Rapid synthesis of imidazo[4,5-b]pyridine containing polycyclics by means of palladium-catalyzed amidation of 2-chloro-3-nitropyridine

Tetrahedron Letters

Volumn 50, Issue 27, 2009, Pages 3798-3800

  Salomé, Christophe ^a   Schmitt, Martine ^a   Bourguignon, Jean Jacques ^a  

^a Faculté de Pharmacie   (France)

Author keywords

[No Author keywords available]

Indexed keywords

2 CHLORO 3 NITROPYRIDINE; AMIDE; HYPOCHLORITE SODIUM; IMIDAZO[4,5 B]PYRIDINE DERIVATIVE; PALLADIUM; PYRIDINE DERIVATIVE; UNCLASSIFIED DRUG;

ACYLATION; AMIDATION; ARTICLE; BUCHWALD REACTION; CATALYSIS; CHEMICAL REACTION; CHEMICAL STRUCTURE; SYNTHESIS;

EID: 65549154214     PISSN: 00404039     EISSN: None     Source Type: Journal    
DOI: 10.1016/j.tetlet.2009.04.031     Document Type: Article

References (13)

1. Arvanitis A., Rescinito J.T., Arnold C.R., Wilde R.G., Cain G.A., Sun J.H., Yan J.-S., Teleha C.A., Fitzgerald L.W., McElroy J., Zaczek R., Hartig P.R., Grossman S., Arneric S.P., Gilligan P.J., Olson R.E., and Robertson D.W. Bioorg. Med. Chem. Lett. 13 (2003) 125-128
2. Janssens F., Torremans J., Janssen M., Stokbroekx R., Luyckx M., and Janssen P. J. Med. Chem. 28 (1985) 1943-1947
3. Chang L.C.W., von Frijtag Drabbe Kunzel J.K., Mulder-Krieger T., Westerhout J., Spangenberg T., Brussee J., and IJzerman A.P. J. Med. Chem. 50 (2007) 828-834
4. Désaubry L., Wermuth C., and Bourguignon J.-J. Tetrahedron Lett. 36 (1995) 4249-4252
5. Yin J., and Buchwald S.L. J. Am. Chem. Soc. 124 (2002) 6043-6048
6. Klapars A., Huang X., and Buchwald S.L. J. Am. Chem. Soc. 124 (2002) 7421-7428
7. Zheng N., and Buchwald S.L. Org. Lett. 9 (2007) 4749-4751
8. Sugahara M., and Ukita T. Chem. Pharm. Bull. 45 (1997) 719
9. + requires 223.0).
10. Yin J., and Buchwald S.L. Org. Lett. 2 8 (2000) 1101-1104
11. + requires 299.0780).
12. + requires 265.29).
13. Loones K.T.J., Maes B.U.W., Dommisse R.A., and Lemière G. Chem. Commun. (2004) 2466-2467