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Volumn , Issue , 2006, Pages 213-221

Varenicline: An α4 Β2 nicotinic acetylcholine receptor partial agonist as an aid to smoking cessation

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EID: 68549089216     PISSN: None     EISSN: None     Source Type: Book    
DOI: None     Document Type: Chapter
Times cited : (4)

References (26)
  • 2
    • 0028849333 scopus 로고
    • Nicotine medications for smoking cessation
    • Henningfield, J.E., Nicotine medications for smoking cessation, New Engl. J. Med., 333(18), 1196-1203, 1995.
    • (1995) New Engl. J. Med. , vol.333 , Issue.18 , pp. 1196-1203
    • Henningfield, J.E.1
  • 3
    • 0035708568 scopus 로고    scopus 로고
    • Cellular mechanisms of nicotine addiction
    • Dani, J.A. and De Biasi, M., Cellular mechanisms of nicotine addiction, Pharmacol. Biochem. Behav., 70(4), 439-446, 2001.
    • (2001) Pharmacol. Biochem. Behav. , vol.70 , Issue.4 , pp. 439-446
    • Dani, J.A.1    De Biasi, M.2
  • 4
    • 0034732318 scopus 로고    scopus 로고
    • Role of dopamine in the behavioural actions of nicotine related addiction
    • Di Chiara, G., Role of dopamine in the behavioural actions of nicotine related addiction, Eur. J. Pharmacol., 393, 295-314, 2000.
    • (2000) Eur. J. Pharmacol. , vol.393 , pp. 295-314
    • Di Chiara, G.1
  • 5
    • 0343933624 scopus 로고
    • Drugs abused by humans preferentially increase synaptic dopamine concentrations in the mesolimbic system of freely moving rats
    • Di Chiara, G. and Imperato, A., Drugs abused by humans preferentially increase synaptic dopamine concentrations in the mesolimbic system of freely moving rats, Proc. Natl. Acad. Sci. USA, 85(14), 5274-5278, 1988.
    • (1988) Proc. Natl. Acad. Sci. USA , vol.85 , Issue.14 , pp. 5274-5278
    • Di Chiara, G.1    Imperato, A.2
  • 6
    • 0029943635 scopus 로고    scopus 로고
    • Effects of nicotine on the nucleus accumbens and similarity to those of addictive drugs [see comment]
    • Pontieri, F.E. et al., Effects of nicotine on the nucleus accumbens and similarity to those of addictive drugs [see comment], Nature, 382(6588), 255-257, 1996.
    • (1996) Nature , vol.382 , Issue.6588 , pp. 255-257
    • Pontieri, F.E.1
  • 7
    • 8344245466 scopus 로고    scopus 로고
    • Nicotine activation of alpha4* receptors: Sufficient for reward, tolerance, and sensitization
    • Tapper, A.R. et al., Nicotine activation of alpha4* receptors: sufficient for reward, tolerance, and sensitization, Science, 306(5698), 1029-1032, 2004.
    • (2004) Science , vol.306 , Issue.5698 , pp. 1029-1032
    • Tapper, A.R.1
  • 8
    • 0032495515 scopus 로고    scopus 로고
    • Acetylcholine receptors containing the beta2 subunit are involved in the reinforcing properties of nicotine
    • Picciotto, M.R. et al., Acetylcholine receptors containing the beta2 subunit are involved in the reinforcing properties of nicotine, Nature, 391(6663), 173-177, 1998.
    • (1998) Nature , vol.391 , Issue.6663 , pp. 173-177
    • Picciotto, M.R.1
  • 9
    • 21844438972 scopus 로고    scopus 로고
    • Nicotine reinforcement and cognition restored by targeted expression of nicotinic receptors
    • Maskos, U. et al., Nicotine reinforcement and cognition restored by targeted expression of nicotinic receptors, Nature, 436(7047), 103-107, 2005.
    • (2005) Nature , vol.436 , Issue.7047 , pp. 103-107
    • Maskos, U.1
  • 10
    • 0015209962 scopus 로고
    • Cytisine (Tabex) as a pharmaceutical aid in stopping smoking [in German]
    • Scharfenberg, G., Benndorf, S., and Kempe, G., Cytisine (Tabex) as a pharmaceutical aid in stopping smoking [in German], Dtsch. Gesundheitsw., 26(10), 463-465, 1971.
    • (1971) Dtsch. Gesundheitsw , vol.26 , Issue.10 , pp. 463-465
    • Scharfenberg, G.1    Benndorf, S.2    Kempe, G.3
  • 11
    • 0028153758 scopus 로고
    • Partial agonist properties of cytisine on neuronal nicotinic receptors containing the beta2 subunit
    • Papke, R.L. and Heinemann, S.F., Partial agonist properties of cytisine on neuronal nicotinic receptors containing the beta2 subunit, Mol. Pharmacol., 45(1), 142-149, 1994.
    • (1994) Mol. Pharmacol , vol.45 , Issue.1 , pp. 142-149
    • Papke, R.L.1    Heinemann, S.F.2
  • 12
    • 0014446583 scopus 로고
    • Some studies on cytisine and its methylated derivatives
    • Barlow, R.B. and McLeod, L.J., Some studies on cytisine and its methylated derivatives, Br. J. Pharmacol., 35(1), 161-174, 1969.
    • (1969) Br. J. Pharmacol. , vol.35 , Issue.1 , pp. 161-174
    • Barlow, R.B.1    McLeod, L.J.2
  • 13
    • 0025289331 scopus 로고
    • Behavioural and pharmacokinetic studies on nicotine, cytisine and lobeline
    • Reavill, C. et al., Behavioural and pharmacokinetic studies on nicotine, cytisine and lobeline, Neuropharmacology, 29(7), 619-624, 1990.
    • (1990) Neuropharmacology , vol.29 , Issue.7 , pp. 619-624
    • Reavill, C.1
  • 14
    • 0027931492 scopus 로고
    • Mecamylamine combined with nicotine skin patch facilitates smoking cessation beyond nicotine patch treatment alone
    • Rose, J.E. et al., Mecamylamine combined with nicotine skin patch facilitates smoking cessation beyond nicotine patch treatment alone, Clin. Pharmacol. Ther., 56, 86-99, 1994.
    • (1994) Clin. Pharmacol. Ther. , vol.56 , pp. 86-99
    • Rose, J.E.1
  • 15
    • 0018147760 scopus 로고
    • Human pharmacology and abuse potential of the analgesic buprenorphine: A potential agent for treating narcotic addiction
    • Jasinski, D.R., Pevnick, J.S., and Griffith, J.D., Human pharmacology and abuse potential of the analgesic buprenorphine: a potential agent for treating narcotic addiction, Arch. Gen. Psychiatry, 35(4), 501-516, 1978.
    • (1978) Arch. Gen. Psychiatry , vol.35 , Issue.4 , pp. 501-516
    • Jasinski, D.R.1    Pevnick, J.S.2    Griffith, J.D.3
  • 16
    • 23344447151 scopus 로고    scopus 로고
    • Medication development for addictive disorders: The state of the science
    • Vocci, F.J., Acri, J., and Elkashef, A., Medication development for addictive disorders: the state of the science, Am. J. Psychiatry, 162(8), 1432-1440, 2005.
    • (2005) Am. J. Psychiatry , vol.162 , Issue.8 , pp. 1432-1440
    • Vocci, F.J.1    Acri, J.2    Elkashef, A.3
  • 17
    • 19944400775 scopus 로고    scopus 로고
    • In pursuit of alpha4beta2 nicotinic receptor partial agonists for smoking cessation: Carbon analogs of (-)-cytisine
    • Coe, J.W. et al., In pursuit of alpha4beta2 nicotinic receptor partial agonists for smoking cessation: carbon analogs of (-)-cytisine, Bioorg. Med. Chem. Lett., 15(12), 2974-9, 2005.
    • (2005) Bioorg. Med. Chem. Lett. , vol.15 , Issue.12 , pp. 2974-2979
    • Coe, J.W.1
  • 18
    • 25844498213 scopus 로고    scopus 로고
    • 3,5-Bicyclic aryl piperidines: A novel class of alpha4beta2 neuronal nicotinic receptor partial agonists for smoking cessation
    • Coe, J.W. et al.,3,5-Bicyclic aryl piperidines: a novel class of alpha4beta2 neuronal nicotinic receptor partial agonists for smoking cessation, Bioorg. Med. Chem. Lett., 15(22), 4889-4897, 2005.
    • (2005) Bioorg. Med. Chem. Lett. , vol.15 , Issue.22 , pp. 4889-4897
    • Coe, J.W.1
  • 19
    • 20844441945 scopus 로고    scopus 로고
    • Varenicline: An alpha4beta2 nicotinic receptor partial agonist for smoking cessation
    • Coe, J.W. et al., Varenicline: an alpha4beta2 nicotinic receptor partial agonist for smoking cessation, J. Med. Chem., 48(10), 3474-3477, 2005.
    • (2005) J. Med. Chem , vol.48 , Issue.10 , pp. 3474-3477
    • Coe, J.W.1
  • 20
    • 0034092892 scopus 로고    scopus 로고
    • Effects of the competitive nicotinic antagonist erysodine on behavior occasioned or maintained by nicotine: Comparison with mecamylamine
    • Mansbach, R.S., Chambers, L.K., and Rovetti, C.C., Effects of the competitive nicotinic antagonist erysodine on behavior occasioned or maintained by nicotine: comparison with mecamylamine, Psychopharmacology, 148(3), 234-242, 2000.
    • (2000) Psychopharmacology , vol.148 , Issue.3 , pp. 234-242
    • Mansbach, R.S.1    Chambers, L.K.2    Rovetti, C.C.3
  • 21
    • 29944435424 scopus 로고    scopus 로고
    • 2 acetylcholine receptor partial agonist, in vivo and in vitro
    • 2 acetylcholine receptor partial agonist, in vivo and in vitro, Drug Metab. Dispos., 34(1), 121-130, 2006.
    • (2006) Drug Metab. Dispos , vol.34 , Issue.1 , pp. 121-130
    • Obach, R.S.1
  • 24
    • 85056954575 scopus 로고    scopus 로고
    • 2 nicotinic receptor partial agonist: Results from a 7-week, randomized, placebo-and bupropion-controlled trial with one-year follow-up
    • press
    • 2 nicotinic receptor partial agonist: results from a 7-week, randomized, placebo-and bupropion-controlled trial with one-year follow-up, Arch. Intern. Med., in press.
    • Arch. Intern. Med.
    • Nides, M.1    Oncken, C.2    Gonzales, D.3    Rennard, S.4    Anziano, R.5
  • 26
    • 85056981754 scopus 로고    scopus 로고
    • 2 nicotinic receptor partial agonist-results from varenicline in cessation therapy: Optimizing results
    • Dallas, TX
    • 2 nicotinic receptor partial agonist-results from varenicline in cessation therapy: optimizing results, in Proc. of the American Heart Association Annual Meeting, Dallas, TX, 2005.
    • (2005) Proc. of the American Heart Association Annual Meeting
    • Tonstad, S.1


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