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Beilstein Journal of Organic Chemistry

Volumn 5, Issue , 2009, Pages

Synthesis and enzymatic evaluation of 2- and 4-aminothiazole-based inhibitors of neuronal nitric oxide synthase

(5) Lawton, Graham R a Ji, Haitao a Martásek, Pavel b,c Roman, Linda J b Silverman, Richard B a

a NORTHWESTERN UNIVERSITY (United States)

b UNIVERSITY OF TEXAS HEALTH SCIENCE CENTER AT SAN ANTONIO (United States)

c CHARLES UNIVERSITY (Czech Republic)

Author keywords

2 aminothiazole; 4 aminothiazole; Nitric oxide synthase inhibitor; NNOS

Indexed keywords

EID: 75949088334 PISSN: 18605397 EISSN: 18605397 Source Type: Journal
DOI: 10.3762/bjoc.5.28 Document Type: Article

Times cited : (12)

References (25)

1
- 28444498107
- Role of nitric oxide in Parkinson's disease
- DOI 10.1016/j.pharmthera.2005.05.007, PII S0163725805001178
- Zhang, L.; Dawson, V. L.; Dawson, T. M. Pharmacol. Ther. 2006, 109 33-41. doi:10.1016/j.pharmthera.2005.05.007 (Pubitemid 41740813)
- (2006) Pharmacology and Therapeutics , vol.109 , Issue.1-2 , pp. 33-41
- Zhang, L.¹ Dawson, V.L.² Dawson, T.M.³

2
- 0028124916
- Nitric oxide synthase activity is elevated in brain microvessels in Alzheimer's disease
- DOI 10.1006/bbrc.1994.2716
- Dorheim, M. A.; Tracey, W. R.; Pollock, J. S.; Grammas, P. Biochem. Biophys. Res. Commun. 1994, 205, 659-665. doi:10.1006/bbrc.1994.2716 (Pubitemid 24381677)
- (1994) Biochemical and Biophysical Research Communications , vol.205 , Issue.1 , pp. 659-665
- Dorheim, M.-A.¹ Tracey, W.R.² Pollock, J.S.³ Grammas, P.⁴

3
- 0036175596
- Mitochondrial contributions to tissue damage in stroke
- DOI 10.1016/S0197-0186(01)00122-X, PII S019701860100122X
- Sims, N. R.; Anderson, M. F. Neurochem. Int. 2002, 40, 511-526. doi:10.1016/S0197-0186(01)00122-X (Pubitemid 34159152)
- (2002) Neurochemistry International , vol.40 , Issue.6 , pp. 511-526
- Sims, N.R.¹ Anderson, M.F.²

4
- 0029865660
- Neonatal mice lacking neuronal nitric oxide synthase are less vulnerable to hypoxic-ischemic injury
- DOI 10.1006/nbdi.1996.0006
- Ferriero, D. M.; Holtzman, D. M.; Black, S. M.; Sheldon, R. A. Neurobiol. Dis. 1996, 3, 64-71. doi:10.1006/nbdi.1996.0006 (Pubitemid 26145406)
- (1996) Neurobiology of Disease , vol.3 , Issue.1 , pp. 64-71
- Ferriero, D.M.¹ Holtzman, D.M.² Black, S.M.³ Sheldon, R.A.⁴

5
- 0141923092
- G-nitro-L-arginine methyl ester (L-NAME) treatment is similar in immature and adult Wistar rats
- DOI 10.1042/CS20030078
- Zicha, J.; Pechanová, O.; Dobešová, Z.; Kuneš. J. Clin. Sci. 2003, 105, 483-489. doi:10.1042/CS20030078 (Pubitemid 37249175)
- (2003) Clinical Science , vol.105 , Issue.4 , pp. 483-489
- Zicha, J.¹ Pechanova, O.² Dobesova, Z.³ Kunes, J.⁴

6
- 23844509261
- Selective neuronal nitric oxide synthase inhibitors
- DOI 10.2174/1568026054679317
- Erdal, E. P.; Litzinger, E. A.; Seo, J. W.; Zhu, Y. Q.; Ji, H.; Silverman, R. B. Curr. Top. Med. Chem. 2005, 5, 603-624. doi:10.2174/ 1568026054679317 (Pubitemid 41179723)
- (2005) Current Topics in Medicinal Chemistry , vol.5 , Issue.7 , pp. 603-624
- Erdal, E.P.¹ Litzinger, E.A.² Seo, J.³ Zhu, Y.⁴ Ji, H.⁵ Silverman, R.B.⁶

7
- 35348853741
- The role of size and charge for blood-brain barrier permeation of drugs and fatty acids
- DOI 10.1007/s12031-007-0055-y
- Seelig, A. J. Mol. Neurosci. 2007, 33, 32-41. doi:10.1007/s12031-007- 0055-y (Pubitemid 47574956)
- (2007) Journal of Molecular Neuroscience , vol.33 , Issue.1 , pp. 32-41
- Seelig, A.¹

8
- 41149145121
- doi:10.1021/ja0772041
- Ji, H.; Stanton, B. Z.; Igarashi, J.; Li, H.; Martásek, P.; Roman, L. J.; Poulos, T. L.; Silverman, R. B. J. Am. Chem. Soc. 2008, 130, 3900-3914. doi:10.1021/ja0772041
- (2008) J. Am. Chem. Soc. , vol.130 , pp. 3900-3914
- Ji, H.¹ Stanton, B.Z.² Igarashi, J.³ Li, H.⁴ Martásek, P.⁵ Roman, L.J.⁶ Poulos, T.L.⁷ Silverman, R.B.⁸

9
- 61449263657
- doi:10.1021/jm801220a
- Ji, H.; Li, H.; Martásek, P.; Roman, L. J.; Poulos, T. L.; Silverman, R. B. J. Med. Chem. 2009, 52, 779-797. doi:10.1021/jm801220a
- (2009) J. Med. Chem. , vol.52 , pp. 779-797
- Ji, H.¹ Li, H.² Martásek, P.³ Roman, L.J.⁴ Poulos, T.L.⁵ Silverman, R.B.⁶

10
- 62549102043
- doi:10.1002/ana.21555
- Ji, H.; Tan, S.; Igarashi, J.; Li, H.; Derrick, M.; Martásek, P.; Roman, L. J.; Vásquez-Vivar, J.; Poulos, T. L.; Silverman, R. B. Ann. Neurol. 2009, 65, 209-217. doi:10.1002/ana.21555
- (2009) Ann. Neurol. , vol.65 , pp. 209-217
- Ji, H.¹ Tan, S.² Igarashi, J.³ Li, H.⁴ Derrick, M.⁵ Martásek, P.⁶ Roman, L.J.⁷ Vásquez-Vivar, J.⁸ Poulos, T.L.⁹ Silverman, R.B.¹⁰

11
- 84962450101
- doi:10.1002/cphc.200400171
- Schmidtam Busch, M.; Knapp, E. W. ChemPhysChem 2004, 5, 1513-1522. doi:10.1002/cphc.200400171
- (2004) Chem Phys Chem , vol.5 , pp. 1513-1522
- Schmidtam Busch, M.¹ Knapp, E.W.²

12
- 75949114112
- in press
- Igarashi, J.; Li, H.; Jamal, J.; Ji, H.; Fang, J.; Silverman, R. B.; Poulos, T. L. J. Med. Chem. 2009, 52, in press.
- (2009) J. Med. Chem. , vol.52
- Igarashi, J.¹ Li, H.² Jamal, J.³ Ji, H.⁴ Fang, J.⁵ Silverman, R.B.⁶ Poulos, T.L.⁷

13
- 0037048352
- doi:10.1016/S0957-4166(02)00477-9
- Allevi, P.; Galligani, M.; Anastasia, M. Tetrahedron: Asymmetry 2002, 13, 1901-1910. doi:10.1016/S0957-4166(02)00477-9
- (2002) Tetrahedron: Asymmetry , vol.13 , pp. 1901-1910
- Allevi, P.¹ Galligani, M.² Anastasia, M.³

14
- 0021952977
- Synthesis of the dioxabicyclononane unit of tirandamycin
- DOI 10.1016/S0040-4039(00)98954-8
- Kelly, T. R.; Chandrakumar, N. S.; Cutting, J. D.; Goehring, R. R.; Weibel, F. R. Tetrahedron Lett. 1985, 26, 2173-2176. doi:10.1016/S0040-4039(00) 98954-8 (Pubitemid 15097582)
- (1985) Tetrahedron Letters , vol.26 , Issue.18 , pp. 2173-2176
- Kelly, T.R.¹ Chandrakumar, N.S.² Cutting, J.D.³

15
- 9644268880
- Simple microwave-assisted method for the synthesis of primary thioamides from nitriles
- DOI 10.1055/s-2004-834812
- Bagley, M. C.; Chapaneri, K.; Glover, C.; Merritt, E. A. Synlett 2004, 2615-2617. doi:10.1055/s-2004-834812 (Pubitemid 39577041)
- (2004) Synlett , Issue.14 , pp. 2615-2617
- Bagley, M.C.¹ Chapaneri, K.² Glover, C.³ Merritt, E.A.⁴

16
- 0003549051
- Barton, A.; Breukelman, S. P.; Kaye, P. T.; Meakins, G. D.; Morgan, D. J. J. Chem. Soc., Perkin Trans. 1 1982, 159-164.
- (1982) J. Chem. Soc., Perkin Trans. 1 , pp. 159-164
- Barton, A.¹ Breukelman, S.P.² Kaye, P.T.³ Meakins, G.D.⁴ Morgan, D.J.⁵

17
- 12344262119
- Synthesis of novel N-methylated thiazole-based cyclic octa- and dodecapeptides
- DOI 10.1016/j.tet.2004.11.032, PII S0040402004019040
- Dudin, L.; Pattenden, G.; Viljoen, M. S.; Wilson, C. Tetrahedron 2005, 61, 1257-1267. doi:10.1016/j.tet.2004.11.032 (Pubitemid 40126728)
- (2005) Tetrahedron , vol.61 , Issue.5 , pp. 1257-1267
- Dudin, L.¹ Pattenden, G.² Viljoen, M.S.³ Wilson, C.⁴

18
- 0037652079
- doi:10.1002/ejoc.200210682
- van Well, R. M.; Overkleeft, H. S.; van Boom, J. H.; Coop, A.; Wang, J. B.; Wang, H. Y.; van der Marel, G. A.; Overhand, M. Eur. J. Org. Chem. 2003, 1704-1710. doi:10.1002/ejoc.200210682
- (2003) Eur. J. Org. Chem. , pp. 1704-1710
- Van Well, R.M.¹ Overkleeft, H.S.² Van Boom, J.H.³ Coop, A.⁴ Wang, J.B.⁵ Wang, H.Y.⁶ Van Der Marel, G.A.⁷ Overhand, M.⁸

19
- 33746023969
- Remote protection prevents unwanted cyclizations with 2-aminopyridines
- DOI 10.1016/j.tetlet.2006.06.091, PII S0040403906012639
- Lawton, G. R.; Ji, H.; Silverman, R. B. Tetrahedron Lett. 2006, 47, 6113-6115. doi:10.1016/j.tetlet.2006.06.091 (Pubitemid 44066424)
- (2006) Tetrahedron Letters , vol.47 , Issue.34 , pp. 6113-6115
- Lawton, G.R.¹ Ji, H.² Silverman, R.B.³

20
- 0010208764
- doi:10.1021/ja01636a038
- Taylor, E. C.; Wolinsky, J.; Lee, H. H. J. Am. Chem. Soc. 1954, 76, 1866-1870. doi:10.1021/ja01636a038
- (1954) J. Am. Chem. Soc. , vol.76 , pp. 1866-1870
- Taylor, E.C.¹ Wolinsky, J.² Lee, H.H.³

21
- 0029114645
- doi:10.1073/pnas.92.18.8428
- Roman, L. J.; Sheta, E. A.; Martasek, P.; Gross, S. S.; Liu, Q.; Masters, B. S. S. Proc. Natl. Acad. Sci. U. S. A. 1995, 92, 8428-8432. doi:10.1073/pnas.92.18.8428
- (1995) Proc. Natl. Acad. Sci. U. S. A. , vol.92 , pp. 8428-8432
- Roman, L.J.¹ Sheta, E.A.² Martasek, P.³ Gross, S.S.⁴ Liu, Q.⁵ Masters, B.S.S.⁶

22
- 0029874753
- Characterization of bovine endothelial nitric oxide synthase expressed in E. coli
- DOI 10.1006/bbrc.1996.0238
- Martásek, P.; Liu, Q.; Liu, J. W.; Roman, L. J.; Gross, S. S.; Sessa, W. C.; Masters, B. S. S. Biochem. Biophys. Res. Commun. 1996, 219, 359-365. doi:10.1006/bbrc.1996.0238 (Pubitemid 26090277)
- (1996) Biochemical and Biophysical Research Communications , vol.219 , Issue.2 , pp. 359-365
- Martasek, P.¹ Liu, Q.² Liu, J.³ Roman, L.J.⁴ Gross, S.S.⁵ Sessa, W.C.⁶ Masters, B.S.S.⁷

23
- 0026323665
- Hevel, J. M.; White, K. A.; Marletta, M. A. J. Biol. Chem. 1991, 266, 22789-22791.
- (1991) J. Biol. Chem. , vol.266 , pp. 22789-22791
- Hevel, J.M.¹ White, K.A.² Marletta, M.A.³

24
- 0028245391
- doi:10.1016/S0076-6879(94)33028-X
- Hevel, J. M.; Marletta, M. A. Method Enzymol. 1994, 233, 250-258. doi:10.1016/S0076-6879(94)33028-X
- (1994) Method Enzymol. , vol.233 , pp. 250-258
- Hevel, J.M.¹ Marletta, M.A.²

25
- 0034604846
- Substituted 2-ammopyridines as inhibitors of nitric oxide synthases
- DOI 10.1016/S0960-894X(00)00389-9, PII S0960894X00003899
- Hagmann, W. H.; Caldwell, C. G.; Chen, P.; Durette, P. L.; Esser, C. K.; Lanza, T. J.; Kopka, I. E.; Guthikonda, R.; Shah, S. K.; MacCoss, M.; Chabin, R. M.; Fletcher, D.; Grant, S. K.; Green, B. G.; Humes, J. L.; Kelly, T. M.; Luell, S.; Meurer, R.; Moore, V.; Pacholok, S. G.; Pavia, T.; Williams, H. R.; Wong, K. K. Bioorg. Med. Chem. Lett. 2000, 10, 1975-1978. doi:10.1016/S0960- 894X(00)00389-9 (Pubitemid 30663353)
- (2000) Bioorganic and Medicinal Chemistry Letters , vol.10 , Issue.17 , pp. 1975-1978
- Hagmann, W.K.¹ Caldwell, C.G.² Chen, P.³ Durette, P.L.⁴ Esser, C.K.⁵ Lanza, T.J.⁶ Kopka, I.E.⁷ Guthikonda, R.⁸ Shah, S.K.⁹ MacCoss, M.¹⁰ Chabin, R.M.¹¹ Fletcher, D.¹² Grant, S.K.¹³ Green, B.G.¹⁴ Humes, J.L.¹⁵ Kelly, T.M.¹⁶ Luell, S.¹⁷ Meurer, R.¹⁸ Moore, V.¹⁹ Pacholok, S.G.²⁰ more..

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