Labelling, purification, and receptor affinity of radioactive iododiethylstilbestrol (*I-DES) with high specific activity and first structure analysis with natI-DES

Journal of Labelled Compounds and Radiopharmaceuticals

Volumn 47, Issue 10, 2004, Pages 669-678

  Fischer, Thomas ^a   Schomäcker, Klaus ^a   Schicha, Harald ^a  

^a UNIVERSITY OF COLOGNE   (Germany)

Author keywords

Diethylstilbestrol; Estrogen; High specific activity; Mamma carcinoma; NMR; Radioiodine

Indexed keywords

AUGER ELECTRON SPECTROSCOPY;

DIETHYLSTILBESTROL; ESTROGEN RECEPTOR; HIGH AFFINITY; HIGH SPECIFIC ACTIVITIES; LABELINGS; MAMMA CARCINOMA; OESTROGENS; RADIOIODINE; STEROIDAL ESTROGENS; STRUCTURE ANALYSIS;

DISSOCIATION;

1 CHLORO 1 (4' HYDROXYPHENYL)PROPENE; 4 TOLUOLSULFONIC ACID AMIDE; CHLORMETHINE; DIETHYLSTILBESTROL; DIETHYLSTILBESTROL BR 77; DIETHYLSTILBESTROL I 125; ESTRADIOL I 125; ESTROGEN; ESTROGEN RECEPTOR; IODINE; IODODIETHYLSTILBESTROL; RADIOPHARMACEUTICAL AGENT; TOLUENESULFONIC ACID DERIVATIVE; UNCLASSIFIED DRUG;

ARTICLE; AUGER ELECTRON SPECTROSCOPY; BINDING AFFINITY; BREAST TUMOR; CARBON NUCLEAR MAGNETIC RESONANCE; CHEMICAL STRUCTURE; COMPARATIVE STUDY; DISSOCIATION CONSTANT; DRUG ACTIVITY; DRUG PURIFICATION; ISOTOPE LABELING; PROTON NUCLEAR MAGNETIC RESONANCE; RADIOCHEMISTRY; RADIOIODINATION; RECEPTOR AFFINITY; REVERSED PHASE HIGH PERFORMANCE LIQUID CHROMATOGRAPHY; SCATCHARD PLOT; STRUCTURE ANALYSIS;

EID: 6344279798     PISSN: 03624803     EISSN: None     Source Type: Journal    
DOI: 10.1002/jlcr.853     Document Type: Article

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