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Bioorganic and Medicinal Chemistry Letters

Volumn 19, Issue 13, 2009, Pages 3651-3656

Non-isotopic dual parameter competition assay suitable for high-throughput screening of histone deacetylases

(7) Riester, Daniel a Hildmann, Christian b Haus, Patricia c Galetovic, Antonia c Schober, Andreas b Schwienhorst, Andreas a Meyer Almes, Franz Josef c

a UNIVERSITY OF GÖTTINGEN (Germany)

b ILMENAU UNIVERSITY OF TECHNOLOGY (Germany)

c DARMSTADT UNIVERSITY OF APPLIED SCIENCES (Germany)

Author keywords

Competition assay; Fluorogenic substrates; FRET; High throughput screening assay; Histone deacetylase

Indexed keywords

1 (3 CARBOXYPROPYL) 11 ETHYL 2,2,8,10,10 PENTAMETHYL 4 (SULFOMETHYL) 2,10 DIHYDRO 1H 13 OXA 1,6,11 TRIAZAPENTACEN 11 IUM; 7 AMINO 4 METHYLCOUMARIN; APICIDIN; COUMARIN DERIVATIVE; FLUORESCENT DYE; HISTONE DEACETYLASE 6; HISTONE DEACETYLASE INHIBITOR; HYDROXAMIC ACID; N (2 AMINOPHENYL) 4 (3 PYRIDINYLMETHOXYCARBONYLAMINOMETHYL)BENZAMIDE; TRICHOSTATIN A; UNCLASSIFIED DRUG; VORINOSTAT;

ANISOTROPY; ARTICLE; ASSAY; CHEMICAL STRUCTURE; COMPETITIVE INHIBITION; ENZYME BINDING; FLUORESCENCE; FLUORESCENCE LIFETIME; FLUORESCENCE POLARIZATION; HIGH THROUGHPUT SCREENING; MOLECULAR PROBE; NON ISOTOPIC DUAL PARAMETER COMPETITION ASSAY; NONHUMAN;

DRUG EVALUATION, PRECLINICAL; ENZYME INHIBITORS; FLUORESCENCE RESONANCE ENERGY TRANSFER; FLUORESCENT DYES; HISTONE DEACETYLASES;

EID: 66349116979 PISSN: 0960894X EISSN: None Source Type: Journal
DOI: 10.1016/j.bmcl.2009.04.102 Document Type: Article

Times cited : (18)

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