One-pot synthesis of 5-carboxanilide-dihydropyrimidinones using etidronic Acid

Arkivoc

Volumn 2009, Issue 7, 2009, Pages 79-85

  Pansuriya, Akshay M ^a   Savant, Mahesh M ^a   Bhuva, Chirag V ^a   Singh, Jyoti ^a   Naliapara, Yogesh T ^a  

^a SAURASHTRA UNIVERSITY   (India)

Author keywords

5 carboxanilide dihydropyrimidinones; Biginelli reaction; Cyclocondensation; Etidronic acid; Excellent yields

Indexed keywords

EID: 67651175956     PISSN: 1551-7012     EISSN: 15517012     Source Type: Journal    
DOI: None     Document Type: Article

References (20)

1. Kappe, C. O. Tetrahedron 1993, 49, 6937.
2. Rovnyak, G. C.; Atwal, K. S.; Hedberg, A.; Kimball, S. D.; Moreland, S.; Gougoutas, J. Z.; O'Reilly, B. C.; Schwartz, J.; Malley, M. F. J. Med. Chem. 1992, 35, 3254.
3. Khania, E. L.; Sillinietse, G. O.; Ya.Ya. Ozel,; Dabur, G.; Yakimenis, A. A. Khim. Pharm Zh. 1978, 12, 1321.
4. Cho, H.; Ueda, M.; Shima, K.; Mizuno, A.; Hayashimatsu, M.; Ohnaka, Y.; Takeuchi, Y.; Hamaguchi, M.; Aisaka, K.; Hidaka, T. J. Med. Chem. 1989, 32, 2399.
5. Varma, R. S. Green Chem. 1999, 1, 43.
6. Rovnyak, G. C.; Kimball, S. D.; Beyer, B.; Cucinotta, G.; DiMarco, J. D.; Gougoutas, J.; Hedberg, A.; Malley, M.; McCarthy, J. P.; Zhang, R. J. Med. Chem. 1995, 38, 119.
7. Loupy, A.; Petit, A.; Hamelin, J.; Texier-Boullet, F.; Jacquault, P.; Mathe, D. Synthesis 1998, 9, 1213.
8. Atwal, K. S.; Swanson, B. N.; Unger, S. E.; Floyd, D. M.; Moreland, S.; Hedberg, A.; O'Reilly, B. C. J. Med. Chem. 1991, 34, 806.
9. Rovnyak, G. C.; Atwal, K. S.; Hedberg, A.; Kimball, S. D.; Moreland, S.; Gougoutas, J. Z.; O'Reilly, B. C.; Schwartz, J.; Malley, M. F. J. Med. Chem. 1992, 35, 3254.
10. Grover, G. J.; Dzwonczyk, S.; McMullen, D. M.; Normandin, D. E.; Parham, C. S.; Sleph, P. G.; Moreland, S. Cardiovasc. Pharmacol. 1995, 26, 289.
11. Kappe, C. O.; Falsone, F. S. Synlett 1998, 7, 718.
12. Bose, A. K.; Banik, B. K.; Lavlinskaia, N.; Jayaraman, M.; Manhas, M. S. Chemtech 1997, 27, 18.
13. Yarim, M,; Sarac, S.; Ertan, M.; Batu, O.; Erol, K. Farmaco 1999, 54, 359.
14. Foroughifar, N.; Mobinikhaledi, A. Asian J. Chem. 2002, 14, 614.
15. Bruce, M. A.; Poindexter, G. S.; Johnson, G. PCT Int. WO 9833791.Hu, E. H.; Sidler, D. R.; Dolling, U. H. J. Org. Chem. 1998, 63, 3454.
16. Yadav, J. S.; Subba, B. V.; Reddy, S. Srinivas, R.; Venugopal, C.; Ramalingam, T. Synthesis 2001, 9, 1341.
17. Srinivas, K. V. N. S.; Das, B. Synthesis 2004, 13, 2091.
18. Falsone, F. S.; Kappe, C. O. Arkivoc 2001, (ii), 122.
19. The Merck Index, An Encyclopedia of Chemicals, Drugs and Biologicals, 13thed., 2001, p 683.
20. Dixon, L. A. In Encyclopedia of Reagents for Organic Synthesis; Paquette, L., Ed.; Wiley: Chichester, 1995; Vol. 6, pp 4166-4169.