An evaluation of a fluorometric method for determining binding parameters of drug-carrier complexes using mathematical models based on total drug concentration

Journal of Fluorescence

Volumn 19, Issue 4, 2009, Pages 747-753

  Chanvorachote, Boontarika ^a   Nimmannit, Ubonthip ^a   Muangsiri, Walaisiri ^a   Kirsch, Lee ^b  

^a CHULALONGKORN UNIVERSITY   (Thailand)

^b UNIVERSITY OF IOWA   (United States)

Author keywords

And Drugcarrier complexes; Capacity constant; Dissociation constant; Drug binding; Fluorescence methods

Indexed keywords

BINDING ISOTHERMS; BINDING MODELS; BINDING PARAMETER; DAPTOMYCIN; DISSOCIATION CONSTANT; DRUG BINDING; DRUG CONCENTRATION; FLUORESCENCE METHOD; FLUOROMETRIC METHOD; LIPOPEPTIDES; MATHEMATICAL SIMULATIONS; MODE OF BINDING; MODEL DRUGS; MODEL EQUATIONS; NON-LINEAR REGRESSION ANALYSIS; PH-DEPENDENT; POLYAMIDOAMINE DENDRIMERS; SENSITIVITY OF PARAMETERS; SITE BINDING;

ANTIBIOTICS; CARRIER CONCENTRATION; DENDRIMERS; DISSOCIATION; DYES; FLUORESCENCE; REGRESSION ANALYSIS; SENSITIVITY ANALYSIS;

MATHEMATICAL MODELS;

ANTIINFECTIVE AGENT; DAPTOMYCIN; DRUG CARRIER; PAMAM STARBURST; POLYAMINE;

ARTICLE; BINDING SITE; CHEMICAL MODEL; CHEMISTRY; COMPUTER SIMULATION; EVALUATION; FLUORESCENCE; FLUOROMETRY; METHODOLOGY; PH;

ANTI-BACTERIAL AGENTS; BINDING SITES; COMPUTER SIMULATION; DAPTOMYCIN; DRUG CARRIERS; FLUORESCENCE; FLUOROMETRY; HYDROGEN-ION CONCENTRATION; MODELS, CHEMICAL; POLYAMINES;

EID: 70349258130     PISSN: 10530509     EISSN: None     Source Type: Journal    
DOI: 10.1007/s10895-009-0471-1     Document Type: Article

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