Synthesis and in vivo diuretic activity of biphenyl benzothiazole-2- carboxamide derivatives

Acta Poloniae Pharmaceutica - Drug Research

Volumn 66, Issue 4, 2009, Pages 387-392

  Yar, Mohammad Shahar ^a   Ansari, Zaheen Hasan ^a  

^a HAMDARD UNIVERSITY   (India)

Author keywords

Benzothiazole; Biphenyl; Carboxamide; Diuretic activity

Indexed keywords

2 AMINOBENZOTHIAZOLE; ACETAZOLAMIDE; BIPHENYL ACID CHLORIDE; BIPHENYL DERIVATIVE; DIURETIC AGENT; N (1,3 BENZOTHIAZOL 2 YL) 1,1' BIPHENYL 4 CARBOXAMIDE; N (4 METHOXY 1,3 BENZOTHIAZOL 2 YL) 1,1' BIPHENYL 4 CARBOXAMIDE; N (4 METHYL 1,3 BENZOTHIAZOL 2 YL) 1,1' BIPHENYL 4 CARBOXAMIDE; N (5 CHLORO 1,3 BENZOTHIAZOL 2 YL) 1,1' BIPHENYL 4 CARBOXAMIDE; N (5 CHLORO 6 FLUORO 1,3 BENZOTHIAZOL 2 YL) 1,1' BIPHENYL 4 CARBOXAMIDE; N (5 METHYL 1,3 BENZOTHIAZOL 2 YL) 1,1' BIPHENYL 4 CARBOXAMIDE; N (6 BROMO 1,3 BENZOTHIAZOL 2 YL) 1,1' BIPHENYL 4 CARBOXAMIDE; N (6 CHLORO 1,3 BENZOTHIAZOL 2 YL) 1,1' BIPHENYL 4 CARBOXAMIDE; N (6 FLUORO 1,3 BENZOTHIAZOL 2 YL) 1,1' BIPHENYL 4 CARBOXAMIDE; N (6 METHOXY 1,3 BENZOTHIAZOL 2 YL) 1,1' BIPHENYL 4 CARBOXAMIDE; N (6 METHYL 1,3 BENZOTHIAZOL 2 YL) 1,1' BIPHENYL 4 CARBOXAMIDE; POTASSIUM ION; SODIUM ION; THIAZOLE DERIVATIVE; UNCLASSIFIED DRUG; UREA; BENZOTHIAZOLE DERIVATIVE;

ANIMAL EXPERIMENT; ARTICLE; CONTROLLED STUDY; DIURETIC ACTIVITY; DRUG EXCRETION; DRUG POTENCY; DRUG SYNTHESIS; NONHUMAN; RAT; URINARY EXCRETION; ANIMAL; STRUCTURE ACTIVITY RELATION; SYNTHESIS;

ANIMALS; BENZOTHIAZOLES; DIURETICS; RATS; STRUCTURE-ACTIVITY RELATIONSHIP;

EID: 69849105373     PISSN: 00016837     EISSN: None     Source Type: Journal    
DOI: None     Document Type: Article

References (12)

1. Emil F.: J. Liebigs Ann. Chem. 212, 316 (1882);
2. Augustin M., Richter M., Salas S.: J. Prakt. Chem. 322, 55 (1980);
3. Hofmann A. W.: Ber. 12, 2539 (1879);
4. Junke W., Feng P., Ju-li J., Zhi-jin L., Le-yong W., Junfeng B., Yi P.: Tetrahedron Lett. 49, 467 (2008).
5. Pattan S. R., Babu S. N., Angadi J.: Ind. J. Heterocycl. Chem. 11, 333 (2002).
6. Palagiano F., Arenare L., De Caprariis P., Grandolini G., Ambrogi V., Perioli L.: Farmaco 51, 483 (1996).
7. Murugan V., Kumar S., Prabu K. S., Suresh B., Reddy V. M.: Ind. J. Heterocycl. Chem. 14, 175 (2004).
8. Paranjape S. D., Bobade A. S., Khadse B. G.: Arzneimittelforschung 51, 916 (2001).
9. Jimonet P., Audiau F., Barreau M., et al.: J. Med. Chem. 42, 2828 (1999).
10. Khadikare P. V., Shalini S., Jyoti S., Maya I., Rajika M.: Arkivoc XVI, 1 (2006).
11. Srivastava S. K., Yadav R., Srivastava S. D.: Ind. J. Chem. 43B, 399 (2004).
12. nd ed., p. 323-325, Springer Verlag, Berlin, Heidelberg, New York 2002.