^a   Xu, Zhidong ^a,b   Whitley, Phillip ^a   Jo Davisson, V ^b   Siddiqui, Rafat A ^a,c  

^a METHODIST RESEARCH INSTITUTE   (United States)

^b PURDUE UNIVERSITY   (United States)

^c INDIANA UNIVERSITY SCHOOL OF MEDICINE   (United States)

Author keywords

2,6 Diisopropylphenol; Breast cancer; Docosahexaenoic acid; Histone deacetylase; Lipid drug conjugates

Indexed keywords

2 CYCLOHEXANEPHENOL DOCOSAHEXAENOATE; 2 ISOPROPYLPHENOL DOCOSAHEXAENOATE; 2,4 DIISOPROPYLPHENOL DOCOSAHEXAENOATE; DOCOSAHEXAENOIC ACID; ESTER; ESTROGEN RECEPTOR ALPHA; HISTONE DEACETYLASE; PEROXISOME PROLIFERATOR ACTIVATED RECEPTOR ALPHA; PEROXISOME PROLIFERATOR ACTIVATED RECEPTOR GAMMA; PHENOL DOCOSAHEXAENOATE; PROPOFOL DOCOSAHEXAENOIC ACID; UNCLASSIFIED DRUG;

ANTINEOPLASTIC ACTIVITY; ARTICLE; BREAST CANCER; BREAST EPITHELIUM; CANCER CELL; CANCER INHIBITION; CELL LOSS; CONTROLLED STUDY; CYTOTOXICITY; DOSE RESPONSE; DRUG CONJUGATION; DRUG SCREENING; DRUG STRUCTURE; DRUG SYNTHESIS; ENZYME ACTIVITY; GENE EXPRESSION; HUMAN; HUMAN CELL; ONCOGENE NEU;

ANIMALS; ANTINEOPLASTIC AGENTS, HORMONAL; BREAST NEOPLASMS; CELL LINE, TUMOR; DOCOSAHEXAENOIC ACIDS; ESTROGEN RECEPTOR ALPHA; FEMALE; HISTONE DEACETYLASES; HUMANS; MICE; PROPOFOL; RECEPTOR, ERBB-2;

CHANDIPURA VIRUS;

EID: 77249091649     PISSN: 09680896     EISSN: None     Source Type: Journal    
DOI: 10.1016/j.bmc.2010.01.045     Document Type: Article

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