The synthesis and activity evaluation of a Bestatin derivative (LYP) as an aminopeptidase N inhibitor

Letters in Drug Design and Discovery

Volumn 6, Issue 6, 2009, Pages 420-423

  Luan, Yepeng ^a   Wang, Xuejian ^a   Zhu, Huawei ^a   Qu, Xianjun ^a   Fang, Hao ^a   Xu, Wenfang ^a  

^a SHANDONG UNIVERSITY   (China)

Author keywords

A549; Aminopeptidase N; Bestatin; ES 2; HL 60; N; N dimethyl ethanolamine

Indexed keywords

BESTATIN; BESTATIN DERIVATIVE; PEPTIDE HYDROLASE INHIBITOR;

ANIMAL EXPERIMENT; ANIMAL MODEL; ANIMAL TISSUE; ANTINEOPLASTIC ACTIVITY; ARTICLE; CONTROLLED STUDY; DRUG EFFICACY; DRUG SYNTHESIS; ENZYME INHIBITION; HUMAN; HUMAN CELL; IC 50; LIVER TUMOR; MOUSE; NONHUMAN; PRIORITY JOURNAL;

EID: 69549117147     PISSN: 15701808     EISSN: None     Source Type: Journal    
DOI: 10.2174/157018009789057535     Document Type: Article

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