Blood plasma model predictions for the proposed bone-seeking radiopharmaceutical [117mSn]Sn(IV)-N,N′,N′-trimethylenephosphonate-po ly(ethyleneimine)

Journal of Inorganic Biochemistry

Volumn 103, Issue 9, 2009, Pages 1265-1272

  Jansen, David R ^a,b   Krijger, Gerard C ^b   Wagener, Judith ^a   Senwedi, Ratanang M ^c   Gabanamotse, Kenneth ^c   Kgadiete, Mpho ^c   Kolar, Zvonimir I ^b   Zeevaart, Jan Rijn ^a,c  

^a NECSA   (South Africa)

^b DELFT UNIVERSITY OF TECHNOLOGY   (Netherlands)

^c NORTH WEST UNIVERSITY   (South Africa)

Author keywords

117mSn Sn(IV) PEI MP; Amino acids; Blood plasma model; Bone metastasis; Radiopharmaceutical; Stability constants

Indexed keywords

AMINO ACID; CALCIUM ION; COPPER ION; GLASS; GLUTAMINE; LEAD; LIGAND; N,N',N' TRIMETHYLENEPHOSPHONATE POLYETHYLENEIMINE SN 117M; RADIOPHARMACEUTICAL AGENT; TIN; UNCLASSIFIED DRUG; ZINC ION;

ARTICLE; BINDING COMPETITION; COMPLEX FORMATION; CONTROLLED STUDY; DRUG STABILITY; DRUG STRUCTURE; ELECTRODE; ENERGY; IN VITRO STUDY; IN VIVO STUDY; INTRAVENOUS DRUG ADMINISTRATION; MOLECULAR STABILITY; PLASMA; POTENTIOMETRY; PREDICTION; THERMODYNAMICS;

AMINO ACIDS; BONE NEOPLASMS; CALCIUM; CARBOXYLIC ACIDS; COMPUTER SIMULATION; DATABASES, FACTUAL; DRUG STABILITY; GLUTAMINE; HUMANS; LIGANDS; MODELS, BIOLOGICAL; MOLECULAR STRUCTURE; ORGANOTIN COMPOUNDS; POTENTIOMETRY; RADIOPHARMACEUTICALS; RADIOTHERAPY; TIN RADIOISOTOPES;

ANIMALIA;

EID: 69249220069     PISSN: 01620134     EISSN: None     Source Type: Journal    
DOI: 10.1016/j.jinorgbio.2009.07.007     Document Type: Article

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