메뉴 건너뛰기




Volumn 26, Issue 7, 2009, Pages 1607-1617

Gastric emptying of pellets under fasting conditions: A mathematical model

Author keywords

Drug dissolution; Gastric emptying; Mathematical models; Multiparticulate systems; Pellets

Indexed keywords

ARTICLE; CONTROLLED STUDY; DIET RESTRICTION; DRUG FORMULATION; GAMMA SCINTIGRAPHY; MATHEMATICAL MODEL; PRIORITY JOURNAL; STOMACH EMPTYING;

EID: 67349272853     PISSN: 07248741     EISSN: 1573904X     Source Type: Journal    
DOI: 10.1007/s11095-009-9869-3     Document Type: Article
Times cited : (36)

References (40)
  • 1
    • 0035293050 scopus 로고    scopus 로고
    • The role of gamma-scintigraphy in oral drug delivery
    • 10.1016/S0169-409X(00)00135-6
    • I. R. Wilding A. J. Coupe S. S. Davis 2001 The role of gamma-scintigraphy in oral drug delivery Adv. Drug. Deliv. Rev. 46 103 124 10.1016/S0169-409X(00) 00135-6
    • (2001) Adv. Drug. Deliv. Rev. , vol.46 , pp. 103-124
    • Wilding, I.R.1    Coupe, A.J.2    Davis, S.S.3
  • 3
    • 0026608368 scopus 로고
    • Biopharmaceutical comparison of oral multiple-unit and single-unit sustained-release dosage forms
    • N. Follonier E. Doelker 1992 Biopharmaceutical comparison of oral multiple-unit and single-unit sustained-release dosage forms S.T.P. Pharma. Sci. 2 141 158
    • (1992) S.T.P. Pharma. Sci. , vol.2 , pp. 141-158
    • Follonier, N.1    Doelker, E.2
  • 7
    • 8744307994 scopus 로고    scopus 로고
    • Multimodel inference-understanding AIC and BIC in model selection
    • 10.1177/0049124104268644
    • K. P. Burnham D. R. Anderson 2004 Multimodel inference-understanding AIC and BIC in model selection Sociol. Method. Res. 33 261 304 10.1177/ 0049124104268644
    • (2004) Sociol. Method. Res. , vol.33 , pp. 261-304
    • Burnham, K.P.1    Anderson, D.R.2
  • 8
    • 0028925905 scopus 로고
    • The description of the gastrointestinal transit of pellets assessed by gamma scintigraphy using statistical moments
    • 10.1023/A:1016200501563
    • F. Podczeck J. M. Newton K. H. Yuen 1995 The description of the gastrointestinal transit of pellets assessed by gamma scintigraphy using statistical moments Pharm. Res. 12 376 379 10.1023/A:1016200501563
    • (1995) Pharm. Res. , vol.12 , pp. 376-379
    • Podczeck, F.1    Newton, J.M.2    Yuen, K.H.3
  • 9
    • 0027240705 scopus 로고
    • Gastrointestinal transit and absorption of theophylline from a multiparticulate controlled-release formulation
    • 10.1016/0378-5173(93)90127-2
    • K. H. Yuen A. A. Deshmukh J. M. Newton M. Short R. Melchor 1993 Gastrointestinal transit and absorption of theophylline from a multiparticulate controlled-release formulation Int. J. Pharm. 97 61 77 10.1016/0378-5173(93) 90127-2
    • (1993) Int. J. Pharm. , vol.97 , pp. 61-77
    • Yuen, K.H.1    Deshmukh, A.A.2    Newton, J.M.3    Short, M.4    Melchor, R.5
  • 10
    • 0742269696 scopus 로고    scopus 로고
    • The use of formulation technology to assess regional gastrointestinal drug absorption in humans
    • 10.1016/j.ejps.2003.10.003
    • A. W. Basit F. Podczeck J. M. Newton W. A. Waddington P. J. Ell L. F. Lacey 2004 The use of formulation technology to assess regional gastrointestinal drug absorption in humans Eur. J. Pharm. Sci. 21 179 189 10.1016/j.ejps.2003. 10.003
    • (2004) Eur. J. Pharm. Sci. , vol.21 , pp. 179-189
    • Basit, A.W.1    Podczeck, F.2    Newton, J.M.3    Waddington, W.A.4    Ell, P.J.5    Lacey, L.F.6
  • 11
    • 0027431325 scopus 로고
    • Gastrointestinal transit of pellets of differing size and density
    • 10.1016/0378-5173(93)90078-T
    • G. M. Clarke J. M. Newton M. D. Short 1993 Gastrointestinal transit of pellets of differing size and density Int. J. Pharm. 100 81 92 10.1016/0378-5173(93)90078-T
    • (1993) Int. J. Pharm. , vol.100 , pp. 81-92
    • Clarke, G.M.1    Newton, J.M.2    Short, M.D.3
  • 12
    • 0028924730 scopus 로고
    • Comparative gastrointestinal transit of pellet systems of varying density
    • 10.1016/0378-5173(94)00200-O
    • G. M. Clarke J. M. Newton M. B. Short 1995 Comparative gastrointestinal transit of pellet systems of varying density Int. J. Pharm. 114 1 11 10.1016/0378-5173(94)00200-O
    • (1995) Int. J. Pharm. , vol.114 , pp. 1-11
    • Clarke, G.M.1    Newton, J.M.2    Short, M.B.3
  • 13
    • 0019945345 scopus 로고
    • The gastric-emptying of pellets contained in hard gelatin capsules
    • 10.3109/03639048209042700
    • E. Hunter J. T. Fell H. Sharma 1982 The gastric-emptying of pellets contained in hard gelatin capsules Drug Dev. Ind. Pharm. 8 751 757 10.3109/03639048209042700
    • (1982) Drug Dev. Ind. Pharm. , vol.8 , pp. 751-757
    • Hunter, E.1    Fell, J.T.2    Sharma, H.3
  • 14
    • 0023119830 scopus 로고
    • The effect of polycarbophil on the gastric emptying of pellets
    • R. Khosla S. S. Davis 1987 The effect of polycarbophil on the gastric emptying of pellets J. Pharm. Pharmacol. 39 47 49
    • (1987) J. Pharm. Pharmacol. , vol.39 , pp. 47-49
    • Khosla, R.1    Davis, S.S.2
  • 15
    • 24844460867 scopus 로고
    • The gastric emptying of pellets in supine volunteers
    • R. Khosla S. S. Davis 1986 The gastric emptying of pellets in supine volunteers J. Pharm. Pharmacol. 38 P10
    • (1986) J. Pharm. Pharmacol. , vol.38 , pp. 10
    • Khosla, R.1    Davis, S.S.2
  • 16
    • 0021942207 scopus 로고
    • Validity of the geometric mean correction in the quantification of whole bowel transit
    • 10.1097/00006231-198504000-00005
    • J. G. Hardy A. C. Perkins 1985 Validity of the geometric mean correction in the quantification of whole bowel transit Nucl. Med. Commun. 6 217 224 10.1097/00006231-198504000-00005
    • (1985) Nucl. Med. Commun. , vol.6 , pp. 217-224
    • Hardy, J.G.1    Perkins, A.C.2
  • 18
    • 0025042445 scopus 로고
    • The influence of density on the gastrointestinal transit of pellets
    • J. E. Devereux J. M. Newton M. B. Short 1990 The influence of density on the gastrointestinal transit of pellets J. Pharm. Pharmacol. 42 500 501
    • (1990) J. Pharm. Pharmacol. , vol.42 , pp. 500-501
    • Devereux, J.E.1    Newton, J.M.2    Short, M.B.3
  • 19
    • 0034812650 scopus 로고    scopus 로고
    • The effect of polyethylene glycol 400 on gastrointestinal transit: Implications for the formulation of poorly-water soluble drugs
    • 10.1023/A:1010927026837
    • A. W. Basit J. M. Newton M. D. Short W. A. Waddington P. J. Ell L. F. Lacey 2001 The effect of polyethylene glycol 400 on gastrointestinal transit: implications for the formulation of poorly-water soluble drugs Pharm. Res. 18 1146 1150 10.1023/A:1010927026837
    • (2001) Pharm. Res. , vol.18 , pp. 1146-1150
    • Basit, A.W.1    Newton, J.M.2    Short, M.D.3    Waddington, W.A.4    Ell, P.J.5    Lacey, L.F.6
  • 20
    • 0025955683 scopus 로고
    • Scintigraphic and pharmacokinetic assessment of a multiparticulate sustained-release formulation of diltiazem
    • 10.1016/0378-5173(91)90351-N
    • I. R. Wilding J. G. Hardy M. Maccari V. Ravelli S. S. Davis 1991 Scintigraphic and pharmacokinetic assessment of a multiparticulate sustained-release formulation of diltiazem Int. J. Pharm. 76 133 143 10.1016/0378-5173(91)90351-N
    • (1991) Int. J. Pharm. , vol.76 , pp. 133-143
    • Wilding, I.R.1    Hardy, J.G.2    MacCari, M.3    Ravelli, V.4    Davis, S.S.5
  • 21
    • 3142756641 scopus 로고    scopus 로고
    • Effect of ethanol and some alcoholic beverages on gastric emptying in humans
    • 10.1080/00365520410005009
    • A. Franke S. Teyssen H. Harder M. V. Singer 2004 Effect of ethanol and some alcoholic beverages on gastric emptying in humans Scand. J. Gastroentero. 39 638 644 10.1080/00365520410005009
    • (2004) Scand. J. Gastroentero. , vol.39 , pp. 638-644
    • Franke, A.1    Teyssen, S.2    Harder, H.3    Singer, M.V.4
  • 22
    • 0026465629 scopus 로고
    • Gamma scintigraphy in the evaluation of pharmaceutical dosage forms
    • 10.1007/BF00175865
    • S. S. Davis J. G. Hardy S. P. Newman I. R. Wilding 1992 Gamma scintigraphy in the evaluation of pharmaceutical dosage forms Eur. J. Nucl. Med. 19 971 986 10.1007/BF00175865
    • (1992) Eur. J. Nucl. Med. , vol.19 , pp. 971-986
    • Davis, S.S.1    Hardy, J.G.2    Newman, S.P.3    Wilding, I.R.4
  • 23
    • 0022538998 scopus 로고
    • Transit of pharmaceutical dosage forms through the small-intestine
    • 10.1136/gut.27.8.886
    • S. S. Davis J. G. Hardy J. W. Fara 1986 Transit of pharmaceutical dosage forms through the small-intestine Gut 27 886 892 10.1136/gut.27.8.886
    • (1986) Gut , vol.27 , pp. 886-892
    • Davis, S.S.1    Hardy, J.G.2    Fara, J.W.3
  • 25
    • 0026639299 scopus 로고
    • The effect of food on the in vivo behaviour of a novel sustained release formulation of tiaprofenic acid
    • 10.1016/0378-5173(82)90018-7
    • I. R. Wilding S. S. Davis R. A. Sparrow J. R. Bloor G. Hayes G. T. Ward 1992 The effect of food on the in vivo behaviour of a novel sustained release formulation of tiaprofenic acid Int. J. Pharm. 83 155 161 10.1016/0378-5173(82) 90018-7
    • (1992) Int. J. Pharm. , vol.83 , pp. 155-161
    • Wilding, I.R.1    Davis, S.S.2    Sparrow, R.A.3    Bloor, J.R.4    Hayes, G.5    Ward, G.T.6
  • 26
    • 0028902712 scopus 로고
    • The effect of food on the gastrointestinal transit and systemic absorption of naproxen from a novel sustained-release formulation
    • 10.1016/0168-3659(94)00118-E
    • C. J. Kenyon G. Hooper D. Tierney J. Butler J. Devane I. R. Wilding 1995 The effect of food on the gastrointestinal transit and systemic absorption of naproxen from a novel sustained-release formulation J. Control. Release 34 31 36 10.1016/0168-3659(94)00118-E
    • (1995) J. Control. Release , vol.34 , pp. 31-36
    • Kenyon, C.J.1    Hooper, G.2    Tierney, D.3    Butler, J.4    Devane, J.5    Wilding, I.R.6
  • 27
    • 0021205310 scopus 로고
    • A comparative-study of the gastrointestinal transit of a pellet and tablet formulation
    • 10.1016/0378-5173(84)90091-7
    • S. S. Davis J. G. Hardy M. J. Taylor D. R. Whalley C. G. Wilson 1984 A comparative-study of the gastrointestinal transit of a pellet and tablet formulation Int. J. Pharm. 21 167 177 10.1016/0378-5173(84)90091-7
    • (1984) Int. J. Pharm. , vol.21 , pp. 167-177
    • Davis, S.S.1    Hardy, J.G.2    Taylor, M.J.3    Whalley, D.R.4    Wilson, C.G.5
  • 28
    • 0022368324 scopus 로고
    • The design and evaluation of controlled release systems for the gastrointestinal tract
    • 10.1016/0168-3659(85)90030-6
    • S. S. Davis 1985 The design and evaluation of controlled release systems for the gastrointestinal tract J. Control. Release 2 27 38 10.1016/0168-3659(85) 90030-6
    • (1985) J. Control. Release , vol.2 , pp. 27-38
    • Davis, S.S.1
  • 30
    • 0032103558 scopus 로고    scopus 로고
    • Gamma scintigraphy: An evolving technology in pharmaceutical formulation development-Part 1
    • 10.1016/S1461-5347(98)00032-7
    • G. A. Digenis E. P. Sandefer R. C. Page W. J. Doll 1998 Gamma scintigraphy: an evolving technology in pharmaceutical formulation development-Part 1 Pharm. Sci. Technol. To. 1 100 107 10.1016/S1461-5347(98) 00032-7
    • (1998) Pharm. Sci. Technol. To. , vol.1 , pp. 100-107
    • Digenis, G.A.1    Sandefer, E.P.2    Page, R.C.3    Doll, W.J.4
  • 31
    • 0025233550 scopus 로고
    • Plasma-concentrations of remoxipride and the gastrointestinal transit of In-111-marked extended-release coated spheres
    • 10.1023/A:1015835609333
    • C. Graffner Z. Wagner M. I. Nilsson E. Widerlov 1990 Plasma- concentrations of remoxipride and the gastrointestinal transit of In-111-marked extended-release coated spheres Pharm. Res. 7 54 58 10.1023/A:1015835609333
    • (1990) Pharm. Res. , vol.7 , pp. 54-58
    • Graffner, C.1    Wagner, Z.2    Nilsson, M.I.3    Widerlov, E.4
  • 34
    • 0029056182 scopus 로고
    • Evaluation of the gastric behavior of coevaporate particles under fasting and nonfasting conditions
    • 10.1016/0378-5173(95)00087-Y
    • D. B. Beten B. Vangansbeke A. Schoutens A. J. Moës 1995 Evaluation of the gastric behavior of coevaporate particles under fasting and nonfasting conditions Int. J. Pharm. 123 145 147 10.1016/0378-5173(95)00087-Y
    • (1995) Int. J. Pharm. , vol.123 , pp. 145-147
    • Beten, D.B.1    Vangansbeke, B.2    Schoutens, A.3    Moës, A.J.4
  • 35
    • 0021092176 scopus 로고
    • The gastric-emptying of hard gelatin capsules
    • 10.1016/0378-5173(83)90018-2
    • E. Hunter J. T. Fell H. Sharma 1983 The gastric-emptying of hard gelatin capsules Int. J. Pharm. 17 59 64 10.1016/0378-5173(83)90018-2
    • (1983) Int. J. Pharm. , vol.17 , pp. 59-64
    • Hunter, E.1    Fell, J.T.2    Sharma, H.3
  • 36
    • 0028895436 scopus 로고
    • Pharmacoscintigraphic evaluation of a modified release Geomatrix(R) diltiazem formulation
    • 10.1016/0168-3659(94)00066-4
    • I. R. Wilding S. S. Davis R. A. Sparrow J. A. Ziemniak D. L. Heald 1995 Pharmacoscintigraphic evaluation of a modified release Geomatrix(R) diltiazem formulation J. Control. Release 33 89 97 10.1016/0168-3659(94)00066-4
    • (1995) J. Control. Release , vol.33 , pp. 89-97
    • Wilding, I.R.1    Davis, S.S.2    Sparrow, R.A.3    Ziemniak, J.A.4    Heald, D.L.5
  • 37
    • 0033983223 scopus 로고    scopus 로고
    • Gastrointestinal spread of oral prolonged-release mesalazine microgranules (Pentasa) dosed as either tablets or sachet
    • 10.1046/j.1365-2036.2000.00696.x
    • I. R. Wilding C. J. Kenyon G. Hooper 2000 Gastrointestinal spread of oral prolonged-release mesalazine microgranules (Pentasa) dosed as either tablets or sachet Aliment. Pharmacol. Ther. 14 163 169 10.1046/j.1365-2036.2000.00696.x
    • (2000) Aliment. Pharmacol. Ther. , vol.14 , pp. 163-169
    • Wilding, I.R.1    Kenyon, C.J.2    Hooper, G.3
  • 38
    • 0037514407 scopus 로고    scopus 로고
    • Combined scintigraphic and pharmacokinetic investigation of enteric-coated mesalazine micropellets in healthy subjects
    • 10.1046/j.1365-2036.2003.01558.x
    • I. R. Wilding C. Behrens S. J. Tardif H. Wray P. Bias W. Albrecht 2003 Combined scintigraphic and pharmacokinetic investigation of enteric-coated mesalazine micropellets in healthy subjects Aliment. Pharmacol. Ther. 17 1153 1162 10.1046/j.1365-2036.2003.01558.x
    • (2003) Aliment. Pharmacol. Ther. , vol.17 , pp. 1153-1162
    • Wilding, I.R.1    Behrens, C.2    Tardif, S.J.3    Wray, H.4    Bias, P.5    Albrecht, W.6
  • 39
    • 0038528399 scopus 로고    scopus 로고
    • Gastrointestinal transit and release of 5-aminosalicylic acid from Sm-153-labelled mesalazine pellets vs. tablets in male healthy volunteers
    • 10.1046/j.1365-2036.2003.01564.x
    • M. Brunner R. Greinwald K. Kletter H. Kvaternik M. E. Corrado H. G. Eichler M. Müller 2003 Gastrointestinal transit and release of 5-aminosalicylic acid from Sm-153-labelled mesalazine pellets vs. tablets in male healthy volunteers Aliment. Pharmacol. Ther. 17 1163 1169 10.1046/j.1365-2036.2003.01564.x
    • (2003) Aliment. Pharmacol. Ther. , vol.17 , pp. 1163-1169
    • Brunner, M.1    Greinwald, R.2    Kletter, K.3    Kvaternik, H.4    Corrado, M.E.5    Eichler, H.G.6    Müller, M.7
  • 40
    • 34447312456 scopus 로고    scopus 로고
    • Gastrointestinal transit of model mini-tablet controlled release oral dosage forms in fasted human volunteers
    • 10.1211/jpp.59.7.0005
    • F. Podczeck N. Course J. M. Newton M. B. Short 2007 Gastrointestinal transit of model mini-tablet controlled release oral dosage forms in fasted human volunteers J. Pharm. Pharmacol. 59 941 945 10.1211/jpp.59.7.0005
    • (2007) J. Pharm. Pharmacol. , vol.59 , pp. 941-945
    • Podczeck, F.1    Course, N.2    Newton, J.M.3    Short, M.B.4


* 이 정보는 Elsevier사의 SCOPUS DB에서 KISTI가 분석하여 추출한 것입니다.