메뉴 건너뛰기




Volumn 16, Issue 2, 2009, Pages 82-91

A combined approach of chemical enhancers and sonophoresis for the transdermal delivery of tizanidine hydrochloride

Author keywords

Chemical enhancer; Skin permeation; Sonophoresis; Tizanidine; Transdermal

Indexed keywords

1 METHYL 2 PYRROLIDINONE; ALCOHOL; CINEOLE; CITRAL; DIETHYLENE GLYCOL MONOETHYL ETHER; DIMETHYL SULFOXIDE; LIMONENE; MYRISTIC ACID ISOPROPYL ESTER; OLEIC ACID; PENETRATION ENHANCING AGENT; POLYSORBATE 80; PROPYLENE GLYCOL; TIZANIDINE; TRIACETIN;

EID: 62249216550     PISSN: 10717544     EISSN: 15210464     Source Type: Journal    
DOI: 10.1080/10717540802605053     Document Type: Article
Times cited : (57)

References (55)
  • 1
    • 0030793498 scopus 로고    scopus 로고
    • Transdermal delivery of drugs
    • Panchagnula R. (1997). Transdermal delivery of drugs. Indian J Pharmacol, 29, 140-56.
    • (1997) Indian J Pharmacol , vol.29 , pp. 140-156
    • Panchagnula, R.1
  • 3
    • 0002855088 scopus 로고    scopus 로고
    • Phonophoresis
    • Bronaugh RL, Maibach HI, eds, 3rd ed. Boca Raton: Taylor & Francis
    • Kost J, Mitragotri S, Langer R. (1999). Phonophoresis. In: Bronaugh RL, Maibach HI, eds. Percutaneous Absorption, 3rd ed. Boca Raton: Taylor & Francis, 615-31.
    • (1999) Percutaneous Absorption , pp. 615-631
    • Kost, J.1    Mitragotri, S.2    Langer, R.3
  • 4
    • 0035965516 scopus 로고    scopus 로고
    • Comparison of the effect of ultrasound and of chemical enhancers on transdermal permeation of caffeine and morphine through hairless mouse skin in vitro
    • Monti D, Giannelli R, Chetoni P, Burgalassi S. (2001). Comparison of the effect of ultrasound and of chemical enhancers on transdermal permeation of caffeine and morphine through hairless mouse skin in vitro. Int J Pharm, 229, 131-7.
    • (2001) Int J Pharm , vol.229 , pp. 131-137
    • Monti, D.1    Giannelli, R.2    Chetoni, P.3    Burgalassi, S.4
  • 5
    • 0038621994 scopus 로고    scopus 로고
    • Skin permeability enhancement by low frequency sonophoresis: Lipid extraction and transport pathways
    • Alvarez-Román R, Merino G, Kalia YN, Naik A, Guy RH. (2003). Skin permeability enhancement by low frequency sonophoresis: lipid extraction and transport pathways. J Pharm Sci, 6, 1138-46.
    • (2003) J Pharm Sci , vol.6 , pp. 1138-1146
    • Alvarez-Román, R.1    Merino, G.2    Kalia, Y.N.3    Naik, A.4    Guy, R.H.5
  • 6
    • 1542328828 scopus 로고    scopus 로고
    • Low-frequency sonophoresis: A review
    • Mitragotri S, Kost J. (2004). Low-frequency sonophoresis: a review. Adv Drug Deliv Rev, 5, 589-601.
    • (2004) Adv Drug Deliv Rev , vol.5 , pp. 589-601
    • Mitragotri, S.1    Kost, J.2
  • 8
    • 62249131367 scopus 로고    scopus 로고
    • Moffat AC, Osselton MD, Widdop B. (2006). Clarke's analysis of drugs and poisons, 2nd 3rd ed. London: Pharmaceutical Press.
    • Moffat AC, Osselton MD, Widdop B. (2006). Clarke's analysis of drugs and poisons, 2nd Vol., 3rd ed. London: Pharmaceutical Press.
  • 9
    • 62249112644 scopus 로고    scopus 로고
    • Reagents, Indicators and solutions
    • USA: Rockville, MD. The United States pharmacopoeial convention
    • USP-NF. (2006). Reagents, Indicators and solutions. 29th (Asian) edition. USA: Rockville, MD. The United States pharmacopoeial convention, 3167-75.
    • (2006) 29th (Asian) edition , pp. 3167-3175
    • NF, U.1
  • 10
    • 62249092259 scopus 로고    scopus 로고
    • Indian Pharmacopoeia. (1996). Reagents and solutions. Appendix 13, 2, Ministry of Health and Family Welfare. Delhi, India: Government of India, A144-7.
    • Indian Pharmacopoeia. (1996). Reagents and solutions. Appendix 13, Vol 2, Ministry of Health and Family Welfare. Delhi, India: Government of India, A144-7.
  • 11
    • 0034712799 scopus 로고    scopus 로고
    • Influence of cyclodextrin complexation on the in vitro permeation and skin metabolism of dexamethasone
    • Renata FVL, Collet JH, Bentley LB. (2000). Influence of cyclodextrin complexation on the in vitro permeation and skin metabolism of dexamethasone. Int J Pharm, 200, 127-32.
    • (2000) Int J Pharm , vol.200 , pp. 127-132
    • Renata, F.V.L.1    Collet, J.H.2    Bentley, L.B.3
  • 12
    • 0033998781 scopus 로고    scopus 로고
    • Skin permeation of testosterone and its ester derivatives in rats
    • Kim MK, Lee CH, Kim DD. (2000). Skin permeation of testosterone and its ester derivatives in rats. J Pharm Pharmacol, 52, 369-375.
    • (2000) J Pharm Pharmacol , vol.52 , pp. 369-375
    • Kim, M.K.1    Lee, C.H.2    Kim, D.D.3
  • 13
    • 0038784742 scopus 로고    scopus 로고
    • Pharmaceutical preformulation: The physicochemical properties of drug substances
    • Aulton ME, ed, London: Churchill Livingstone
    • Wells J. (2002). Pharmaceutical preformulation: the physicochemical properties of drug substances. In: Aulton ME, ed. Pharmaceutics. London: Churchill Livingstone, 113-51.
    • (2002) Pharmaceutics , pp. 113-151
    • Wells, J.1
  • 14
    • 0026621780 scopus 로고
    • Enhancement effects in the permeation of alprazolam through hairless mouse skin
    • Carelli V, Di Colo G, Nannipieri E, Serafini MF. (1992). Enhancement effects in the permeation of alprazolam through hairless mouse skin. Int J Pharm, 88, 89-97.
    • (1992) Int J Pharm , vol.88 , pp. 89-97
    • Carelli, V.1    Di Colo, G.2    Nannipieri, E.3    Serafini, M.F.4
  • 15
    • 0033959861 scopus 로고    scopus 로고
    • Evaluation of transcutol as a clonazepam transdermal permeation enhancer from hydrophilic gel formulations
    • Mura P, Faucci MT, Bramanti G, Corti P. (2000). Evaluation of transcutol as a clonazepam transdermal permeation enhancer from hydrophilic gel formulations. Eur J Pharm Sci, 9, 365-72.
    • (2000) Eur J Pharm Sci , vol.9 , pp. 365-372
    • Mura, P.1    Faucci, M.T.2    Bramanti, G.3    Corti, P.4
  • 16
    • 0030787333 scopus 로고    scopus 로고
    • Mechanism of transdermal transport of 5-fluorouracil by terpenes: Carvone, 1,8-cineole and thymol
    • Gao S, Singh J. (1997). Mechanism of transdermal transport of 5-fluorouracil by terpenes: carvone, 1,8-cineole and thymol. Int J Pharm, 154, 67-77.
    • (1997) Int J Pharm , vol.154 , pp. 67-77
    • Gao, S.1    Singh, J.2
  • 17
    • 18044397839 scopus 로고    scopus 로고
    • Effect of penetration enhancers on the transdermal delivery of bupranolol through rat skin
    • Babu RJ, Pandit JK. (2005). Effect of penetration enhancers on the transdermal delivery of bupranolol through rat skin. Drug Deliv, 3, 165-9.
    • (2005) Drug Deliv , vol.3 , pp. 165-169
    • Babu, R.J.1    Pandit, J.K.2
  • 18
    • 0036141739 scopus 로고    scopus 로고
    • Synergistic effect of low-frequency ultrasound and surfactants on skin permeability
    • Tezel A, Sens A, Tuchscherer J, Mitragotri S. (2002). Synergistic effect of low-frequency ultrasound and surfactants on skin permeability. J Pharm Sci, 1, 91-100.
    • (2002) J Pharm Sci , vol.1 , pp. 91-100
    • Tezel, A.1    Sens, A.2    Tuchscherer, J.3    Mitragotri, S.4
  • 19
    • 0037436014 scopus 로고    scopus 로고
    • Frequency and thermal effects on the enhancement of transdermal transport by sonophoresis
    • Merino G, Kalia YN, Delgado-Charro MB, Potts RO, Guy RH. (2003). Frequency and thermal effects on the enhancement of transdermal transport by sonophoresis. J Contr Rel, 88, 85-94.
    • (2003) J Contr Rel , vol.88 , pp. 85-94
    • Merino, G.1    Kalia, Y.N.2    Delgado-Charro, M.B.3    Potts, R.O.4    Guy, R.H.5
  • 22
    • 0036587703 scopus 로고    scopus 로고
    • Effect of the solvent system on the in vitro permeability of nicardipine hydrochloride through excised rat epidermis
    • Krishnaiah YS, Satyanarayana V, Karthikeyan RS. (2002). Effect of the solvent system on the in vitro permeability of nicardipine hydrochloride through excised rat epidermis. J Pharm Pharm Sci, 2, 123-30.
    • (2002) J Pharm Pharm Sci , vol.2 , pp. 123-130
    • Krishnaiah, Y.S.1    Satyanarayana, V.2    Karthikeyan, R.S.3
  • 23
    • 0022868189 scopus 로고
    • Influence of solvents on paraben permeation through idealized skin model membranes
    • Twist JN, Zatz JL. (1986). Influence of solvents on paraben permeation through idealized skin model membranes. J Soc Cosmetic Chem, 37, 429-44.
    • (1986) J Soc Cosmetic Chem , vol.37 , pp. 429-444
    • Twist, J.N.1    Zatz, J.L.2
  • 24
    • 0037020515 scopus 로고    scopus 로고
    • Effect of vehicles on the transdermal delivery of melatonin across porcine skin in vitro
    • Kikwai L, Kanikkannan N, Babu RJ, Singh M. (2002). Effect of vehicles on the transdermal delivery of melatonin across porcine skin in vitro. J Contr Rel, 2, 307-11.
    • (2002) J Contr Rel , vol.2 , pp. 307-311
    • Kikwai, L.1    Kanikkannan, N.2    Babu, R.J.3    Singh, M.4
  • 25
    • 34247480143 scopus 로고    scopus 로고
    • Ex-vivo study of transdermal permeation of four diclofenac salts from different vehicles
    • Minghetti P, Cilurzo F, Casiraghi A, Montanari L, Fini A. (2007). Ex-vivo study of transdermal permeation of four diclofenac salts from different vehicles. J Pharm Sci, 4, 814-23.
    • (2007) J Pharm Sci , vol.4 , pp. 814-823
    • Minghetti, P.1    Cilurzo, F.2    Casiraghi, A.3    Montanari, L.4    Fini, A.5
  • 26
    • 0025733949 scopus 로고
    • Development and evaluation of an intracutaneous depot formulation of corticosteroids using Transcutol as a cosolvent: In-vitro, ex-vivo and in-vivo rat studies
    • Panchagnula R, Ritschel WA. (1991). Development and evaluation of an intracutaneous depot formulation of corticosteroids using Transcutol as a cosolvent: in-vitro, ex-vivo and in-vivo rat studies. J Pharm Pharmacol, 9, 609-14.
    • (1991) J Pharm Pharmacol , vol.9 , pp. 609-614
    • Panchagnula, R.1    Ritschel, W.A.2
  • 27
    • 0032821253 scopus 로고    scopus 로고
    • A therapeutic dose of primaquine can be delivered across human skin from simple transdermal patches
    • Jeans CW, Heard CM. (1999). A therapeutic dose of primaquine can be delivered across human skin from simple transdermal patches. Int J Pharm, 189, 1-6.
    • (1999) Int J Pharm , vol.189 , pp. 1-6
    • Jeans, C.W.1    Heard, C.M.2
  • 28
    • 0033812031 scopus 로고    scopus 로고
    • Mechanism(s) of in vitro percutaneous absorption enhancement of tamoxifen by enhancers
    • Zhao K, Singh J. (2000). Mechanism(s) of in vitro percutaneous absorption enhancement of tamoxifen by enhancers. J Pharm Sci, 6, 771-80.
    • (2000) J Pharm Sci , vol.6 , pp. 771-780
    • Zhao, K.1    Singh, J.2
  • 29
    • 0035895235 scopus 로고    scopus 로고
    • Effect of some enhancers on the permeation of haloperidol through rat skin in vitro
    • Vaddi HK, Wang LZ, Ho PC, Chan SY. (2001). Effect of some enhancers on the permeation of haloperidol through rat skin in vitro. Int J Pharm, 212, 247-55.
    • (2001) Int J Pharm , vol.212 , pp. 247-255
    • Vaddi, H.K.1    Wang, L.Z.2    Ho, P.C.3    Chan, S.Y.4
  • 30
    • 0036365893 scopus 로고    scopus 로고
    • In vitro skin permeation of morphine hydrochloride during the finite application of penetration enhancing system containing water, ethanol and l-menthol
    • Morimoto Y, Wada Y, Seki T, Sugibayashi K. (2002). In vitro skin permeation of morphine hydrochloride during the finite application of penetration enhancing system containing water, ethanol and l-menthol. Biol Pharm Bull, 1, 134-6.
    • (2002) Biol Pharm Bull , vol.1 , pp. 134-136
    • Morimoto, Y.1    Wada, Y.2    Seki, T.3    Sugibayashi, K.4
  • 31
    • 0029942121 scopus 로고    scopus 로고
    • Formulation study of a transdermal delivery system of primaquine
    • Mayorga P, Puisieux F, Couarraze G. (1996). Formulation study of a transdermal delivery system of primaquine. Int J Pharm, 132, 71-9.
    • (1996) Int J Pharm , vol.132 , pp. 71-79
    • Mayorga, P.1    Puisieux, F.2    Couarraze, G.3
  • 32
    • 33750507126 scopus 로고    scopus 로고
    • Microemulsions as transdermal drug delivery vehicles
    • Kogan A, Garti N. (2006). Microemulsions as transdermal drug delivery vehicles. Adv Colloid Interface Sci, 123-6, 369-85.
    • (2006) Adv Colloid Interface Sci , vol.123 -6 , pp. 369-385
    • Kogan, A.1    Garti, N.2
  • 33
    • 0036912766 scopus 로고    scopus 로고
    • Transdermal delivery of glibenclamide and glipizide: In vitro permeation studies through mouse skin
    • Mutalik S, Udupa N. (2002). Transdermal delivery of glibenclamide and glipizide: in vitro permeation studies through mouse skin. Pharmazie, 12, 838-41.
    • (2002) Pharmazie , vol.12 , pp. 838-841
    • Mutalik, S.1    Udupa, N.2
  • 34
    • 0345735503 scopus 로고    scopus 로고
    • Effect of some penetration enhancers on the permeation of glibenclamide and glipizide through mouse skin
    • Mutalik S, Udupa N. (2003). Effect of some penetration enhancers on the permeation of glibenclamide and glipizide through mouse skin. Pharmazie, 12, 891-4.
    • (2003) Pharmazie , vol.12 , pp. 891-894
    • Mutalik, S.1    Udupa, N.2
  • 36
    • 0036812998 scopus 로고    scopus 로고
    • Transdermal delivery of nicardipine: An approach to in vitro permeation enhancement
    • Aboofazeli R, Zia H, Needham TE. (2002). Transdermal delivery of nicardipine: an approach to in vitro permeation enhancement. Drug Deliv, 9, 239-47.
    • (2002) Drug Deliv , vol.9 , pp. 239-247
    • Aboofazeli, R.1    Zia, H.2    Needham, T.E.3
  • 37
    • 0036360730 scopus 로고    scopus 로고
    • Formulation optimization and stability study of transdermal therapeutic system of nicorandil
    • Tipre DN, Vavia PR. (2002). Formulation optimization and stability study of transdermal therapeutic system of nicorandil. Pharm Dev Tech, 3, 325-32.
    • (2002) Pharm Dev Tech , vol.3 , pp. 325-332
    • Tipre, D.N.1    Vavia, P.R.2
  • 38
    • 0034988944 scopus 로고    scopus 로고
    • Transdermal absorption of bupranolol in rabbit skin in vitro and in vivo
    • Ogiso T, Hata T, Iwaki M, Tanino T. (2001). Transdermal absorption of bupranolol in rabbit skin in vitro and in vivo. Biol Pharm Bull, 5, 588-91.
    • (2001) Biol Pharm Bull , vol.5 , pp. 588-591
    • Ogiso, T.1    Hata, T.2    Iwaki, M.3    Tanino, T.4
  • 39
    • 27744463374 scopus 로고    scopus 로고
    • Feasibility of transdermal delivery of fluoxetine
    • Parikh DK, Ghosh TK. (2005). Feasibility of transdermal delivery of fluoxetine. AAPS Pharm Sci Tech, 2, E144-9.
    • (2005) AAPS Pharm Sci Tech , vol.2
    • Parikh, D.K.1    Ghosh, T.K.2
  • 41
    • 23144440197 scopus 로고    scopus 로고
    • Suwanpidokkul N, Thongnopnua P, Umprayn K. (2004). Transdermal delivery of zidovudine (AZT): the effects of vehicles, enhancers, and polymer membranes on permeation across cadaver pig skin. AAPS Pharm Sci Tech, 3, Article 48, E1-8.
    • Suwanpidokkul N, Thongnopnua P, Umprayn K. (2004). Transdermal delivery of zidovudine (AZT): the effects of vehicles, enhancers, and polymer membranes on permeation across cadaver pig skin. AAPS Pharm Sci Tech, 3, Article 48, E1-8.
  • 42
    • 0028881228 scopus 로고
    • Transdermal delivery of zalcitabine: In vitro skin permeation study
    • Kim DD, Chien YW. (1995). Transdermal delivery of zalcitabine: in vitro skin permeation study. AIDS, 12, 1331-6.
    • (1995) AIDS , vol.12 , pp. 1331-1336
    • Kim, D.D.1    Chien, Y.W.2
  • 43
    • 0034042520 scopus 로고    scopus 로고
    • Structure-activity relationship of chemical penetration enhancers in transdermal drug delivery
    • Kanikkannan N, Kandimalla K, Lamba SS, Singh M. (2000). Structure-activity relationship of chemical penetration enhancers in transdermal drug delivery. Curr Med Chem, 6, 593-608.
    • (2000) Curr Med Chem , vol.6 , pp. 593-608
    • Kanikkannan, N.1    Kandimalla, K.2    Lamba, S.S.3    Singh, M.4
  • 45
    • 33947606082 scopus 로고    scopus 로고
    • The effect of terpene concentrations on the skin penetration of diclofenac sodium
    • Nokhodchi A, Sharabiani K, Rashidi MR, Ghafourian T. (2007). The effect of terpene concentrations on the skin penetration of diclofenac sodium. Int J Pharm, 335, 97-105.
    • (2007) Int J Pharm , vol.335 , pp. 97-105
    • Nokhodchi, A.1    Sharabiani, K.2    Rashidi, M.R.3    Ghafourian, T.4
  • 46
    • 0025169207 scopus 로고
    • Transdermal delivery of 5-fluorouracil through skin of hairless mice and humans in vitro: A comparison of the effect of formulations and a prodrug
    • Sherertz EF, Sloan KB, McTiernan RG. (1990). Transdermal delivery of 5-fluorouracil through skin of hairless mice and humans in vitro: a comparison of the effect of formulations and a prodrug. Arch Dermatol Res, 282, 463-8.
    • (1990) Arch Dermatol Res , vol.282 , pp. 463-468
    • Sherertz, E.F.1    Sloan, K.B.2    McTiernan, R.G.3
  • 47
    • 0025162194 scopus 로고
    • Transdermal delivery of levonorgestrel VIII. Effect of enhancers on rat skin, hairless mouse skin, hairless guinea pig skin, and human skin
    • Catz P, Friend DR. (1990). Transdermal delivery of levonorgestrel VIII. Effect of enhancers on rat skin, hairless mouse skin, hairless guinea pig skin, and human skin. Int J Pharm, 58, 93-102.
    • (1990) Int J Pharm , vol.58 , pp. 93-102
    • Catz, P.1    Friend, D.R.2
  • 48
    • 0032732922 scopus 로고    scopus 로고
    • Gorukanti SR, Li L, Kim KH. (1999). Transdermal delivery of antiparkinsonian agent, benztropine. I. Effect of vehicles on skin permeation. Int J Pharm, 192, 159-72.
    • Gorukanti SR, Li L, Kim KH. (1999). Transdermal delivery of antiparkinsonian agent, benztropine. I. Effect of vehicles on skin permeation. Int J Pharm, 192, 159-72.
  • 49
    • 0035848413 scopus 로고    scopus 로고
    • In vitro transdermal ion-tophoretic transport of timolol maleate: Effect of age and species
    • Kanikkannan N, Singh J, Ramarao P. (2001). In vitro transdermal ion-tophoretic transport of timolol maleate: effect of age and species. J Contr Rel, 71, 99-105.
    • (2001) J Contr Rel , vol.71 , pp. 99-105
    • Kanikkannan, N.1    Singh, J.2    Ramarao, P.3
  • 50
    • 18944375393 scopus 로고    scopus 로고
    • Low-frequency ultrasound as a transcutaneous immunization adjuvant
    • Tezel A, Paliwal S, Shen Z, Mitragotri S. (2005). Low-frequency ultrasound as a transcutaneous immunization adjuvant. Vaccine, 29, 3800-7.
    • (2005) Vaccine , vol.29 , pp. 3800-3807
    • Tezel, A.1    Paliwal, S.2    Shen, Z.3    Mitragotri, S.4
  • 51
    • 34247507592 scopus 로고    scopus 로고
    • Anaesthetic effects of lidocaine hydrochloride gel using low frequency ultrasound of 0.5 MHz
    • Kim TY, Jung DI, Kim YI, Yang JH, Shin SC. (2007). Anaesthetic effects of lidocaine hydrochloride gel using low frequency ultrasound of 0.5 MHz. J Pharm Sci, 1, 1-8.
    • (2007) J Pharm Sci , vol.1 , pp. 1-8
    • Kim, T.Y.1    Jung, D.I.2    Kim, Y.I.3    Yang, J.H.4    Shin, S.C.5
  • 52
  • 53
    • 1442325314 scopus 로고    scopus 로고
    • Influence of ultrasound on the percutaneous absorption of ketorolac tromethamine in vitro across rat skin
    • Tiwari SB, Pai RM, Udupa N. (2004). Influence of ultrasound on the percutaneous absorption of ketorolac tromethamine in vitro across rat skin. Drug Deliv, 1, 47-51.
    • (2004) Drug Deliv , vol.1 , pp. 47-51
    • Tiwari, S.B.1    Pai, R.M.2    Udupa, N.3
  • 55
    • 0029070955 scopus 로고
    • A mechanistic study of ultrasonically-enhanced transdermal drug delivery
    • Mitragotri S, Edwards DA, Blankschtein D, Langer R. (1995). A mechanistic study of ultrasonically-enhanced transdermal drug delivery. J Pharm Sci, 6, 697-706.
    • (1995) J Pharm Sci , vol.6 , pp. 697-706
    • Mitragotri, S.1    Edwards, D.A.2    Blankschtein, D.3    Langer, R.4


* 이 정보는 Elsevier사의 SCOPUS DB에서 KISTI가 분석하여 추출한 것입니다.